Asymmetric addition of benzothiazole to N-tert-butanesulfinyl imine for the synthesis of chiral alpha-branched heteroaryl amines
文献类型：期刊论文
| 作者 | Zhang, Jinlong1,2; Yang, Yuhong1,2; Wang, Mei1,2; Lin, Li1,2; Wang R(王锐)1,2,3 |
| 刊名 | Tetrahedron Letters
 |
| 出版日期 | 2012 |
| 卷号 | 53期号:51页码:6893-6896 |
| 关键词 | Asymmetric synthesis Benzothiazole Diarylmethylamine Diastereoselectivity N-tert-Butanesulfinyl imine |
| ISSN号 | 0040-4039 |
| 通讯作者 | Lin, Li ; 王锐 |
| 英文摘要 | This work concerns the asymmetric additions of benzothiazole to a variety of N-tert-butanesulfinyl imines with excellent diastereoselectivities (d.r. up to >99:1). Amino alkoxyl lithium was the key additive to obtain the excellent diastereoselectivity. More functionalized 4-methyl-5-vinyl thiazole and alkyl imines which can isomerize to enamines are also compatible substrates to the present protocol. |
| 学科主题 | 物理化学与绿色催化 |
| 收录类别 | SCI |
| 资助信息 | NSFC (nos. 21002043;21272107;20932003);the National S&T Major Project of China (2012ZX09504-001-003);Fundamental Research Funds for the Central Universities (lzujbky-2010-184) |
| 语种 | 英语 |
| WOS记录号 | WOS:000312231400005 |
| 公开日期 | 2016-05-03 |
| 源URL | [http://210.77.64.217/handle/362003/19432]  |
| 专题 | 兰州化学物理研究所_OSSO国家重点实验室 |
| 作者单位 | 1.Lanzhou Univ, Key Lab Preclin Study New Drugs Gansu Prov, State Key Lab Appl Organ Chem, Lanzhou 730000, Peoples R China 2.Lanzhou Univ, Inst Biochem & Mol Biol, Lanzhou 730000, Peoples R China 3.Chinese Acad Sci, Lanzhou Inst Chem Phys, State Key Lab Oxo Synth & Select Oxidat, Lanzhou 730000, Peoples R China |
| 推荐引用方式 GB/T 7714 | Zhang, Jinlong,Yang, Yuhong,Wang, Mei,et al. Asymmetric addition of benzothiazole to N-tert-butanesulfinyl imine for the synthesis of chiral alpha-branched heteroaryl amines[J]. Tetrahedron Letters,2012,53(51):6893-6896. |
| APA | Zhang, Jinlong,Yang, Yuhong,Wang, Mei,Lin, Li,&Wang R.(2012).Asymmetric addition of benzothiazole to N-tert-butanesulfinyl imine for the synthesis of chiral alpha-branched heteroaryl amines.Tetrahedron Letters,53(51),6893-6896. |
| MLA | Zhang, Jinlong,et al."Asymmetric addition of benzothiazole to N-tert-butanesulfinyl imine for the synthesis of chiral alpha-branched heteroaryl amines".Tetrahedron Letters 53.51(2012):6893-6896. |
入库方式： OAI收割
来源：兰州化学物理研究所
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