Environmental-benign oxidation of 2-oxazolines to oxazoles by dioxygen as the sole oxidant
文献类型：期刊论文
| 作者 | Huang, Yue2; Ni, Lijun2; Gan, Haifeng2; He, Yu2; Xu, Jinyi2; Wu, Xiaoming1; Yao, Hequan2,3 |
| 刊名 | TETRAHEDRON
 |
| 出版日期 | 2011-03-18 |
| 卷号 | 67期号:11页码:2066-2071 |
| 关键词 | Oxidation 2-Oxazolines Oxazoles Dioxygen Environmental-benign |
| ISSN号 | 0040-4020 |
| DOI | 10.1016/j.tet.2011.01.050 |
| 文献子类 | Article |
| 英文摘要 | A facile and environment-benign oxidation by dioxygen as the sole oxidant was applied for the conversion of 2-oxazolines to oxazoles. The substituent effect on 2-oxazoline ring was investigated. The use of this methodology for the synthesis of a key intermediate of a CDC25 phosphatase inhibitor (SC-alpha alpha delta 9) as an anticancer agent was also described. (C) 2011 Elsevier Ltd. All rights reserved. |
| WOS关键词 | PEPTIDE ANTIBIOTICS ; THIAZOLINES ; BIOSYNTHESIS ; PRECURSORS ; EPOTHILONE ; ALDEHYDES ; PRODUCTS |
| 资助项目 | State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences)[SIMM090104-KF-04] ; National Natural Science Foundation[20902111] ; Program for New Century Excellent Talents in University (NCET)[00000000] ; Ministry of Education of China[00000000] ; Fundamental Research Funds[JKZ2009002] ; Fundamental Research Funds[JKY2009013] |
| WOS研究方向 | Chemistry |
| 语种 | 英语 |
| WOS记录号 | WOS:000293037300009 |
| 出版者 | PERGAMON-ELSEVIER SCIENCE LTD |
| 源URL | [http://119.78.100.183/handle/2S10ELR8/278579]  |
| 专题 | 中国科学院上海药物研究所 |
| 通讯作者 | Yao, Hequan |
| 作者单位 | 1.China Pharmaceut Univ, Ctr Drug Discovery, Nanjing 210009, Jiangsu, Peoples R China; 2.China Pharmaceut Univ, Dept Med Chem, Sch Pharm, Nanjing 210009, Jiangsu, Peoples R China; 3.Chinese Acad Sci, Shanghai Inst Mat Med, Shanghai 201203, Peoples R China |
| 推荐引用方式 GB/T 7714 | Huang, Yue,Ni, Lijun,Gan, Haifeng,et al. Environmental-benign oxidation of 2-oxazolines to oxazoles by dioxygen as the sole oxidant[J]. TETRAHEDRON,2011,67(11):2066-2071. |
| APA | Huang, Yue.,Ni, Lijun.,Gan, Haifeng.,He, Yu.,Xu, Jinyi.,...&Yao, Hequan.(2011).Environmental-benign oxidation of 2-oxazolines to oxazoles by dioxygen as the sole oxidant.TETRAHEDRON,67(11),2066-2071. |
| MLA | Huang, Yue,et al."Environmental-benign oxidation of 2-oxazolines to oxazoles by dioxygen as the sole oxidant".TETRAHEDRON 67.11(2011):2066-2071. |
入库方式： OAI收割
来源：上海药物研究所
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