One-pot Synthesis of 6-Aza-chromone Derivatives Through Cascade Carbonylation-Sonogashira-Cyclization
文献类型：期刊论文
| 作者 | Cheng, Gang1; Qi, Yingbei1; Zhou, Xiaoqian1; Sheng, Rong1; Hu, Yong-Zhou1; Hu, Youhong2
|
| 刊名 | SCIENTIFIC REPORTS
 |
| 出版日期 | 2017-06-30 |
| 卷号 | 7 |
| ISSN号 | 2045-2322 |
| DOI | 10.1038/s41598-017-04693-7 |
| 文献子类 | Article |
| 英文摘要 | We developed an efficient synthesis of aza-chromones from 3-iodo-4-(1H)-pyridones and terminal acetylenes via a cascade carbonylation-Sonogashira-cyclization reaction. By controlling the use of bases, both 6-aza-chromones 5 and 3-(4-oxo-1,4-dihydroquinoline-3-carbonyl)-4H-pyrano[3,2-c] quinolin-4-ones 6 could be selectively obtained in moderate to good yields. |
| WOS关键词 | TERMINAL ACETYLENES ; ARYL IODIDES ; CO SOURCE ; FLAVONES ; CHROMONES ; FUROCOUMARINS ; IODOPHENOLS ; ANNULATION |
| 资助项目 | National Natural Science Foundation of China[81502916] ; Zhejiang Provincial Natural Science Foundation of China[LY16H300002] |
| WOS研究方向 | Science & Technology - Other Topics |
| 语种 | 英语 |
| WOS记录号 | WOS:000404451300004 |
| 出版者 | NATURE PUBLISHING GROUP |
| 源URL | [http://119.78.100.183/handle/2S10ELR8/272596]  |
| 专题 | 药物化学研究室 中科院受体结构与功能重点实验室 新药研究国家重点实验室 |
| 通讯作者 | Sheng, Rong; Hu, Youhong |
| 作者单位 | 1.Zhejiang Univ, Coll Pharmaceut Sci, Hangzhou 310058, Zhejiang, Peoples R China; 2.Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, 555 Zu Chong Zhi Rd, Shanghai 201203, Peoples R China |
| 推荐引用方式 GB/T 7714 | Cheng, Gang,Qi, Yingbei,Zhou, Xiaoqian,et al. One-pot Synthesis of 6-Aza-chromone Derivatives Through Cascade Carbonylation-Sonogashira-Cyclization[J]. SCIENTIFIC REPORTS,2017,7. |
| APA | Cheng, Gang,Qi, Yingbei,Zhou, Xiaoqian,Sheng, Rong,Hu, Yong-Zhou,&Hu, Youhong.(2017).One-pot Synthesis of 6-Aza-chromone Derivatives Through Cascade Carbonylation-Sonogashira-Cyclization.SCIENTIFIC REPORTS,7. |
| MLA | Cheng, Gang,et al."One-pot Synthesis of 6-Aza-chromone Derivatives Through Cascade Carbonylation-Sonogashira-Cyclization".SCIENTIFIC REPORTS 7(2017). |
入库方式： OAI收割
来源：上海药物研究所
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