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Formation of 1,3-diazocine by palladium catalyzed C-H arylation

文献类型：期刊论文

作者Tang, Le1,2; Ren, Jing2,3; Ma, Yuchi2,3; Wang, Xin2,3; Chen, Lin2,3; Shen, Jingkang2,3; Chen, Yue-Lei2,3; Xiong, Bing2,3
刊名TETRAHEDRON LETTERS
出版日期2016-05-25
卷号57期号:21页码:2311-2314
关键词1,3-Diazocine C-H arylation 8-Aminoimidazo[1,2-alpha]pyrazines 8-Membered ring Groebke-Blackburn-Bienayme reaction
ISSN号0040-4039
DOI10.1016/j.tetlet.2016.04.050
文献子类Article
英文摘要From multi-substituted 8-aminoimidazo[1,2-alpha]pyrazines, prepared via modified Grothke-Blackburn-Bienayme reaction, a Pd-catalyzed cyclization reaction was discovered, leading to a rare (Z)-4,5-dihydro-3H-[1,3]diazocine system. Conditions of this cyclization were screened and DMF solvent was found as one of the key factors for the cyclization. (C) 2016 Elsevier Ltd. All rights reserved.
WOS关键词SUZUKI COUPLING REACTION ; LIGAND ; AMIDE
资助项目National Natural Science Foundation of China[81273368] ; National Science & Technology Major Project - Key New Drug Creation and Manufacturing Program - of China[2014ZX09507-002]
WOS研究方向Chemistry
语种英语
WOS记录号WOS:000376212300026
出版者PERGAMON-ELSEVIER SCIENCE LTD
源URL[http://119.78.100.183/handle/2S10ELR8/276038]  
专题药物化学研究室
中科院受体结构与功能重点实验室
新药研究国家重点实验室
通讯作者Chen, Yue-Lei; Xiong, Bing
作者单位1.Nanchang Univ, Coll Pharm, 461 Bayi Rd, Nanchang 330006, Peoples R China;
2.Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, 555 Zuchongzhi Rd, Shanghai 201203, Peoples R China;
3.Univ Chinese Acad Sci, 19A Yuquan Rd, Beijing 100049, Peoples R China
推荐引用方式
GB/T 7714		 Tang, Le,Ren, Jing,Ma, Yuchi,et al. Formation of 1,3-diazocine by palladium catalyzed C-H arylation[J]. TETRAHEDRON LETTERS,2016,57(21):2311-2314.
APA Tang, Le.,Ren, Jing.,Ma, Yuchi.,Wang, Xin.,Chen, Lin.,...&Xiong, Bing.(2016).Formation of 1,3-diazocine by palladium catalyzed C-H arylation.TETRAHEDRON LETTERS,57(21),2311-2314.
MLA Tang, Le,et al."Formation of 1,3-diazocine by palladium catalyzed C-H arylation".TETRAHEDRON LETTERS 57.21(2016):2311-2314.

入库方式： OAI收割

来源：上海药物研究所

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