A facile trifluoromethylthiolation of 3-chloro-1H-inden-1-ones employing AgSCF3 and KI
文献类型：期刊论文
| 作者 | Dong, Biao1; Zhang, Xiaofei2,3; Liu, Ruiling2,3; Yang, Chunhao2,3
|
| 刊名 | ARKIVOC
 |
| 出版日期 | 2016 |
| 页码 | 296-305 |
| 关键词 | 3-Chloro-1H-inden-1-ones trifluoromethylthiolation AgSCF3 KI |
| ISSN号 | 1551-7004 |
| DOI | 10.3998/ark.5550190.p009.606 |
| 文献子类 | Article |
| 英文摘要 | An efficient method for trifluoromethylthiolation of functionalized 3-chloro-1H-inden-1-ones was described. Within this method, AgSCF3 was employed as a nucleophilic reagent and KI was functionalized as an activator. This reaction provided the trifluoromethylthiolated indenones with excellent yields under moderate conditions. |
| WOS关键词 | ENANTIOSELECTIVE TRIFLUOROMETHYLTHIOLATION ; ANTICANCER AGENTS ; RECEPTOR ; INHIBITORS ; OXINDOLES ; FLUORINE ; INDOLES |
| 资助项目 | National Natural Science Foundation of China[81321092] ; SKLDR/SIMM[SIMM1601ZZ-03] |
| WOS研究方向 | Chemistry |
| 语种 | 英语 |
| WOS记录号 | WOS:000387971100005 |
| 出版者 | ARKAT USA INC |
| 源URL | [http://119.78.100.183/handle/2S10ELR8/276190]  |
| 专题 | 药物化学研究室 中科院受体结构与功能重点实验室 新药研究国家重点实验室 |
| 通讯作者 | Yang, Chunhao |
| 作者单位 | 1.Univ Sci & Technol China, Nano Sci & Technol Inst, Suzhou 215123, Peoples R China; 2.Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Shanghai 201203, Peoples R China; 3.Univ Chinese Acad Sci, 19A Yuquan Rd, Beijing 100049, Peoples R China |
| 推荐引用方式 GB/T 7714 | Dong, Biao,Zhang, Xiaofei,Liu, Ruiling,et al. A facile trifluoromethylthiolation of 3-chloro-1H-inden-1-ones employing AgSCF3 and KI[J]. ARKIVOC,2016:296-305. |
| APA | Dong, Biao,Zhang, Xiaofei,Liu, Ruiling,&Yang, Chunhao.(2016).A facile trifluoromethylthiolation of 3-chloro-1H-inden-1-ones employing AgSCF3 and KI.ARKIVOC,296-305. |
| MLA | Dong, Biao,et al."A facile trifluoromethylthiolation of 3-chloro-1H-inden-1-ones employing AgSCF3 and KI".ARKIVOC (2016):296-305. |
入库方式： OAI收割
来源：上海药物研究所
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