Indium-Mediated Asymmetric Intramolecular Allenylation of N-tert-Butanesulfinyl Imines: Efficient and Practical Access to Chiral 3-Allenyl-4-aminochromanes
文献类型：期刊论文
| 作者 | Su, Lin; Zhu, Ting-Shun; Xu, Ming-Hua
|
| 刊名 | ORGANIC LETTERS
 |
| 出版日期 | 2014-08-15 |
| 卷号 | 16期号:16页码:4118-4121 |
| ISSN号 | 1523-7060 |
| DOI | 10.1021/ol501815e |
| 文献子类 | Article |
| 英文摘要 | An efficient method for the preparation of highly optically active 3-allenyl- and 3-vinyl-4-aminochromanes by In-mediated intramolecular cyclization has been developed. The synthetic utilities of the approach were demonstrated by the construction of various chiral polycyclic heterocycles, especially the interesting spiroheterocyclic compound 9 and steroid analogue 10. |
| WOS关键词 | ONE-POT SYNTHESIS ; ENANTIOSELECTIVE HYDROGENATION ; AMINES. APPLICATION ; KHAND REACTION ; DERIVATIVES ; ALLYLATION ; KETIMINES ; ANALOGS ; ACIDS |
| 资助项目 | National Natural Science Foundation of China[21325209] ; Shanghai Municipal Committee of Science and Technology[14XD1404400] |
| WOS研究方向 | Chemistry |
| 语种 | 英语 |
| WOS记录号 | WOS:000340517200016 |
| 出版者 | AMER CHEMICAL SOC |
| 源URL | [http://119.78.100.183/handle/2S10ELR8/276943]  |
| 专题 | 药物化学研究室 中科院受体结构与功能重点实验室 新药研究国家重点实验室 |
| 通讯作者 | Xu, Ming-Hua |
| 作者单位 | Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Shanghai 201203, Peoples R China |
| 推荐引用方式 GB/T 7714 | Su, Lin,Zhu, Ting-Shun,Xu, Ming-Hua. Indium-Mediated Asymmetric Intramolecular Allenylation of N-tert-Butanesulfinyl Imines: Efficient and Practical Access to Chiral 3-Allenyl-4-aminochromanes[J]. ORGANIC LETTERS,2014,16(16):4118-4121. |
| APA | Su, Lin,Zhu, Ting-Shun,&Xu, Ming-Hua.(2014).Indium-Mediated Asymmetric Intramolecular Allenylation of N-tert-Butanesulfinyl Imines: Efficient and Practical Access to Chiral 3-Allenyl-4-aminochromanes.ORGANIC LETTERS,16(16),4118-4121. |
| MLA | Su, Lin,et al."Indium-Mediated Asymmetric Intramolecular Allenylation of N-tert-Butanesulfinyl Imines: Efficient and Practical Access to Chiral 3-Allenyl-4-aminochromanes".ORGANIC LETTERS 16.16(2014):4118-4121. |
入库方式： OAI收割
来源：上海药物研究所
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