Synthesis of Multisubstituted 2-Aminopyrroles/pyridines via Chemoselective Michael Addition/Intramolecular Cyclization Reaction
文献类型：期刊论文
| 作者 | Qi, Xueyu; Xiang, Haoyue; He, Qian ; Yang, Chunhao
|
| 刊名 | ORGANIC LETTERS
 |
| 出版日期 | 2014-08-15 |
| 卷号 | 16期号:16页码:4186-4189 |
| ISSN号 | 1523-7060 |
| DOI | 10.1021/ol5018855 |
| 文献子类 | Article |
| 英文摘要 | A facile and efficient synthetic strategy to construct polysubstituted 2-aminopyrroles/pyridines was developed via chemoselective Michael addition/intramolecular cydization reaction under very mild conditions. It suggested that the chemoselectivity of the process could be controlled by the leaving ability of the halides. |
| WOS关键词 | INHIBITORS ; 2-AMINOPYRIDINES ; DERIVATIVES ; EFFICIENT ; PYRROLES ; ALKYNES ; ALPHA ; MILD ; IDENTIFICATION ; MULTICOMPONENT |
| 资助项目 | Ministry of Science and Technology of China[2012ZX09301001-001] ; National Natural Science Foundation of China[81321092] ; SKLDR/SIMM[SIMM1403ZZ-01] |
| WOS研究方向 | Chemistry |
| 语种 | 英语 |
| WOS记录号 | WOS:000340517200033 |
| 出版者 | AMER CHEMICAL SOC |
| 源URL | [http://119.78.100.183/handle/2S10ELR8/276944]  |
| 专题 | 药物化学研究室 中科院受体结构与功能重点实验室 新药研究国家重点实验室 |
| 通讯作者 | Yang, Chunhao |
| 作者单位 | Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Shanghai 201203, Peoples R China |
| 推荐引用方式 GB/T 7714 | Qi, Xueyu,Xiang, Haoyue,He, Qian,et al. Synthesis of Multisubstituted 2-Aminopyrroles/pyridines via Chemoselective Michael Addition/Intramolecular Cyclization Reaction[J]. ORGANIC LETTERS,2014,16(16):4186-4189. |
| APA | Qi, Xueyu,Xiang, Haoyue,He, Qian,&Yang, Chunhao.(2014).Synthesis of Multisubstituted 2-Aminopyrroles/pyridines via Chemoselective Michael Addition/Intramolecular Cyclization Reaction.ORGANIC LETTERS,16(16),4186-4189. |
| MLA | Qi, Xueyu,et al."Synthesis of Multisubstituted 2-Aminopyrroles/pyridines via Chemoselective Michael Addition/Intramolecular Cyclization Reaction".ORGANIC LETTERS 16.16(2014):4186-4189. |
入库方式： OAI收割
来源：上海药物研究所
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