Copper-Mediated, Palladium-Catalyzed Cross-Coupling of 3-Iodochromones, Thiochromones, and Quinolones with Ethyl Bromodifluoroacetate
文献类型：期刊论文
| 作者 | Han, Xiaodong1,2; Yue, Zhizhou2; Zhang, Xiaofei1; He, Qian1 ; Yang, Chunhao1
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| 刊名 | JOURNAL OF ORGANIC CHEMISTRY
 |
| 出版日期 | 2013-05-17 |
| 卷号 | 78期号:10页码:4850-4856 |
| ISSN号 | 0022-3263 |
| DOI | 10.1021/jo400412k |
| 文献子类 | Article |
| 英文摘要 | The palladium-catalyzed cross-coupling reaction of 3-iodochromones, thiochromones, and quinolones with ethyl bromodifluoroacetate in the presence of a copper mediator is reported. Under optimized conditions, all reactions worked well and provided difluoro-containing products in moderate to excellent yields. |
| WOS关键词 | CHROMONE DERIVATIVES ; MEDICINAL CHEMISTRY ; HALO-ENONES ; INHIBITORS ; TRIFLUOROMETHYLATION ; DIFLUOROMETHYLATION ; TRANSFORMATION ; SUBSTITUTION ; HETEROCYCLES ; DISCOVERY |
| 资助项目 | "Interdisciplinary Cooperation Team" Program for Science and Technology Innovation of Chinese Academy of Science[00000000] ; National Natural Science Foundation of China[21072205] ; National Natural Science Foundation of China[SIMM1203ZZ-0103] |
| WOS研究方向 | Chemistry |
| 语种 | 英语 |
| WOS记录号 | WOS:000319721200019 |
| 出版者 | AMER CHEMICAL SOC |
| 源URL | [http://119.78.100.183/handle/2S10ELR8/277615]  |
| 专题 | 药物化学研究室 中科院受体结构与功能重点实验室 新药研究国家重点实验室 |
| 通讯作者 | Yang, Chunhao |
| 作者单位 | 1.Chinese Acad Sci, Shanghai Inst Mat Med, SIBS, State Key Lab Drug Res, Shanghai 201203, Peoples R China; 2.Wuhan Univ Technol, Sch Chem Engn, Dept Pharmaceut Engn, Wuhan 430070, Hubei, Peoples R China |
| 推荐引用方式 GB/T 7714 | Han, Xiaodong,Yue, Zhizhou,Zhang, Xiaofei,et al. Copper-Mediated, Palladium-Catalyzed Cross-Coupling of 3-Iodochromones, Thiochromones, and Quinolones with Ethyl Bromodifluoroacetate[J]. JOURNAL OF ORGANIC CHEMISTRY,2013,78(10):4850-4856. |
| APA | Han, Xiaodong,Yue, Zhizhou,Zhang, Xiaofei,He, Qian,&Yang, Chunhao.(2013).Copper-Mediated, Palladium-Catalyzed Cross-Coupling of 3-Iodochromones, Thiochromones, and Quinolones with Ethyl Bromodifluoroacetate.JOURNAL OF ORGANIC CHEMISTRY,78(10),4850-4856. |
| MLA | Han, Xiaodong,et al."Copper-Mediated, Palladium-Catalyzed Cross-Coupling of 3-Iodochromones, Thiochromones, and Quinolones with Ethyl Bromodifluoroacetate".JOURNAL OF ORGANIC CHEMISTRY 78.10(2013):4850-4856. |
入库方式： OAI收割
来源：上海药物研究所
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