Design and Synthesis of (R)-1-Arylsulfonylpiperidine-2-carboxamides as 11 beta-Hydroxysteroid Dehydrogenase Type 1 Inhibitors
文献类型:期刊论文
作者 | Xia, Guangxin1,2; Liu, Lin1,2; Liu, Haiyan1; Yu, Jianxin1; Xu, Zhenmin1; Chen, Qian1; Ma, Chen1; Li, Ping1; Xiong, Bing2![]() |
刊名 | CHEMMEDCHEM
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出版日期 | 2013-04 |
卷号 | 8期号:4页码:577-581 |
关键词 | 11-HSD1 diabetes docking inhibitors |
ISSN号 | 1860-7179 |
DOI | 10.1002/cmdc.201300022 |
文献子类 | Article |
WOS关键词 | 11-BETA-HSD1 INHIBITORS ; SELECTIVE INHIBITORS ; DISCOVERY ; DOCKING ; POTENT |
资助项目 | New Drug Creation Project of the National Science and Technology Major Foundation of China[2010ZX09401-404] ; Shanghai Pharmaceutical Holding, Shanghai Postdoctoral Sustentation Fund China[07R214213] ; Program of Excellent Young Scientist of the Chinese Academy of Sciences[KSCX2-EW-Q-3-01] |
WOS研究方向 | Pharmacology & Pharmacy |
语种 | 英语 |
WOS记录号 | WOS:000316811100005 |
出版者 | WILEY-V C H VERLAG GMBH |
源URL | [http://119.78.100.183/handle/2S10ELR8/277675] ![]() |
专题 | 药物化学研究室 中科院受体结构与功能重点实验室 新药研究国家重点实验室 |
通讯作者 | Xia, Guangxin |
作者单位 | 1.Shanghai Pharmaceut Holding Co Ltd, Cent Res Inst, Shanghai 201203, Peoples R China; 2.Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, Shanghai 201203, Peoples R China |
推荐引用方式 GB/T 7714 | Xia, Guangxin,Liu, Lin,Liu, Haiyan,et al. Design and Synthesis of (R)-1-Arylsulfonylpiperidine-2-carboxamides as 11 beta-Hydroxysteroid Dehydrogenase Type 1 Inhibitors[J]. CHEMMEDCHEM,2013,8(4):577-581. |
APA | Xia, Guangxin.,Liu, Lin.,Liu, Haiyan.,Yu, Jianxin.,Xu, Zhenmin.,...&Shen, Jingkang.(2013).Design and Synthesis of (R)-1-Arylsulfonylpiperidine-2-carboxamides as 11 beta-Hydroxysteroid Dehydrogenase Type 1 Inhibitors.CHEMMEDCHEM,8(4),577-581. |
MLA | Xia, Guangxin,et al."Design and Synthesis of (R)-1-Arylsulfonylpiperidine-2-carboxamides as 11 beta-Hydroxysteroid Dehydrogenase Type 1 Inhibitors".CHEMMEDCHEM 8.4(2013):577-581. |
入库方式: OAI收割
来源:上海药物研究所
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