Nickel-Catalyzed ortho-C-H Thiolation of N-Benzoyl alpha-Amino Acid Derivatives
文献类型：期刊论文
| 作者 | Gao, Feng; Zhu, Wei; Zhang, Dengyou; Li, Shuangjie; Wang, Jiang ; Liu, Hong
|
| 刊名 | JOURNAL OF ORGANIC CHEMISTRY
 |
| 出版日期 | 2016-10-07 |
| 卷号 | 81期号:19页码:9122-9130 |
| ISSN号 | 0022-3263 |
| DOI | 10.1021/acs.joc.6b01702 |
| 文献子类 | Article |
| 英文摘要 | We developed the first nickel-catalyzed direct ortho-thiolation of N-benzoyl alpha-amino acid derivatives. This novel strategy showed wide generality, functional tolerance, and high regioselectivity. In addition, dipeptide derivatives were also compatible with this transformation system, providing a potential protocol for the direct modification of peptide derivatives. |
| WOS关键词 | BOND ACTIVATION ; ALIPHATIC AMIDES ; C(SP(3))-H BONDS ; DIRECTING GROUP ; ARYL SULFIDES ; INHIBITORS ; FUNCTIONALIZATION ; ARENES ; SULFENYLATION ; ANALOGS |
| 资助项目 | National Natural Science Foundation of China[91229204] ; National Natural Science Foundation of China[21632008] ; National Natural Science Foundation of China[81620108027] ; Major Project of Chinese National Programs for Fundamental Research and Development[2015CB910304] ; National S&T Major Projects[2013ZX09507-001] ; National S&T Major Projects[2014ZX09507002-001] |
| WOS研究方向 | Chemistry |
| 语种 | 英语 |
| WOS记录号 | WOS:000385054300041 |
| 出版者 | AMER CHEMICAL SOC |
| 源URL | [http://119.78.100.183/handle/2S10ELR8/275864]  |
| 专题 | 药物化学研究室 |
| 通讯作者 | Liu, Hong |
| 作者单位 | Chinese Acad Sci, Shanghai Inst Mat Med, CAS Key Lab Receptor Res, 555 Zuchongzhi Rd, Shanghai 201203, Peoples R China |
| 推荐引用方式 GB/T 7714 | Gao, Feng,Zhu, Wei,Zhang, Dengyou,et al. Nickel-Catalyzed ortho-C-H Thiolation of N-Benzoyl alpha-Amino Acid Derivatives[J]. JOURNAL OF ORGANIC CHEMISTRY,2016,81(19):9122-9130. |
| APA | Gao, Feng,Zhu, Wei,Zhang, Dengyou,Li, Shuangjie,Wang, Jiang,&Liu, Hong.(2016).Nickel-Catalyzed ortho-C-H Thiolation of N-Benzoyl alpha-Amino Acid Derivatives.JOURNAL OF ORGANIC CHEMISTRY,81(19),9122-9130. |
| MLA | Gao, Feng,et al."Nickel-Catalyzed ortho-C-H Thiolation of N-Benzoyl alpha-Amino Acid Derivatives".JOURNAL OF ORGANIC CHEMISTRY 81.19(2016):9122-9130. |
入库方式： OAI收割
来源：上海药物研究所
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