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Rhodium-catalyzed oxidative coupling of N-acyl anilines with alkynes using an acylamino moiety as the traceless directing group

文献类型：期刊论文

作者Geng, Kaijun; Fan, Zhoulong; Zhang, Ao1,2
刊名ORGANIC CHEMISTRY FRONTIERS
出版日期2016
卷号3期号:3页码:349-353
ISSN号2052-4129
DOI10.1039/c5qo00387c
文献子类Article
英文摘要A rhodium-catalyzed oxidative annulation of N-acyl anilines with alkynes was developed by using the acylamino group as a traceless directing group for the first time. Various N-acyl anilines and para-or meta-substituted diphenylacetylenes were well tolerated, and a series of 1,2,3,4-tetrasubstituted naphthalenes were readily synthesized in good to excellent yields. Meanwhile, this method also provides a new strategy for the N-dearylation of N-phenylamides.
WOS关键词C-H ACTIVATION ; CARBOXYLIC-ACIDS ; BOND ACTIVATION ; FUNCTIONALIZATION ; ARENES ; SEMICONDUCTORS ; OLEFINATION ; AMINATION ; ARYLATION ; DIVERSE
资助项目Chinese NSF[81430080] ; Chinese NSF[81125021] ; Major State Basic Research Development Program[2015CB910603] ; SIMM[CASIMM0120154002/2002]
WOS研究方向Chemistry
语种英语
WOS记录号WOS:000371235300012
出版者CHINESE CHEMICAL SOC
源URL[http://119.78.100.183/handle/2S10ELR8/276246]  
专题药物化学研究室
通讯作者Zhang, Ao
作者单位1.Chinese Acad Sci, SIMM, CAS Key Lab Receptor Res, Shanghai 201203, Peoples R China;
2.Chinese Acad Sci, SIMM, SOMCL, Shanghai 201203, Peoples R China
推荐引用方式
GB/T 7714		 Geng, Kaijun,Fan, Zhoulong,Zhang, Ao. Rhodium-catalyzed oxidative coupling of N-acyl anilines with alkynes using an acylamino moiety as the traceless directing group[J]. ORGANIC CHEMISTRY FRONTIERS,2016,3(3):349-353.
APA Geng, Kaijun,Fan, Zhoulong,&Zhang, Ao.(2016).Rhodium-catalyzed oxidative coupling of N-acyl anilines with alkynes using an acylamino moiety as the traceless directing group.ORGANIC CHEMISTRY FRONTIERS,3(3),349-353.
MLA Geng, Kaijun,et al."Rhodium-catalyzed oxidative coupling of N-acyl anilines with alkynes using an acylamino moiety as the traceless directing group".ORGANIC CHEMISTRY FRONTIERS 3.3(2016):349-353.

入库方式： OAI收割

来源：上海药物研究所

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