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Microwave-assisted synthesis of 5,6-dihydroindolo[1,2-a] quinoxaline derivatives through copper-catalyzed intramolecular N-arylation

文献类型：期刊论文

作者Zhao, Fei; Zhang, Lei; Liu, Hailong; Zhou, Shengbin; Liu, Hong
刊名BEILSTEIN JOURNAL OF ORGANIC CHEMISTRY
出版日期2013-11-14
卷号9页码:2463-2469
关键词copper 5,6-dihydroindolo[1,2-a]quinoxaline intramolecular N-arylation microwave irradiation
ISSN号1860-5397
DOI10.3762/bjoc.9.285
文献子类Article
英文摘要An efficient and practical protocol has been developed to synthesize 5,6-dihydroindolo[ 1,2-a] quinoxaline derivatives by CuI-catalyzed intramolecular N-arylation under microwave irradiation. This method rapidly afforded the tetracyclic products with good to excellent yields (83-97%) in short reaction times (45-60 min).
WOS关键词INDOLE ALKALOIDS ; DRUG DISCOVERY ; ARYL HALIDES ; HETEROCYCLES ; CHEMISTRY ; EFFICIENT ; CASCADE ; AMINES ; MILD ; ACID
资助项目National Natural Science Foundation of China[21021063] ; National Natural Science Foundation of China[91229204] ; National Natural Science Foundation of China[81025017] ; National S& T Major Projects[2012ZX09103101-072] ; National S& T Major Projects[2012ZX09301001005]
WOS研究方向Chemistry
语种英语
WOS记录号WOS:000327708000001
出版者BEILSTEIN-INSTITUT
源URL[http://119.78.100.183/handle/2S10ELR8/277378]  
专题药物化学研究室
通讯作者Liu, Hong
作者单位Chinese Acad Sci, Shanghai Inst Mat Med, CAS Key Lab Receptor Res, Shanghai 201203, Peoples R China
推荐引用方式
GB/T 7714		 Zhao, Fei,Zhang, Lei,Liu, Hailong,et al. Microwave-assisted synthesis of 5,6-dihydroindolo[1,2-a] quinoxaline derivatives through copper-catalyzed intramolecular N-arylation[J]. BEILSTEIN JOURNAL OF ORGANIC CHEMISTRY,2013,9:2463-2469.
APA Zhao, Fei,Zhang, Lei,Liu, Hailong,Zhou, Shengbin,&Liu, Hong.(2013).Microwave-assisted synthesis of 5,6-dihydroindolo[1,2-a] quinoxaline derivatives through copper-catalyzed intramolecular N-arylation.BEILSTEIN JOURNAL OF ORGANIC CHEMISTRY,9,2463-2469.
MLA Zhao, Fei,et al."Microwave-assisted synthesis of 5,6-dihydroindolo[1,2-a] quinoxaline derivatives through copper-catalyzed intramolecular N-arylation".BEILSTEIN JOURNAL OF ORGANIC CHEMISTRY 9(2013):2463-2469.

入库方式： OAI收割

来源：上海药物研究所

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