Proline potassium salt: a superior catalyst to synthesize 4-trifluoromethyl quinoline derivatives via Friedlander annulation
文献类型：期刊论文
| 作者 | Du, Xiao Long1; Jiang, Biao2; Li, Yuan Chao1 |
| 刊名 | TETRAHEDRON
 |
| 出版日期 | 2013-09-02 |
| 卷号 | 69期号:35页码:7481-7486 |
| 关键词 | Proline potassium salt 2-Trifluoroacetyl anilines 4-Trifluoromethyl quinoline |
| ISSN号 | 0040-4020 |
| DOI | 10.1016/j.tet.2013.06.017 |
| 文献子类 | Article |
| 英文摘要 | Proline potassium salt was successfully firstly used to catalyze the Friedlander annulation toward the synthesis of 4-trifluoromethyl-substituted quinolines from the substituted 2-trifluoroacetyl anilines and variety carbonyl compounds under mild conditions in good to excellent yields. This catalyst provides several advantages, such as shorter reaction time, high regioselectivity, functional group tolerance, and broad substrate scope. (C) 2013 The Authors. Published by Elsevier Ltd. All rights reserved. |
| WOS关键词 | ONE-POT SYNTHESIS ; REGIOSELECTIVE SYNTHESIS ; EFFICIENT SYNTHESIS ; CYCLIZATION ; ACID ; MECHANISM |
| WOS研究方向 | Chemistry |
| 语种 | 英语 |
| WOS记录号 | WOS:000322557500038 |
| 出版者 | PERGAMON-ELSEVIER SCIENCE LTD |
| 源URL | [http://119.78.100.183/handle/2S10ELR8/277470]  |
| 专题 | 药物化学研究室 |
| 通讯作者 | Jiang, Biao |
| 作者单位 | 1.Chinese Acad Sci, Shanghai Inst Mat Med, Shanghai 201203, Peoples R China; 2.Chinese Acad Sci, Shanghai Inst Organ Chem, Shanghai 200032, Peoples R China |
| 推荐引用方式 GB/T 7714 | Du, Xiao Long,Jiang, Biao,Li, Yuan Chao. Proline potassium salt: a superior catalyst to synthesize 4-trifluoromethyl quinoline derivatives via Friedlander annulation[J]. TETRAHEDRON,2013,69(35):7481-7486. |
| APA | Du, Xiao Long,Jiang, Biao,&Li, Yuan Chao.(2013).Proline potassium salt: a superior catalyst to synthesize 4-trifluoromethyl quinoline derivatives via Friedlander annulation.TETRAHEDRON,69(35),7481-7486. |
| MLA | Du, Xiao Long,et al."Proline potassium salt: a superior catalyst to synthesize 4-trifluoromethyl quinoline derivatives via Friedlander annulation".TETRAHEDRON 69.35(2013):7481-7486. |
入库方式： OAI收割
来源：上海药物研究所
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