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InBr3-Catalyzed Glycosidation of Glycals with Arylamines: An Alternative Approach To Access 4-Aminocyclopent-2-enones

文献类型：期刊论文

作者Li, Fulong1,2; Ding, Chunyong1,2; Wang, Meining2; Yao, Qizheng1; Zhang, Ao2
刊名JOURNAL OF ORGANIC CHEMISTRY
出版日期2011-04-15
卷号76期号:8页码:2820-2827
ISSN号0022-3263
DOI10.1021/jo200243d
文献子类Article
英文摘要To turn side products into major products, a novel strategy to access biologically active 4-aminocyclopent-2-enones was developed. These compounds were originally identified as side products but became major products when 3,5-dimethylpyran-3,4-diol 7a was used as the substrate and 30% InBr3 as the catalyst. Aryl- or heteroarylamines as well as variously substituted glycals can be used in this reaction, and the corresponding 4-aminocyclopent-2-enones were obtained in moderate to good yields. These compounds can be further used to prepare 4-aminocarbocyclic nucleosides.
WOS关键词ANTIVIRAL ACTIVITY ; CYCLIZATION ; THYMINE
资助项目Key Laboratory of Pesticide & Chemical Biology, Central China Normal University[201005A02]
WOS研究方向Chemistry
语种英语
WOS记录号WOS:000289187300045
出版者AMER CHEMICAL SOC
源URL[http://119.78.100.183/handle/2S10ELR8/278555]  
专题药物化学研究室
通讯作者Yao, Qizheng
作者单位1.China Pharmaceut Univ, Dept Med Chem, Nanjing 210009, Peoples R China;
2.SIMM, SOMCL, Shanghai 201203, Peoples R China
推荐引用方式
GB/T 7714		 Li, Fulong,Ding, Chunyong,Wang, Meining,et al. InBr3-Catalyzed Glycosidation of Glycals with Arylamines: An Alternative Approach To Access 4-Aminocyclopent-2-enones[J]. JOURNAL OF ORGANIC CHEMISTRY,2011,76(8):2820-2827.
APA Li, Fulong,Ding, Chunyong,Wang, Meining,Yao, Qizheng,&Zhang, Ao.(2011).InBr3-Catalyzed Glycosidation of Glycals with Arylamines: An Alternative Approach To Access 4-Aminocyclopent-2-enones.JOURNAL OF ORGANIC CHEMISTRY,76(8),2820-2827.
MLA Li, Fulong,et al."InBr3-Catalyzed Glycosidation of Glycals with Arylamines: An Alternative Approach To Access 4-Aminocyclopent-2-enones".JOURNAL OF ORGANIC CHEMISTRY 76.8(2011):2820-2827.

入库方式： OAI收割

来源：上海药物研究所

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