synthesisandevaluationofpde5inhibitoryactivityofnovelpyrido2151pyrazolo43dpyrimidin4onederivatives
文献类型:期刊论文
作者 | GuangHui Tian1; GuangXin Xia1; WeiXi Jin2; XinJian Chen1; ShunAn Lai3; YaBing Wei2; RuYun Ji1; JingShan Shen1![]() |
刊名 | chinesejournalofchemistry
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出版日期 | 2007 |
卷号 | 25期号:2页码:241 |
关键词 | ERECTILE DYSFUNCTION RECEPTOR ANTAGONISTS SILDENAFIL ANALOGS POTENT PHOSPHODIESTERASE |
ISSN号 | 1001-604X |
英文摘要 | Novel pyridopyrazolopyrimidinone derivatives were designed and synthesized as potential PDE5 inhibitors. The target compounds demonstrated significant inhibitory activity against human platelet PDE5, but less potent than sildenafil. |
语种 | 英语 |
源URL | [http://119.78.100.183/handle/2S10ELR8/285225] ![]() |
专题 | 中国科学院上海药物研究所 |
作者单位 | 1.中国科学院上海药物研究所 2.南京工业大学 3.Topharman Shanghai Co., Ltd |
推荐引用方式 GB/T 7714 | GuangHui Tian,GuangXin Xia,WeiXi Jin,et al. synthesisandevaluationofpde5inhibitoryactivityofnovelpyrido2151pyrazolo43dpyrimidin4onederivatives[J]. chinesejournalofchemistry,2007,25(2):241. |
APA | GuangHui Tian.,GuangXin Xia.,WeiXi Jin.,XinJian Chen.,ShunAn Lai.,...&JingShan Shen.(2007).synthesisandevaluationofpde5inhibitoryactivityofnovelpyrido2151pyrazolo43dpyrimidin4onederivatives.chinesejournalofchemistry,25(2),241. |
MLA | GuangHui Tian,et al."synthesisandevaluationofpde5inhibitoryactivityofnovelpyrido2151pyrazolo43dpyrimidin4onederivatives".chinesejournalofchemistry 25.2(2007):241. |
入库方式: OAI收割
来源:上海药物研究所
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