中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
首页 机构 成果 学者
  
  1. CAS IR Grid
  2. 上海药物研究所
  3. 中国科学院上海药物研究所
  4. 新药研究国家重点实验室
One Pot and Metal-Free Approach to 3-(2-Hydroxybenzoyl)-1-aza-anthraquinones

文献类型：期刊论文

作者Yuan, Jiaqi1,2; He, Qian1; Song, Shanshan1; Zhang, Xiaofei1; Miao, Zehong1; Yang, Chunhao1,2
刊名MOLECULES
出版日期2019-08-01
卷号24期号:16页码:12
关键词3-(2-hydroxybenzoyl)-1-aza-anthraquinones chromones anti-proliferation agent
DOI10.3390/molecules24163017
通讯作者Zhang, Xiaofei(xiaofeizhang@simm.ac.cn) ; Yang, Chunhao(chyang@simm.ac.cn)
英文摘要Herein, a direct strategy to synthesize 3-(2-hydroxybenzoyl)-1-aza-anthraquinones with excellent efficiency, mild conditions, and benign functional group compatibility was reported. A variety of 3-formylchromone compounds were employed as compatible substrates and this protocol gave the 3-(2-hydroxybenzoyl)-1-aza-anthraquinone derivatives in good to excellent yields without inert gas and expensive transition metal catalysts. Some compounds displayed good anti-proliferative activities.
WOS关键词CATALYZED INTRAMOLECULAR CYCLIZATION ; DIELS-ALDER ; FACILE ROUTE ; ANALOGS ; 3-FORMYLCHROMONES ; CYCLOADDITION ; KALASINAMIDE ; DERIVATIVES
资助项目Science and Technology Commission of Shanghai Municipality[18431907100] ; Shanghai Sailing Program[17YF1423400] ; SKLDR/SIMM[SIMM1903ZZ-03]
WOS研究方向Biochemistry & Molecular Biology ; Chemistry
语种英语
WOS记录号WOS:000482998900038
出版者MDPI
源URL[http://119.78.100.183/handle/2S10ELR8/288680]  
专题新药研究国家重点实验室
通讯作者Zhang, Xiaofei; Yang, Chunhao
作者单位1.Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, 555 Zuchongzhi Rd, Shanghai 201203, Peoples R China
2.Univ Chinese Acad Sci, Sch Pharm, 19A Yuquan Rd, Beijing 100049, Peoples R China
推荐引用方式
GB/T 7714		 Yuan, Jiaqi,He, Qian,Song, Shanshan,et al. One Pot and Metal-Free Approach to 3-(2-Hydroxybenzoyl)-1-aza-anthraquinones[J]. MOLECULES,2019,24(16):12.
APA Yuan, Jiaqi,He, Qian,Song, Shanshan,Zhang, Xiaofei,Miao, Zehong,&Yang, Chunhao.(2019).One Pot and Metal-Free Approach to 3-(2-Hydroxybenzoyl)-1-aza-anthraquinones.MOLECULES,24(16),12.
MLA Yuan, Jiaqi,et al."One Pot and Metal-Free Approach to 3-(2-Hydroxybenzoyl)-1-aza-anthraquinones".MOLECULES 24.16(2019):12.

入库方式： OAI收割

来源：上海药物研究所

浏览0
下载0
收藏0
其他版本

除非特别说明，本系统中所有内容都受版权保护，并保留所有权利。