中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
Substituent-Oriented Synthesis of Substituted Pyrazoles/Chromeno[3,2-c]pyrazoles via Sequential Reactions of Chromones/3-Chlorochromones and Tosylhydrazones

文献类型:期刊论文

作者Dai, Tianzi1,2; Li, Qunyi3; Zhang, Xiaofei1,2; Yang, Chunhao1,2
刊名JOURNAL OF ORGANIC CHEMISTRY
出版日期2019-05-03
卷号84期号:9页码:5913-5921
ISSN号0022-3263
DOI10.1021/acs.joc.9b00282
通讯作者Zhang, Xiaofei(xiaofeizhang@simm.ac.cn) ; Yang, Chunhao(chyang@simm.ac.cn)
英文摘要A facile and efficient synthetic strategy for the chemoselective synthesis of monocyclic/tricyclic-fused pyrazoles was developed, and it was oriented by different 3-position substituents (H or Cl) on the chromones. The reaction proceeded in a one-pot sequential way with a broad substrate scope and moderate to excellent yields.
WOS关键词INHIBITORS
资助项目NSFC[81872722] ; National Science & Technology Major Project Key New Drug Creation and Manufacturing Program, China[2018ZX09711002] ; SKLDR/SIMM[SIMM1803KF-07]
WOS研究方向Chemistry
语种英语
WOS记录号WOS:000467319600096
出版者AMER CHEMICAL SOC
源URL[http://119.78.100.183/handle/2S10ELR8/289627]  
专题新药研究国家重点实验室
通讯作者Zhang, Xiaofei; Yang, Chunhao
作者单位1.Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, 555 Zuchongzhi Rd, Shanghai 201203, Peoples R China
2.Univ Chinese Acad Sci, Sch Pharm, 19A Yuquan Rd, Beijing 100049, Peoples R China
3.Fudan Univ, Huashan Hosp North, Dept Pharm, 108 Luxiang Rd, Shanghai 201907, Peoples R China
推荐引用方式
GB/T 7714
Dai, Tianzi,Li, Qunyi,Zhang, Xiaofei,et al. Substituent-Oriented Synthesis of Substituted Pyrazoles/Chromeno[3,2-c]pyrazoles via Sequential Reactions of Chromones/3-Chlorochromones and Tosylhydrazones[J]. JOURNAL OF ORGANIC CHEMISTRY,2019,84(9):5913-5921.
APA Dai, Tianzi,Li, Qunyi,Zhang, Xiaofei,&Yang, Chunhao.(2019).Substituent-Oriented Synthesis of Substituted Pyrazoles/Chromeno[3,2-c]pyrazoles via Sequential Reactions of Chromones/3-Chlorochromones and Tosylhydrazones.JOURNAL OF ORGANIC CHEMISTRY,84(9),5913-5921.
MLA Dai, Tianzi,et al."Substituent-Oriented Synthesis of Substituted Pyrazoles/Chromeno[3,2-c]pyrazoles via Sequential Reactions of Chromones/3-Chlorochromones and Tosylhydrazones".JOURNAL OF ORGANIC CHEMISTRY 84.9(2019):5913-5921.

入库方式: OAI收割

来源:上海药物研究所

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