Substituent-Oriented Synthesis of Substituted Pyrazoles/Chromeno[3,2-c]pyrazoles via Sequential Reactions of Chromones/3-Chlorochromones and Tosylhydrazones
文献类型：期刊论文
| 作者 | Dai, Tianzi1,2; Li, Qunyi3; Zhang, Xiaofei1,2; Yang, Chunhao1,2
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| 刊名 | JOURNAL OF ORGANIC CHEMISTRY
 |
| 出版日期 | 2019-05-03 |
| 卷号 | 84期号:9页码:5913-5921 |
| ISSN号 | 0022-3263 |
| DOI | 10.1021/acs.joc.9b00282 |
| 通讯作者 | Zhang, Xiaofei(xiaofeizhang@simm.ac.cn) ; Yang, Chunhao(chyang@simm.ac.cn) |
| 英文摘要 | A facile and efficient synthetic strategy for the chemoselective synthesis of monocyclic/tricyclic-fused pyrazoles was developed, and it was oriented by different 3-position substituents (H or Cl) on the chromones. The reaction proceeded in a one-pot sequential way with a broad substrate scope and moderate to excellent yields. |
| WOS关键词 | INHIBITORS |
| 资助项目 | NSFC[81872722] ; National Science & Technology Major Project Key New Drug Creation and Manufacturing Program, China[2018ZX09711002] ; SKLDR/SIMM[SIMM1803KF-07] |
| WOS研究方向 | Chemistry |
| 语种 | 英语 |
| WOS记录号 | WOS:000467319600096 |
| 出版者 | AMER CHEMICAL SOC |
| 源URL | [http://119.78.100.183/handle/2S10ELR8/289627]  |
| 专题 | 新药研究国家重点实验室 |
| 通讯作者 | Zhang, Xiaofei; Yang, Chunhao |
| 作者单位 | 1.Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, 555 Zuchongzhi Rd, Shanghai 201203, Peoples R China 2.Univ Chinese Acad Sci, Sch Pharm, 19A Yuquan Rd, Beijing 100049, Peoples R China 3.Fudan Univ, Huashan Hosp North, Dept Pharm, 108 Luxiang Rd, Shanghai 201907, Peoples R China |
| 推荐引用方式 GB/T 7714 | Dai, Tianzi,Li, Qunyi,Zhang, Xiaofei,et al. Substituent-Oriented Synthesis of Substituted Pyrazoles/Chromeno[3,2-c]pyrazoles via Sequential Reactions of Chromones/3-Chlorochromones and Tosylhydrazones[J]. JOURNAL OF ORGANIC CHEMISTRY,2019,84(9):5913-5921. |
| APA | Dai, Tianzi,Li, Qunyi,Zhang, Xiaofei,&Yang, Chunhao.(2019).Substituent-Oriented Synthesis of Substituted Pyrazoles/Chromeno[3,2-c]pyrazoles via Sequential Reactions of Chromones/3-Chlorochromones and Tosylhydrazones.JOURNAL OF ORGANIC CHEMISTRY,84(9),5913-5921. |
| MLA | Dai, Tianzi,et al."Substituent-Oriented Synthesis of Substituted Pyrazoles/Chromeno[3,2-c]pyrazoles via Sequential Reactions of Chromones/3-Chlorochromones and Tosylhydrazones".JOURNAL OF ORGANIC CHEMISTRY 84.9(2019):5913-5921. |
入库方式： OAI收割
来源：上海药物研究所
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