Rh(III)-catalyzed selective C7-H functionalization of indolines with 1,3-enynes enables access to six-membered 1,7-fused indolines
文献类型：期刊论文
| 作者 | Shi, Yunkai1,2,3; Chen, Chao3,6; Yang, Yaxi3,4,5 ; Zhou, Bing3,4,5
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| 刊名 | TETRAHEDRON LETTERS
 |
| 出版日期 | 2021-05-25 |
| 卷号 | 72页码:4 |
| 关键词 | C-H activation 1,7-Fused indoline Enynes |
| ISSN号 | 0040-4039 |
| DOI | 10.1016/j.tetlet.2021.153065 |
| 通讯作者 | Zhou, Bing(zhoubing@simm.ac.cn) |
| 英文摘要 | We described herein a Rh(III)-catalyzed C7-selective C-H activation/annulation of indolines with 1,3-enynes to efficiently access various privileged 1,7-fused indolines bearing an all-carbon quaternary stereogenic carbon center. Notably, the resulting products can be readily transformed into 1,7-fused indoles, further widening the C-7 derivatization of indoles and highlighting the synthetic utility of this methodology. (C) 2021 Elsevier Ltd. All rights reserved. |
| WOS关键词 | C-H FUNCTIONALIZATION ; OXIDATIVE ANNULATIONS ; BOND FORMATION ; ACTIVATION ; ALKYNES ; ALKYLATION ; ALKALOIDS |
| 资助项目 | National Natural Science Foundation of China[81973166] ; Youth Innovation Promotion Association[2017333] ; Science and Technology Commission of Shanghai Municipality[18431907100] |
| WOS研究方向 | Chemistry |
| 语种 | 英语 |
| WOS记录号 | WOS:000650994000014 |
| 出版者 | PERGAMON-ELSEVIER SCIENCE LTD |
| 源URL | [http://119.78.100.183/handle/2S10ELR8/297379]  |
| 专题 | 新药研究国家重点实验室 |
| 通讯作者 | Zhou, Bing |
| 作者单位 | 1.Zhengzhou Univ, Inst Pharmaceut Res, Zhengzhou 450001, Peoples R China 2.Zhengzhou Univ, Sch Pharmaceut Sci, Zhengzhou 450001, Peoples R China 3.Chinese Acad Sci, Shanghai Inst Mat Med, State Key Lab Drug Res, 555 Chong Zhi Rd, Shanghai 201203, Peoples R China 4.Univ Chinese Acad Sci, 19 Yuquan Rd, Beijing 100049, Peoples R China 5.Univ Chinese Acad Sci, Sch Pharmaceut Sci & Technol, Hangzhou Inst Adv Study, Hangzhou 310024, Peoples R China 6.Fudan Univ, Sch Pharm, Dept Med Chem, 826 Zhangheng Rd, Shanghai 201203, Peoples R China |
| 推荐引用方式 GB/T 7714 | Shi, Yunkai,Chen, Chao,Yang, Yaxi,et al. Rh(III)-catalyzed selective C7-H functionalization of indolines with 1,3-enynes enables access to six-membered 1,7-fused indolines[J]. TETRAHEDRON LETTERS,2021,72:4. |
| APA | Shi, Yunkai,Chen, Chao,Yang, Yaxi,&Zhou, Bing.(2021).Rh(III)-catalyzed selective C7-H functionalization of indolines with 1,3-enynes enables access to six-membered 1,7-fused indolines.TETRAHEDRON LETTERS,72,4. |
| MLA | Shi, Yunkai,et al."Rh(III)-catalyzed selective C7-H functionalization of indolines with 1,3-enynes enables access to six-membered 1,7-fused indolines".TETRAHEDRON LETTERS 72(2021):4. |
入库方式： OAI收割
来源：上海药物研究所
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