C3-Arylation of indoles with aryl ketones via C-C/C-H activations
文献类型：期刊论文
| 作者 | Guo, Zi-Qiong1; Xu, Hui1; Wang, Xing1,2; Wang, Zhen-Yu3; Ma, Biao1; Dai, Hui-Xiong1,2
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| 刊名 | CHEMICAL COMMUNICATIONS
 |
| 出版日期 | 2021-08-25 |
| 页码 | 4 |
| ISSN号 | 1359-7345 |
| DOI | 10.1039/d1cc03954g |
| 通讯作者 | Dai, Hui-Xiong(hxdai@simm.ac.cn) |
| 英文摘要 | C3-Arylation of indoles with aryl ketones is accomplished via palladium-catalyzed ligand-promoted Ar-C(O) cleavage and subsequent C-H arylation of indole. Various (hetero)aryl ketones are compatible in this reaction, affording the corresponding 3-arylindoles in moderate to good yields. Further introduction of an indole moiety into the natural products desoxyestrone and evodiamine demonstrate the synthetic utility of this protocol. |
| WOS关键词 | REGIOSELECTIVE DIRECT ARYLATION ; CATALYZED C-3 ARYLATION ; METAL-FREE ; PALLADIUM ; FUNCTIONALIZATION ; DERIVATIVES ; COPPER ; LIGHT ; CYCLIZATION ; ALKALOIDS |
| WOS研究方向 | Chemistry |
| 语种 | 英语 |
| WOS记录号 | WOS:000692477200001 |
| 出版者 | ROYAL SOC CHEMISTRY |
| 源URL | [http://119.78.100.183/handle/2S10ELR8/297761]  |
| 专题 | 中国科学院上海药物研究所 |
| 通讯作者 | Dai, Hui-Xiong |
| 作者单位 | 1.Univ Chinese Acad Sci, Chinese Acad Sci Key Lab Receptor Res, Shanghai Inst Mat Med, Shanghai 201203, Peoples R China 2.Univ Chinese Acad Sci, Beijing 100049, Peoples R China 3.Nanjing Univ Chinese Med, Sch Chinese Mat Med, Nanjing 210023, Jiangsu, Peoples R China |
| 推荐引用方式 GB/T 7714 | Guo, Zi-Qiong,Xu, Hui,Wang, Xing,et al. C3-Arylation of indoles with aryl ketones via C-C/C-H activations[J]. CHEMICAL COMMUNICATIONS,2021:4. |
| APA | Guo, Zi-Qiong,Xu, Hui,Wang, Xing,Wang, Zhen-Yu,Ma, Biao,&Dai, Hui-Xiong.(2021).C3-Arylation of indoles with aryl ketones via C-C/C-H activations.CHEMICAL COMMUNICATIONS,4. |
| MLA | Guo, Zi-Qiong,et al."C3-Arylation of indoles with aryl ketones via C-C/C-H activations".CHEMICAL COMMUNICATIONS (2021):4. |
入库方式： OAI收割
来源：上海药物研究所
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