Fluorine-18 labeling by click chemistry: Multiple probes in one pot
文献类型:期刊论文
作者 | Jia, Lina ; Cheng, Zhen ; Shi, Lingli ; Li, Jianbo ; Wang, Cheng ; Jiang, Dawei ; Zhou, Wei(周伟) ; Meng, Hu ; Qi, Yujin(漆玉金) ; Cheng, Dengfeng ; Zhang, Lan(张岚) |
刊名 | APPLIED RADIATION AND ISOTOPES
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出版日期 | 2013 |
卷号 | 75页码:CONCATENATE(Sheet1!I131,-Sheet1!J131) |
ISSN号 | 0969-8043 |
英文摘要 | Click chemistry has been widely applied in drug development including radiopharmaceuticals and has shown great advantages. Here we reported a novel strategy for rapid preparation of multiple F-18 labeled PET probes in one pot using the 'Click Reaction' of Cu(I)-catalyzed Huisgen 1,3-dipolar cycloaddition of terminal alkynes and organic azides (CuAAC). Preliminary results showed its high efficiency and potential for speeding up the preclinical screening of PET probes. (C) 2013 Elsevier Ltd. All rights reserved. |
收录类别 | SCI |
语种 | 英语 |
WOS记录号 | WOS:000317558900012 |
公开日期 | 2014-06-13 |
源URL | [http://ir.sinap.ac.cn/handle/331007/13754] ![]() |
专题 | 上海应用物理研究所_中科院上海应用物理研究所2011-2017年 |
推荐引用方式 GB/T 7714 | Jia, Lina,Cheng, Zhen,Shi, Lingli,et al. Fluorine-18 labeling by click chemistry: Multiple probes in one pot[J]. APPLIED RADIATION AND ISOTOPES,2013,75:CONCATENATE(Sheet1!I131,-Sheet1!J131). |
APA | Jia, Lina.,Cheng, Zhen.,Shi, Lingli.,Li, Jianbo.,Wang, Cheng.,...&Zhang, Lan.(2013).Fluorine-18 labeling by click chemistry: Multiple probes in one pot.APPLIED RADIATION AND ISOTOPES,75,CONCATENATE(Sheet1!I131,-Sheet1!J131). |
MLA | Jia, Lina,et al."Fluorine-18 labeling by click chemistry: Multiple probes in one pot".APPLIED RADIATION AND ISOTOPES 75(2013):CONCATENATE(Sheet1!I131,-Sheet1!J131). |
入库方式: OAI收割
来源:上海应用物理研究所
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