中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
机构
  • 上海药物研究所 [37]
采集方式
  • OAI收割 [37]
内容类型
  • 期刊论文 [37]
发表日期
  • 2017 [37]
学科主题
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浏览/检索结果: 共37条,第1-10条 帮助

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Benzo[c][1,2,5] thiadiazole derivatives: A new class of potent Src homology-2 domain containing protein tyrosine phosphatase-2 (SHP2) inhibitors 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2017, 卷号: 27, 期号: 23, 页码: 5154-5157
作者:  
Wang, Wen-Long;  Chen, Xiao-Yu;  Gao, Ya;  Gao, Li-Xin;  Sheng, Li
  |  收藏  |  浏览/下载:28/0  |  提交时间:2019/01/08
Discovery of novel BET inhibitors by drug repurposing of nitroxoline and its analogues 期刊论文  OAI收割
ORGANIC & BIOMOLECULAR CHEMISTRY, 2017, 卷号: 15, 期号: 44, 页码: 9352-9361
作者:  
Jiang, Hao;  Xing, Jing;  Wang, Chen;  Zhang, Hao;  Yue, Liyan
  |  收藏  |  浏览/下载:108/0  |  提交时间:2019/01/08
Label-free brainwide visualization of senile plaque using cryo-micro-optical sectioning tomography 期刊论文  OAI收割
OPTICS LETTERS, 2017, 卷号: 42, 期号: 21, 页码: 4247-4250
作者:  
Luo, Yilin;  Wang, Anle;  Liu, Mengmeng;  Lei, Tian;  Zhang, Xiaochuan
  |  收藏  |  浏览/下载:31/0  |  提交时间:2019/01/08
Src-dependent phosphorylation of mu-opioid receptor at Tyr(336) modulates opiate withdrawal 期刊论文  OAI收割
EMBO MOLECULAR MEDICINE, 2017, 卷号: 9, 期号: 11, 页码: 1521-1536
作者:  
Zhang, Lei;  Kibaly, Cherkaouia;  Wang, Yu-Jun;  Xu, Chi;  Song, Kyu Young
  |  收藏  |  浏览/下载:34/0  |  提交时间:2019/01/08
Discovery of cycloalkyl-fused N-thiazol-2-yl-benzamides as tissue non-specific glucokinase activators: Design, synthesis, and biological evaluation 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 139, 页码: 128-152
作者:  
Wang, Zhengyu;  Shi, Xiaofan;  Zhang, Huan;  Yu, Liang;  Cheng, Yanhua
  |  收藏  |  浏览/下载:33/0  |  提交时间:2019/01/08
Synthesis and biological evaluation of benzothiazol-based 1,3,4-oxadiazole derivatives as amyloid beta-targeted compounds against Alzheimer's disease 期刊论文  OAI收割
MONATSHEFTE FUR CHEMIE, 2017, 卷号: 148, 期号: 10, 页码: 1807-1815
作者:  
Mei, Wen-wen;  Ji, Sha-sha;  Xiao, Wei;  Wang, Xue-dong;  Jiang, Cheng-shi
  |  收藏  |  浏览/下载:62/0  |  提交时间:2019/01/08
Cyanobacterial peptides as a prototype for the design of cathepsin D inhibitors 期刊论文  OAI收割
JOURNAL OF PEPTIDE SCIENCE, 2017, 卷号: 23, 期号: 9, 页码: 701-706
作者:  
Xu, Hao;  Bao, Keting;  Tang, Shuai;  Ai, Jing;  Hu, Haiyan
  |  收藏  |  浏览/下载:31/0  |  提交时间:2019/01/08
Cytotoxic cassane diterpenoids from the seeds of Caesalpinia sappan 期刊论文  OAI收割
CHINESE CHEMICAL LETTERS, 2017, 卷号: 28, 期号: 8, 页码: 1711-1715
作者:  
Wu, Zheng-Feng;  Bao, Han;  Zhou, Fa-Yang;  Liu, Jing-Xin;  Meng, Fan-Cheng
  |  收藏  |  浏览/下载:17/0  |  提交时间:2019/01/08
Multiple Dose Pharmacokinetics and Safety of Sulcardine Sulfate in Healthy Chinese Male Subjects: An Open-Label Phase I Clinical Study 期刊论文  OAI收割
EUROPEAN JOURNAL OF DRUG METABOLISM AND PHARMACOKINETICS, 2017, 卷号: 42, 期号: 4, 页码: 593-599
作者:  
Wang, Wei;  Qian, Hong-jie;  Xin, Liang;  Zhang, Meng-qi;  Lu, Dong-ying
  |  收藏  |  浏览/下载:12/0  |  提交时间:2019/01/08
The Small GTPase Rac1 Contributes to Extinction of Aversive Memories of Drug Withdrawal by Facilitating GABA(A) Receptor Endocytosis in the vmPFC 期刊论文  OAI收割
JOURNAL OF NEUROSCIENCE, 2017, 卷号: 37, 期号: 30, 页码: 7096-7110
作者:  
Wang, Weisheng;  Ju, Yun-Yue;  Zhou, Qi-Xin;  Tang, Jian-Xin;  Li, Meng
  |  收藏  |  浏览/下载:35/0  |  提交时间:2019/01/08