中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
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上海药物研究所 [243]
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期刊论文 [783]
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Discovery of YFJ-36: Design, Synthesis, and Antibacterial Activities of Catechol-Conjugated β-Lactams against Gram-Negative Bacteria
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 21
作者:
Liu, Fangjun
;
Kou, Qunhuan
;
Li, Hongyuan
;
Cao, Yangzhi
;
Chen, Meng
  |  
收藏
  |  
浏览/下载:0/0
  |  
提交时间:2024/05/22
Design, Synthesis, and Biological Evaluation of Novel Arylomycins against Multidrug-Resistant Gram-Negative Bacteria
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 25
作者:
Zhang, Yinyong
;
Zhang, Dan
;
Zhao, Wenhao
;
Li, Hongyuan
;
Lu, Zhengyu
  |  
收藏
  |  
浏览/下载:0/0
  |  
提交时间:2024/05/22
Design and Synthesis of Cyclolipopeptide Mimics of Dysoxylactam A and Evaluation of the Reversing Potencies against P-Glycoprotein-Mediated Multidrug Resistance
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 6, 页码: 4560-4582
作者:
Yang, Guan-Zhou
;
Wang, Lei
;
Gao, Kun
;
Zhu, Xi
;
Lou, Li-Guang
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2024/05/07
Identification of a Novel Selective CDK9 Inhibitor for the Treatment of CRC: Design, Synthesis, and Biological Activity Evaluation
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 6, 页码: 4739-4756
作者:
Zhong, Ye
;
Xu, Jing
;
Zhou, Ruochen
;
Tang, Li
;
Ding, Shaoyue
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2024/05/07
Design, synthesis and biological evaluation of thiazolyl-halogenated pyrroles or pyrazoles as novel antibacterial and antibiofilm agents
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 268, 页码: 9
作者:
Zhong, Yuanchen
;
Liu, Huan
;
Chen, Feifei
;
He, Qian
;
Zhang, Xiaofei
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2024/05/07
Pyrrolomycin analogues
Antibacterial agents
Anti-biofilm
Drug -resistant bacteria
Thiazole
Functional structural domain synthesis of anti-pancreatic carcinoma pectin-like polysaccharide RN1
期刊论文
OAI收割
CARBOHYDRATE POLYMERS, 2024, 卷号: 327, 页码: 11
作者:
Cai, Deqin
;
He, Fei
;
Wu, Shengjie
;
Wang, Zixuan
;
Bian, Ya
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2024/02/19
Polysaccharide
Pectin
Functional structural domain
Pancreatic cancer
Glycan synthesis
RN1
Discovery of Pyrido[2,3-
d
]pyrimidin-7-one Derivatives as Highly Potent and Efficacious Ectonucleotide Pyrophosphatase/Phosphodiesterase 1 (ENPP1) Inhibitors for Cancer Treatment
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 5, 页码: 3986-4006
作者:
Sun, Yaoliang
;
Chen, Manman
;
Han, Yuyan
;
Li, Weiqiang
;
Ma, Xiaoyu
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收藏
  |  
浏览/下载:1/0
  |  
提交时间:2024/05/07
Synthesis and Characterization of Slow-Release Chitosan Oligosaccharide Pyridine Schiff Base Copper Complexes with Antifungal Activity
期刊论文
OAI收割
JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY, 2024, 卷号: 72, 期号: 8, 页码: 3872-3883
作者:
Liu, Weixiang
;
Qin, Yukun
;
Liu, Song
;
Xing, Ronge
;
Yu, Huahua
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2024/04/07
antifungal
chitosan oligosaccharide
coppercomplex
Schiff base
slow-release
7-Dehydrocholesterol dictates ferroptosis sensitivity
期刊论文
OAI收割
NATURE, 2024, 卷号: 626, 期号: 7998, 页码: 29
作者:
Li, Yaxu
;
Ran, Qiao
;
Duan, Qiuhui
;
Jin, Jiali
;
Wang, Yanjin
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2024/04/09
Design and synthesis of cantharidin derivative DCZ5418 as a TRIP13 inhibitor with anti-multiple myeloma activity
in
vitro
and
in
vivo
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2024, 卷号: 98, 页码: 7
作者:
Dong, Sanfeng
;
Hu, Ke
;
Shi, Yulong
;
Wang, Guanli
;
Yu, Dandan
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2024/02/19
Multiple myeloma
TRIP13 inhibitor
Cantharidin
DCZ5418
DCZ0415