中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共113条,第1-10条 帮助

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Structure-Based Drug Design of 2-Amino-[1,1′-biphenyl]-3-carboxamide Derivatives as Selective PKMYT1 Inhibitors for the Treatment of CCNE1-Amplified Breast Cancer 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 21
作者:  
Wang, Chaofan;  Fang, Yan;  Zhou, Ziqin;  Liu, Zhuoheng;  Feng, Fang
  |  收藏  |  浏览/下载:17/0  |  提交时间:2024/09/26
Discovery of HCD3514 as a potent EGFR inhibitor against C797S mutation in vitro and in vivo 期刊论文  OAI收割
JOURNAL OF CANCER, 2023, 卷号: 14, 期号: 1, 页码: 152-162
作者:  
Lai, Mengzhen;  Zhang, Tao;  Chen, Hao;  Song, Peiran;  Tong, Linjiang
  |  收藏  |  浏览/下载:132/0  |  提交时间:2023/04/10
Conformational Constrained 4-(1-Sulfonyl-3-indol)yl-2-phenylaminopyrimidine Derivatives as New Fourth-GenerationEpidermal Growth Factor Receptor Inhibitors Targeting T790M/C797S Mutations 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 9, 页码: 6840-6858
作者:  
Chen, Hao;  Lai, Mengzhen;  Zhang, Tao;  Chen, Yuqing;  Tong, Linjiang
  |  收藏  |  浏览/下载:30/0  |  提交时间:2024/03/21
Conformational Constrained 4-(1-Sulfonyl-3-indol)yl-2-phenylaminopyrimidine Derivatives as New Fourth-GenerationEpidermal Growth Factor Receptor Inhibitors Targeting T790M/C797S Mutations br 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 9, 页码: 6840-6858
作者:  
Chen, Hao;  Lai, Mengzhen;  Zhang, Tao;  Chen, Yuqing;  Tong, Linjiang
  |  收藏  |  浏览/下载:41/0  |  提交时间:2022/08/16
The p300 Inhibitor A-485 Exerts Antitumor Activity in Growth Hormone Pituitary Adenoma 期刊论文  OAI收割
JOURNAL OF CLINICAL ENDOCRINOLOGY & METABOLISM, 2022, 页码: 10
作者:  
Ji, Chenxing;  Xu, Wen;  Ding, Hong;  Chen, Zhengyuan;  Shi, Chengzhang
  |  收藏  |  浏览/下载:62/0  |  提交时间:2022/06/15
Optimization of Brigatinib as New Wild-Type Sparing Inhibitors of EGFR(T790M/C797S) Mutants 期刊论文  OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2022, 页码: 7
作者:  
Li, Shan;  Zhang, Tao;  Zhu, Su-Jie;  Lei, Chong;  Lai, Mengzhen
  |  收藏  |  浏览/下载:54/0  |  提交时间:2022/06/15
LS-106, a novel EGFR inhibitor targeting C797S, exhibits antitumor activities both in vitro and in vivo 期刊论文  OAI收割
CANCER SCIENCE, 2021, 页码: 12
作者:  
Liu, Yingqiang;  Lai, Mengzhen;  Li, Shan;  Wang, Yanan;  Feng, Fang
  |  收藏  |  浏览/下载:114/0  |  提交时间:2022/01/18
Electron-ion collider in China 期刊论文  OAI收割
FRONTIERS OF PHYSICS, 2021, 卷号: 16, 期号: 6, 页码: 78
作者:  
Anderle, Daniele P.;  Bertone, Valerio;  Cao, Xu;  Chang, Lei;  Chang, Ningbo
  |  收藏  |  浏览/下载:132/0  |  提交时间:2021/12/08
Effect of FeCo2S4 on electrocatalytic I-3(-) reduction: Theoretical and experimental aspects 期刊论文  OAI收割
CHEMICAL ENGINEERING JOURNAL, 2021, 卷号: 424
作者:  
Zhang, Xiaoyun;  Chen, Pin;  Yang, Fan;  Wang, Lian;  Yin, Jie
  |  收藏  |  浏览/下载:73/0  |  提交时间:2022/01/10
Maize is stressed by salt rather than water under drip irrigation with soil matric potential higher than-50 kPa in an arid saline area 期刊论文  OAI收割
JOURNAL OF AGRONOMY AND CROP SCIENCE, 2021, 页码: 15
作者:  
Zhang, Tibin;  Ji, Xiangxiang;  Zhan, Xiaoyun;  Ding, Yuntao;  Zou, Yufeng
  |  收藏  |  浏览/下载:57/0  |  提交时间:2021/06/10