中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共25条,第1-10条 帮助

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Novel thieno[2,3-b]quinoline-procaine hybrid molecules: A new class of allosteric SHP-1 activators evolved from PTP1B inhibitors 期刊论文  OAI收割
CHINESE CHEMICAL LETTERS, 2023, 卷号: 34, 期号: 8, 页码: 6
作者:  
Xu, Lei;  Xuyan, Xuyang;  Minmi, Minmin;  Wang, Zhiji;  Shee, Chao
  |  收藏  |  浏览/下载:48/0  |  提交时间:2023/10/17
Discovery of a Novel Androgen Receptor Antagonist Manifesting Evidence to Disrupt the Dimerization of the Ligand-Binding Domain via Attenuating the Hydrogen-Bonding Network Between the Two Monomers 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64
作者:  
Fu, Weitao;  Zhang, Minkui;  Liao, Jianing;  Tang, Qing;  Lei, Yixuan
  |  收藏  |  浏览/下载:34/0  |  提交时间:2022/03/21
Structural insights into ligand recognition and activation of the melanocortin-4 receptor 期刊论文  OAI收割
CELL RESEARCH, 2021, 页码: 13
作者:  
Zhang, Huibing;  Chen, Li-Nan;  Yang, Dehua;  Mao, Chunyou;  Shen, Qingya
  |  收藏  |  浏览/下载:79/0  |  提交时间:2021/11/04
Discovery of Novel Androgen Receptor Ligands by Structure-based Virtual Screening and Bioassays 期刊论文  OAI收割
GENOMICS PROTEOMICS & BIOINFORMATICS, 2019, 卷号: 16, 期号: 6, 页码: 416-427
作者:  
Hou, Tingjun;  Li, Dan;  Chang, Shan;  Xu, Lei;  Sun, Huiyong
  |  收藏  |  浏览/下载:277/0  |  提交时间:2019/06/24
Communication between the Ligand-Binding Pocket and the Activation Function-2 Domain of Androgen Receptor Revealed by Molecular Dynamics Simulations 期刊论文  OAI收割
JOURNAL OF CHEMICAL INFORMATION AND MODELING, 2019, 卷号: 59, 期号: 2, 页码: 842-857
作者:  
Hou, Tingjun;  Li, Youyong;  Yu, Huidong;  Li, Dan;  Liu, Hui
  |  收藏  |  浏览/下载:82/0  |  提交时间:2019/06/24
锦屏深地核天体物理实验(JUNA)进展 期刊论文  OAI收割
原子能科学技术, 2019, 卷号: 53.0, 期号: 010, 页码: 1729
作者:  
柳卫平;  李志宏;  何建军;  唐晓东;  连钢
  |  收藏  |  浏览/下载:97/0  |  提交时间:2021/12/06
Molecular Dynamics Simulations Revealed the Regulation of Ligands to the Interactions between Androgen Receptor and Its Coactivator 期刊论文  OAI收割
JOURNAL OF CHEMICAL INFORMATION AND MODELING, 2018, 卷号: 58, 期号: 8, 页码: 1652-1661
作者:  
Liu, Na;  Zhou, Wenfang;  Guo, Yue;  Wang, Junmei;  Fu, Weitao
  |  收藏  |  浏览/下载:81/0  |  提交时间:2018/11/05
discoveryofnovelandrogenreceptorligandsbystructurebasedvirtualscreeningandbioassays 期刊论文  OAI收割
genomicsproteomicsbioinformatics, 2018, 卷号: 16, 期号: 6, 页码: 416
作者:  
Zhou Wenfang;  Duan Mojie;  Fu Weitao;  Pang Jinping;  Tang Qin
  |  收藏  |  浏览/下载:36/0  |  提交时间:2020/01/14