中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
首页
机构
成果
学者
登录
注册
登陆
×
验证码:
换一张
忘记密码?
记住我
×
校外用户登录
CAS IR Grid
机构
上海药物研究所 [33]
心理研究所 [3]
化学研究所 [2]
成都生物研究所 [1]
国家天文台 [1]
高能物理研究所 [1]
更多
采集方式
OAI收割 [41]
iSwitch采集 [2]
内容类型
期刊论文 [42]
学位论文 [1]
发表日期
2024 [1]
2023 [2]
2022 [4]
2021 [2]
2020 [2]
2019 [1]
更多
学科主题
Energy & F... [1]
Engineerin... [1]
Plant Scie... [1]
创伤心理学 [1]
医学心理学 [1]
筛选
浏览/检索结果:
共43条,第1-10条
帮助
条数/页:
5
10
15
20
25
30
35
40
45
50
55
60
65
70
75
80
85
90
95
100
排序方式:
请选择
提交时间升序
提交时间降序
题名升序
题名降序
作者升序
作者降序
发表日期升序
发表日期降序
A novel phthalazinone derivative as a capsid assembly modulator inhibits hepatitis B virus expression
期刊论文
OAI收割
ANTIVIRAL RESEARCH, 2024, 卷号: 221, 页码: 14
作者:
Yang, Li
;
Gong, Ying
;
Liu, Feifei
;
Chen, Wuhong
;
Wang, Xinran
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2024/02/19
Hepatitis B virus
Capsid assembly
Phthalazinone derivatives
Apoptosis
A prodrug of the capsid assembly modulator improved druggability and lowing HBsAg and HBeAg for the treatment of chronic hepatitis B
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 257, 页码: 8
作者:
Chen, Wuhong
;
Gong, Ying
;
Long, Guozhang
;
Wang, Xinran
;
Yang, Yurong
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2023/10/17
HBV
Capsid assembly modulators
Prodrug
Hepatitis B surface antigen
Discovery of (S)-N-(2-Amino-4-fluorophenyl)-4-(1-(3-(4-((dimethylamino)methyl)phenyl)-6-oxopyridazin-1(6H)-yl)ethyl)benzamide as Potent Class I Selective HDAC Inhibitor for Oral Anticancer Drug Candidate
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 10, 页码: 7016-7037
作者:
Li, Daqiang
;
Zhang, Zhuo
;
Li, Yalei
;
Wang, Xinyi
;
Zhong, Hanyue
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2023/10/17
Discovery of potent ebola entry inhibitors with (3S,4aS,8aS)-2-(3-amino-2-hydroxypropyl) decahydroisoquinoline-3-carboxamide scaffold
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 240, 页码: 12
作者:
Han, Sheng
;
Li, Heng
;
Chen, Weixiong
;
Yang, Li
;
Tong, Xiankun
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2022/11/11
Ebola virus
Entry inhibitor
Structural optimization
Experimental study on hydraulic fracturing behavior of frozen clayey silt and hydrate-bearing clayey silt
期刊论文
OAI收割
FUEL, 2022, 卷号: 322, 期号: -, 页码: -
作者:
Ma, Xiaolong
;
Jiang, Dandan
;
Sun, Youhong
;
Li, Shengli
  |  
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2023/08/02
Clayey silt
Gas hydrate
Hydraulic fracturing
Fracture propagation
Fracture initiation
Fracture morphology
Adjusted degradation of BRD4 S and BRD4 L based on fine structural modifications of the pyrrolopyridone scaffold
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 236, 页码: 14
作者:
Chen, Jingjing
;
He, Huixin
;
Wei, Aihuan
;
Li, Yalei
;
Cheng, Gang
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2022/08/16
PROTAC
Pyrrolopyridone
BRD4 S
Selectivity
Discovery of highly potent SARS-CoV-2 M-pro inhibitors based on benzoisothiazolone scaffold
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2022, 卷号: 58, 页码: 6
作者:
Chen, Weixiong
;
Feng, Bo
;
Han, Sheng
;
Wang, Peipei
;
Chen, Wuhong
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2022/06/15
COVID-19
SARS-CoV-2
Main protease inhibitors
Benzoisothiazolone
Discovery of Potent Antiallergic Agents Based on an o-Aminopyridinyl Alkynyl Scaffold
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 18, 页码: 13588-13603
作者:
Xie, Zhicheng
;
Xiang, Caigui
;
Li, Xin
;
Fan, Chen
;
Chen, Taiwen
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2024/03/21
Discovery of selective HDAC/BRD4 dual inhibitors as epigenetic probes
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 209, 页码: 20
作者:
Chen, Jingjing
;
Li, Yalei
;
Zhang, Jie
;
Zhang, Minmin
;
Wei, Aihuan
  |  
收藏
  |  
浏览/下载:59/0
  |  
提交时间:2021/05/24
HDAC
BRD4
Selective dual inhibitors
Anticancer
Targeted Proteomics Combined with Affinity Mass Spectrometry Analysis Reveals Antagonist E7 Acts As an Intracellular Covalent Ligand of Orphan Receptor GPR52
期刊论文
OAI收割
ACS CHEMICAL BIOLOGY, 2020, 卷号: 15, 期号: 12, 页码: 3275-3284
作者:
Ma, Mengna
;
Guo, Shimeng
;
Lin, Xi
;
Li, Shanshan
;
Wu, Yiran
  |  
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2021/05/24