中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共107条,第1-10条 帮助

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Design, synthesis, and evaluation of Menin-targeting compounds for the treatment of acute Myelocytic leukemia (AML) 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 296, 页码: 17
作者:  
Mo, Jun;  Wang, Yuxian;  Pan, Youlu;  Xiao, Qitao;  Zhao, Jinyi
  |  收藏  |  浏览/下载:4/0  |  提交时间:2025/08/20
Discovery of a potential hematologic malignancies therapy: Selective and potent HDAC7 PROTAC degrader targeting non-enzymatic function 期刊论文  OAI收割
ACTA PHARMACEUTICA SINICA B, 2025, 卷号: 15, 期号: 3, 页码: 1659-1679
作者:  
Jin, Yuheng;  Qi, Xuxin;  Yu, Xiaoli;  Cheng, Xirui;  Chen, Boya
  |  收藏  |  浏览/下载:20/0  |  提交时间:2025/06/23
Discovery of KW0113 as a First and Effective PROTAC Degrader of DNMT1 Protein 期刊论文  OAI收割
CHEMMEDCHEM, 2024, 页码: 16
作者:  
Wang, Huihui;  Wang, Zhaoliang;  Hu, Linghao;  Yang, Bingjie;  Zong, Liangyi
  |  收藏  |  浏览/下载:31/0  |  提交时间:2024/12/16
Discovery of a Highly Potent, Selective and Efficacious USP7 Degrader for the Treatment of Acute Lymphoblastic Leukemia 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 20
作者:  
Xu, Miaomiao;  Fu, Jingfeng;  Pei, Yuan;  Li, Mengna;  Kan, Weijuan
  |  收藏  |  浏览/下载:33/0  |  提交时间:2024/08/22
Design, Synthesis, and Biological Evaluation of 2,4-Diaminopyrimidine Derivatives as Potent CDK7 Inhibitors 期刊论文  OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2024, 页码: 8
作者:  
Zhang, Hualin;  Tu, Yutong;  Tao, Zhaofan;  Gao, Lixin;  Huang, Shengjie
  |  收藏  |  浏览/下载:32/0  |  提交时间:2024/08/22
Discovery of a Highly Potent and Selective BRD9 PROTAC Degrader Based on E3 Binder Investigation for the Treatment of Hematological Tumors 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 28
作者:  
Duan, Haiting
  |  收藏  |  浏览/下载:33/0  |  提交时间:2024/08/20
Discovery of potent small molecule ubiquitin-specific protease 10 inhibitors with anti-hepatocellular carcinoma activity through regulating YAP expression 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 272, 页码: 21
作者:  
Lu, Yang;  Gao, Jian
  |  收藏  |  浏览/下载:27/0  |  提交时间:2024/07/12
Structured diary introspection training: A kind of critical thinking training method can enhance the Pro-C creativity of interior designers 期刊论文  OAI收割
THINKING SKILLS AND CREATIVITY, 2024, 卷号: 52, 页码: 14
作者:  
Li, Hao;  Yang, Liu;  Wang, Ting;  Xiao, Ruoyu;  Song, Lili
  |  收藏  |  浏览/下载:29/0  |  提交时间:2024/06/29
Integrative proteogenomic and pharmacological landscape of acute myeloid leukaemia 期刊论文  OAI收割
SCIENCE BULLETIN, 2024, 卷号: 70, 期号: 7, 页码: 1051-1056
作者:  
Wang, Hanlin;  Tang, Gusheng;  Ye, Yunfei;  Li, Jia;  Xu, Jun-Yu
  |  收藏  |  浏览/下载:12/0  |  提交时间:2025/06/04
Discovery of potent PROTAC degraders of Pin1 for the treatment of acute myeloid leukemia 期刊论文  OAI收割
CHEMICAL SCIENCE, 2024, 卷号: 15, 期号: 13, 页码: 5027-5035
作者:  
Shi, Yunkai;  Liu, Minmin;  Li, Mengna;  Mao, Yiwen;  Ma, Jingkun
  |  收藏  |  浏览/下载:51/0  |  提交时间:2024/05/07