中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共19条,第1-10条 帮助

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Design, Synthesis, and biological evaluation of 7H-Pyrrolo[2,3-d] pyrimidines as potent HPK1 kinase inhibitors 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2025, 卷号: 119, 页码: 13
作者:  
Wu, Feifei;  Li, Huiyu;  Li, Weiqiang;  Zhang, Laishun;  An, Qi
  |  收藏  |  浏览/下载:8/0  |  提交时间:2025/04/01
Design, Synthesis, and Pharmacological Evaluation of Quinazoline and Quinoline Derivatives as Potent ENPP1 Inhibitors for Cancer Immunotherapy 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 页码: 18
作者:  
He, Jie;  Ma, Xiaoyu;  Sun, Jia;  Chen, Manman;  Xu, Lan
  |  收藏  |  浏览/下载:9/0  |  提交时间:2025/04/01
Selective Degradation of TEADs by a PROTAC Molecule Exhibited Robust Anticancer Efficacy In Vitro and In Vivo 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 页码: 25
作者:  
Lu, Yuhang;  Yan, Ziqin;  Sun, Jiaqi;  Wang, Chenxu;  Xu, Lan
  |  收藏  |  浏览/下载:16/0  |  提交时间:2025/04/01
METI: deep profiling of tumor ecosystems by integrating cell morphology and spatial transcriptomics 期刊论文  OAI收割
NATURE COMMUNICATIONS, 2024, 卷号: 15
作者:  
Jiang, Jiahui;  Liu, Yunhe;  Qin, Jiangjiang;  Chen, Jianfeng;  Wu, Jingjing
  |  收藏  |  浏览/下载:13/0  |  提交时间:2024/11/20
Discovery of Pyrido[2,3-d]pyrimidin-7-one Derivatives as Highly Potent and Efficacious Ectonucleotide Pyrophosphatase/Phosphodiesterase 1 (ENPP1) Inhibitors for Cancer Treatment 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 5, 页码: 3986-4006
作者:  
Sun, Yaoliang;  Chen, Manman;  Han, Yuyan;  Li, Weiqiang;  Ma, Xiaoyu
  |  收藏  |  浏览/下载:24/0  |  提交时间:2024/05/07
Discovery, SAR Study of GST Inhibitors from a Novel Quinazolin-4(1H)-one Focused DNA-Encoded Library 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 页码: 15
作者:  
Wen, Xin;  Zhang, Minmin;  Duan, Zhiqiang;  Suo, Yanrui;  Lu, Weiwei
  |  收藏  |  浏览/下载:49/0  |  提交时间:2023/10/17
Discovery of 7H-Pyrrolo[2,3-d]pyrimidine Derivatives as potent hematopoietic progenitor kinase 1 (HPK1) inhibitors 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 254, 页码: 15
作者:  
Wu, Feifei;  Li, Huiyu;  An, Qi;  Sun, Yaoliang;  Yu, Jinghua
  |  收藏  |  浏览/下载:26/0  |  提交时间:2023/10/17
Intact regulation of G1/S transition renders esophageal squamous cell carcinoma sensitive to PI3Kα inhibitors 期刊论文  OAI收割
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2023, 卷号: 8, 期号: 1, 页码: 153
作者:  
Zhang, Xu;  Wang, Yuxiang;  Zhang, Xi;  Shen, Yanyan;  Yang, Kang
  |  收藏  |  浏览/下载:25/0  |  提交时间:2024/03/27
基于紫外可见光谱技术和色素组成区分橄榄油与其他食用油 期刊论文  OAI收割
食品安全质量检测学报, 2023, 卷号: 14, 期号: 5, 页码: 130-137
作者:  
卢聪慧;  胥玲花;  黄新异;  裴栋;  邸多隆
  |  收藏  |  浏览/下载:8/0  |  提交时间:2023/11/06
Genome-wide gain-of-function screening identifies EZH2 mediating resistance to PI3K alpha inhibitors in oesophageal squamous cell carcinoma 期刊论文  OAI收割
CLINICAL AND TRANSLATIONAL MEDICINE, 2022, 卷号: 12, 期号: 5, 页码: 17
作者:  
Xing, Hui;  Gao, Mengshi;  Wang, Yuxiang;  Zhang, Xu;  Shi, Jiajie
  |  收藏  |  浏览/下载:55/0  |  提交时间:2022/08/16