中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
金属研究所 [6]
上海药物研究所 [6]
昆明植物研究所 [3]
合肥物质科学研究院 [2]
天津工业生物技术研究... [2]
西双版纳热带植物园 [1]
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OAI收割 [23]
内容类型
期刊论文 [23]
发表日期
2024 [4]
2023 [2]
2022 [4]
2021 [4]
2020 [1]
2019 [1]
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Multidisci... [1]
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Discovery of a Potent, selective and orally bioavailable CDK9 degrader for targeting transcription regulation in Triple-Negative breast cancer
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2024, 卷号: 153, 页码: 16
作者:
Nie, Hui-Jun
;
Li, Ben-Fu
;
Sun, Jingya
;
Yuan, Yali
;
Zhang, Zhi-Gao
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2024/11/26
Triple-negative breast cancer
Targeting transcription regulation
Orally bioavailable degrader
PROTAC
Cyclin-dependent Kinase 9
Improving ellipse fitting via multi-scale smoothing and key-point searching
期刊论文
OAI收割
PATTERN RECOGNITION, 2024, 卷号: 151, 页码: 15
作者:
Chen, Xiao-Diao
;
Qian, Cheng
;
Zhao, Mingyang
;
Yong, Jun -Hai
;
Yan, Dong-Ming
  |  
收藏
  |  
浏览/下载:41/0
  |  
提交时间:2024/07/03
Ellipse fitting
Least-squares
RANSAC
Multi-scale smoothing
Key-point searching
Rapid summer Russian Arctic sea-ice loss enhances the risk of recent Eastern Siberian wildfires
期刊论文
OAI收割
NATURE COMMUNICATIONS, 2024, 卷号: 15, 期号: 1, 页码: 17
作者:
Luo, Binhe
;
Luo, Dehai
;
Dai, Aiguo
;
Xiao, Cunde
;
Simmonds, Ian
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2024/09/02
Discovery of Orally Bioavailable and Potent CDK9 Inhibitors for Targeting Transcription Regulation in Triple-Negative Breast Cancer
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 12, 页码: 10035-10056
作者:
Wang, Wen-Jing
;
Gao, Lixin
;
Wang, Simei
;
Huang, Wensi
;
Meng, Xin-Yu
  |  
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2024/08/20
Atomic-Dispersed Rh Enables Efficient Catalytic Nitrile Hydrogenation: Size Effect and Metal-Dependent Effect
期刊论文
OAI收割
ACS CATALYSIS, 2023, 页码: 8354-8361
作者:
Chen, Jiawei
;
Jiao, Yueyue
;
Qin, Xuetao
;
Cai, Xiangbin
;
Wang, Maolin
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2024/01/07
nitriles
hydrogenation
Rh catalyst
atomically dispersed
amines
Structure-dependence and metal-dependence on atomically dispersed Ir catalysts for efficient n-butane dehydrogenation
期刊论文
OAI收割
NATURE COMMUNICATIONS, 2023, 卷号: 14, 期号: 1, 页码: 11
作者:
Chen, Xiaowen
;
Qin, Xuetao
;
Jiao, Yueyue
;
Peng, Mi
;
Diao, Jiangyong
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2024/01/07
A potent PGK1 antagonist reveals PGK1 regulates the production of IL-1 beta and IL-6
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2022, 卷号: 12, 期号: 11, 页码: 4180-4192
作者:
Liao, Liping
;
Dang, Wenzhen
;
Lin, Tingting
;
Yu, Jinghua
;
Liu, Tonghai
  |  
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2023/04/10
Glycolysis
Phosphoglycerate kinase 1
Macrophages
NRF2
Inflammation
Absorption, distribution, metabolism, and excretion of [C-14]Mefuparib (CVL218), a novel PARP1/2 inhibitor, in rats
期刊论文
OAI收割
CANCER CHEMOTHERAPY AND PHARMACOLOGY, 2022, 页码: 12
作者:
Li, Xin-mei
;
Zheng, Yuan-dong
;
Zhang, Yi-fan
;
Huan, Xia-juan
;
Yang, Chen
  |  
收藏
  |  
浏览/下载:42/0
  |  
提交时间:2022/12/13
[C-14]Mefuparib
Mefuparib (CVL218)
Blood-brain barrier
Mass balance
Tissue distribution
GastroPlus simulation
Fully Exposed Platinum Clusters on a Nanodiamond/Graphene Hybrid for Efficient Low-Temperature CO Oxidation
期刊论文
OAI收割
ACS CATALYSIS, 2022, 页码: 9
作者:
Jia, Zhimin
;
Peng, Mi
;
Cai, Xiangbin
;
Chen, Yunlei
;
Chen, Xiaowen
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2023/05/09
CO oxidation
nanodiamond
Pt catalyst
atomically dispersed
cluster
Fully Exposed Platinum Clusters on a Nanodiamond/Graphene Hybrid for Efficient Low-Temperature CO Oxidation
期刊论文
OAI收割
ACS CATALYSIS, 2022, 页码: 9
作者:
Jia, Zhimin
;
Peng, Mi
;
Cai, Xiangbin
;
Chen, Yunlei
;
Chen, Xiaowen
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2023/05/09
CO oxidation
nanodiamond
Pt catalyst
atomically dispersed
cluster