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Chinese Academy of Sciences Institutional Repositories Grid
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Design and synthesis of CDK9/EZH2 dual-target inhibitors to achieve synergistic antitumor effects
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 294, 页码: 14
作者:
Tian, Lina
;
Xiao, Jian
  |  
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2025/08/20
CDK9
EZH2
Dual target inhibitor
DLBCL
Efficient and high-quality algorithms for the layout optimization of wave energy converter arrays based on many-body expansion
期刊论文
OAI收割
OCEAN ENGINEERING, 2025, 卷号: 333, 页码: 20
作者:
Chen, Jiahao
;
Cui, Zhehua
;
Kang, Yuanshun
;
Li, Lijun
;
Zeng, Xiaohui
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2025/07/22
Layout optimization
Wave energy converters
Many-body expansion
Guiding precision medicine strategy for intravenous ginsenosides via pharmacokinetic-informed bioinformatic approaches: a study on XueShuanTong
期刊论文
OAI收割
PHYTOMEDICINE, 2025, 卷号: 143, 页码: 18
作者:
Jia, Wei-Wei
;
Tian, Nan-Nan
;
Song, Zi-Jing
;
Lan, Xiao-Fang
;
Yang, Xi-He
  |  
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2025/08/20
Precision medicine
Physiologically based pharmacokinetic model
Ginsenoside
Albumin-facilitated dissociation
Drug interaction
Drug transporter
Hepatic impairment
Benzothiazole amide analogues as antagonists of TRPC 6 channels: A therapeutic approach for kidney fibrosis
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 291, 页码: 16
作者:
Ren, Chunlin
;
Xu, Qiding
;
Luo, Qiusi
;
Qiao, Xue
;
Ding, Taotao
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2025/06/23
Transient receptor potential canonical 6
channels
Antagonist
Renal fibrosis
Benzothiazole derivatives
Unilateral ureteral obstruction
Opposed flame spread over a thermally-thin charring material under varied flow velocities and ambient pressures in a narrow channel apparatus
期刊论文
OAI收割
FIRE SAFETY JOURNAL, 2025, 卷号: 154, 页码: 14
作者:
Wang, Wenlong
;
Tao, Shangqing
;
Fang, Jun
;
Zeng, Yi
;
Wang, Jiyun
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2025/06/23
Narrow channel
Buoyancy suppression
Periodic fingering flamelets
Global equivalence ratio
Flammability boundary
Study of ultra-high-energy gamma-ray source 1LHAASO J0056+6346u and its possible origins
期刊论文
OAI收割
SCIENCE CHINA-PHYSICS MECHANICS & ASTRONOMY, 2025, 卷号: 68, 期号: 7
作者:
Cao, Zhen
;
Aharonian, F.
;
Axikegu
;
Bai, Y. X.
;
Bao, Y. W.
  |  
收藏
  |  
浏览/下载:36/0
  |  
提交时间:2025/06/10
gamma rays
cosmic rays
supernova remnant
young massive cluster
pulsar
Risk assessment of CYP3A induction by ginsenoside's metabolites from oral Panax notoginseng (sanqi) extract
期刊论文
OAI收割
JOURNAL OF ETHNOPHARMACOLOGY, 2025, 卷号: 349, 页码: 11
作者:
Deng, Yang
;
Du, Jing
;
He, Xin
;
Dong, Yan-Xi
;
Wang, Xiao-Lei
  |  
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2025/08/20
Panax notoginseng
Ginsenoside
Intestinal microbiota
CYP3A induction
Drug interaction
Contrastive learning-based drug screening model for GluN1/GluN3A inhibitors
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2025, 页码: 13
作者:
Li, Kun
;
Zeng, Yue
;
Xiong, Yi-da
;
Wu, Hao-chen
;
Fang, Sui
  |  
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2025/08/20
drug-target affinity prediction
virtual screening
contrastive learning
graph neural network
N
-methyl-
D
-aspartate (NMDA) receptors
GluN3A subunit.
Discovery of novel GluN1/GluN3A NMDA receptor inhibitors using a deep learning-based method
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2025, 页码: 8
作者:
Wang, Shi-hang
;
Zeng, Yue
;
Yang, Hao
;
Tian, Si-yuan
;
Zhou, Yong-qi
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2025/07/25
N
-methyl-
D
-aspartate receptors
GluN1/GluN3A
ligand-based virtual screening
scaffold hopping
deep learning
GeminiMol
Enhancing fluorescent probe design through multilayer interaction convolutional networks: advancing biosensing and bioimaging precision
期刊论文
OAI收割
CHEMICAL SCIENCE, 2025, 页码: 8
作者:
Ma, Gongcheng
;
Ding, Qihang
;
Zhang, Yuding
;
Zeng, Xiaodong
;
Zhu, Kai
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2025/06/23