中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [11]
自动化研究所 [3]
新疆理化技术研究所 [1]
水生生物研究所 [1]
武汉植物园 [1]
植物研究所 [1]
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OAI收割 [20]
内容类型
期刊论文 [17]
会议论文 [3]
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2025 [2]
2024 [2]
2023 [2]
2022 [1]
2021 [2]
2020 [1]
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学科主题
Biochemist... [1]
Multidisci... [1]
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Discovery of a potential hematologic malignancies therapy: Selective and potent HDAC7 PROTAC degrader targeting non-enzymatic function
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2025, 卷号: 15, 期号: 3, 页码: 1659-1679
作者:
Jin, Yuheng
;
Qi, Xuxin
;
Yu, Xiaoli
;
Cheng, Xirui
;
Chen, Boya
  |  
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2025/06/23
HDAC7
PROTAC
Selectivity
Hematologic malignancies
Non-enzymatic function
Auto-RapTAC: A Versatile and Sustainable Platform for the Automated Rapid Synthesis and Evaluation of PROTAC
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 页码: 15
作者:
Chen, Jiexuan
;
Wu, Mingfei
;
Mo, Jun
;
Hong, Ju
;
Wang, Wei
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2025/04/01
Discovery of potent small molecule ubiquitin-specific protease 10 inhibitors with anti-hepatocellular carcinoma activity through regulating YAP expression
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 272, 页码: 21
作者:
Lu, Yang
;
Gao, Jian
;
Wang, Peipei
;
Chen, Haifeng
;
He, Xinjun
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2024/07/12
Hepatocellular carcinoma
Ubiquitin-specific protease 10
Deubiquitination
Selectivity
Zero-Shot Cross-Lingual Document-Level Event Causality Identification with Heterogeneous Graph Contrastive Transfer Learning
会议论文
OAI收割
Torino, Italia, 2024-5
作者:
Zhitao He
;
Pengfei Cao
;
Zhuoran Jin
;
Yubo Chen
;
Kang Liu
  |  
收藏
  |  
浏览/下载:39/0
  |  
提交时间:2024/06/25
LEGO: A Multi-agent Collaborative Framework with Role-playing and Iterative Feedback for Causality Explanation Generation
会议论文
OAI收割
Singapore, 2023-12
作者:
Zhitao He
;
Pengfei Cao
;
Yubo Chen
;
Kang Liu
;
Jun Zhao
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2024/06/25
CogNet2: A Multi-Level Frame Organized Knowledge Base Integrating Linguistic, World and Commonsense Knowledge
会议论文
OAI收割
Athens, Greece, 2023-11
作者:
Wang, Chenhao
;
Guo, Shaoru
;
He, Zhitao
;
Xue, Zhipeng
;
Chen, Yubo
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2024/05/30
Self-Lubricative Organic–Inorganic Hybrid Coating with Anti-Icing and Anti-Waxing Performances by Grafting Liquid-Like Polydimethylsiloxane
期刊论文
OAI收割
Advanced Materials Interfaces, 2022, 卷号: 9, 期号: 18, 页码: 2200160
作者:
Xiaoqing Hao
;
Zhengrong Sun
;
Shuwang Wu
;
Ta-Wei Wang
;
Yubo Liu
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2023/01/09
SARS-CoV-2 envelope protein causes acute respiratory distress syndrome (ARDS)-like pathological damages and constitutes an antiviral target
期刊论文
OAI收割
CELL RESEARCH, 2021, 页码: 14
作者:
Xia, Bingqing
;
Shen, Xurui
;
He, Yang
;
Pan, Xiaoyan
;
Liu, Feng-Liang
  |  
收藏
  |  
浏览/下载:103/0
  |  
提交时间:2021/08/17
Optimization of piperidine constructed peptidyl derivatives as proteasome inhibitors
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2021, 卷号: 29, 页码: 14
作者:
Zhao, Yanmei
;
Xu, Lei
;
Zhang, Jiankang
;
Zhang, Mengmeng
;
Lu, Jingyi
  |  
收藏
  |  
浏览/下载:46/0
  |  
提交时间:2021/05/24
Proteasome inhibitor
Piperidine
Peptidyl
Anti-cancer
SAR
Manipulating the Click Reactivity of Dibenzoazacyclooctynes: From Azide Click Component to Caged Acylation Reagent by Silver Catalysis
期刊论文
OAI收割
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2020, 页码: 6
作者:
Shi, Wei
;
Tang, Feng
;
Ao, Jiwei
;
Yu, Qun
;
Liu, Junjie
  |  
收藏
  |  
浏览/下载:142/0
  |  
提交时间:2020/12/21
acylation
click chemistry
peptides
rearrangements
silver