中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [96]
昆明植物研究所 [27]
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期刊论文 [472]
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浏览/检索结果:
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Oxytocin inhibits the activity of acid-sensing ion channels through the vasopressin-1a receptor in primary sensory neurons1
期刊论文
OAI收割
出版物, 3111, 期号: 0, 页码: 1-34
作者:
Fang Qiu
;
Chun-Yu Qiu
;
Huilan Cai
;
Ting-Ting Liu
;
Zu-Wei Qu
  |  
收藏
  |  
浏览/下载:398/0
  |  
提交时间:2017/07/24
Oxytocin
Acid-sensing Ion Channel
Proton-gated Current
Vasopressin-1a Receptor
Dorsal Root Ganglion Neuron
Electrophysiology
Pain
Synthesis, fluorescence properties of novel thiazolo[3,2-b][1,2,4]triazol derivatives as potent SHP2 inhibitors and its uses in sensing for Fe3+and cell imaging
期刊论文
OAI收割
JOURNAL OF MOLECULAR STRUCTURE, 2025, 卷号: 1324, 页码: 12
作者:
Yan, Xue
;
Zhang, Chun
;
Gao, Li-Xin
;
Cao, Zi-Tong
;
Gan, Su-Ya
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2025/01/14
Thiazolo[3,2-b][1,2,4]triazole
Salicylic acid
Fe3+ion
Fluorescence property
SHP2
Harnessing the Magic Methyl Effect: Discovery of CLPP-2068 as a Novel
Hs
ClpP Activator for the Treatment of Diffuse Large B-Cell Lymphoma
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 4, 页码: 4287-4307
作者:
Sun, Mingyang
;
Chen, Beijing
;
Teng, Dan
;
Zhao, Hongshen
;
Liao, Yilie
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2025/04/01
6
H
-Indolo-[2,3-
b
]-quinoxaline derivatives as promising bifunctional SHP1 inhibitors
期刊论文
OAI收割
ORGANIC & BIOMOLECULAR CHEMISTRY, 2024, 页码: 12
作者:
Zhang, Chun
;
Dong, Yi-Xin
;
Gao, Li-Xin
;
Gan, Suya
;
Gao, Wenran
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2025/02/28
Major specialized natural products from the endangered plant
Heptacodium
miconioides,
, potential medicinal uses and insights into its longstanding unresolved systematic classification
期刊论文
OAI收割
PHYTOCHEMISTRY, 2024, 卷号: 228, 页码: 15
作者:
Zhao, Ze-Yu
;
Wan, Jiang
;
Chen, Hao-Wei
;
Sun, Zhong-Shuai
;
Tao, Yu-Tian
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2024/10/21
Heptacodium miconioides
Caprifoliaceae
Systematic position
Chemotaxonomy
Enantiomeric lignans
Triterpenoids
Quinic acid derivatives
ACL inhibitory
Bis-Iridoid Glycosides and Triterpenoids from
Kolkwitzia amabilis
and Their Potential as Inhibitors of ACC1 and ACL
期刊论文
OAI收割
MOLECULES, 2024, 卷号: 29, 期号: 24, 页码: 18
作者:
Wan, Jiang
;
Zhao, Ze-Yu
;
Wang, Can
;
Jiang, Chun-Xiao
;
Tong, Ying-Peng
  |  
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2025/02/28
Kolkwitzia amabilis
bis-iridoid glycosides
triterpenoids
acetyl CoA carboxylase 1
ATP-citrate lyase
Discovery of CLPP-1071 as an Exceptionally Potent and Orally Efficacious Human ClpP Activator with Strong In Vivo Antitumor Activity
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 21
作者:
Chen, Beijing
;
Sun, Mingyang
;
Zhang, Chun
;
Huang, Qi
;
Teng, Dan
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2024/12/25
Mass balance, metabolism, and pharmacokinetics of [
14
C]amdizalisib, a clinical-stage novel oral selective PI3Kδ inhibitor for the treatment of non-hodgkin's lymphoma, in healthy Chinese volunteers
期刊论文
OAI收割
FRONTIERS IN PHARMACOLOGY, 2024, 卷号: 15, 页码: 13
作者:
Zhao, Chun-Yang
;
Zhang, Li-Jun
;
Sun, Chan
;
Yu, Cheng-Yin
;
Wang, Jian
  |  
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2025/01/06
amdizalisib
PI3K delta kinase
metabolism
mass balance
metabolite identification
pharmacokinetics
safety
Transcriptomic decoding of regional cortical vulnerability to major depressive disorder
期刊论文
OAI收割
COMMUNICATIONS BIOLOGY, 2024, 卷号: 7, 期号: 1, 页码: 12
作者:
Zhu, Jiajia
;
Chen, Xiao
;
Lu, Bin
;
Li, Xue-Ying
;
Wang, Zi-Han
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2024/09/10
Skyway: Accelerate Graph Applications with a Dual-Path Architecture and Fine-Grained Data Management
期刊论文
OAI收割
JOURNAL OF COMPUTER SCIENCE AND TECHNOLOGY, 2024, 卷号: 39, 期号: 4, 页码: 871-894
作者:
Zou, Mo
;
Zhang, Ming-Zhe
;
Wang, Ru-Jia
;
Sun, Xian-He
;
Ye, Xiao-Chun
  |  
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2024/12/06
graph application
computer architecture
memory hierarchy