中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
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昆明植物研究所 [31]
上海药物研究所 [24]
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期刊论文 [297]
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Optimization and Biological Evaluation of Novel 1
H
-Pyrrolo[2,3-
c
]pyridin Derivatives as Potent and Reversible Lysine Specific Demethylase 1 Inhibitors for the Treatment of Acute Myelogenous Leukemia
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 24, 页码: 22080-22103
作者:
Jiang, Hong
;
Li, Cong
;
Li, Na
;
Sheng, Li
;
Wang, Jingkai
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2025/01/14
Global risk dynamics of Borrelia miyamotoi in the context of climate change
期刊论文
OAI收割
ENVIRONMENTAL MICROBIOLOGY, 2024, 卷号: 26, 期号: 10, 页码: e70000
作者:
Tang, Tian
;
Ge, Hong-Han
;
Ma, Tian
;
Hao, Meng-meng
;
Chen, Shuai
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2024/11/19
Global risk dynamics of
Borrelia miyamotoi
in the context of climate change
期刊论文
OAI收割
ENVIRONMENTAL MICROBIOLOGY, 2024, 卷号: 26, 期号: 10, 页码: 14
作者:
Tang, Tian
;
Ge, Hong-Han
;
Ma, Tian
;
Hao, Meng-meng
;
Chen, Shuai
  |  
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2024/12/30
Discovery of Novel Nonpeptidic and Noncovalent Small Molecule 3CL
pro
Inhibitors as anti-SARS-CoV-2 Drug Candidate
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 15, 页码: 12760-12783
作者:
Jiang, Zhidong
;
Feng, Bo
;
Chen, Lu
;
Nie, Tianqing
;
Chen, Shizhao
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2024/09/26
Discovery and characterization of novel potent non-covalent small molecule inhibitors targeting papain-like protease from SARS-CoV-2
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2024, 卷号: 14, 期号: 7, 页码: 3286-3290
作者:
Zheng, Miao
;
Feng, Bo
;
Zhang, Yumin
;
Liu, Xin
;
Zhao, Na
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2024/08/22
Non-covalent PLpro inhibitors
Antiviral activity
Structural-based drug design
Imidazo[4,5-b]pyridine scaffold
A first-in-human phase 1 study of simnotrelvir, a 3CL-like protease inhibitor for treatment of COVID-19, in healthy adult subjects
期刊论文
OAI收割
EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES, 2023, 卷号: 191, 页码: 9
作者:
Yang, Xin-Mei
;
Yang, Yang
;
Yao, Bu-Fan
;
Ye, Pan-Pan
;
Xu, Yan
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2023/12/11
COVID-19
Simnotrelvir
Safety
Pharmacokinetics
Healthy subjects
Enhancement of in-plane thermal conductivity of flexible boron nitride heat spreaders by micro/nanovoid filling using deformable liquid metal nanoparticles
期刊论文
OAI收割
RARE METALS, 2023, 页码: 11
作者:
Tao, Pei-Di
;
Wang, Shao-Gang
;
Chen, Lu
;
Ying, Jun-Feng
;
Lv, Le
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2024/01/08
Boron nitride nanosheet
Liquid metal
Eutectic gallium-indium
In-plane thermal conductivity
Heat spreader
Comparative Characterization of the Ginsenosides from Six Panax Herbal Extracts and Their In Vitro Rat Gut Microbial Metabolites by Advanced Liquid Chromatography-Mass Spectrometry Approaches
期刊论文
OAI收割
JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY, 2023, 卷号: 71, 期号: 24, 页码: 9391-9403
作者:
Mi, Yue-Guang
;
Xu, Xiao-Yan
;
Hong, Li-Li
;
Jiang, Mei-Ting
;
Chen, Bo-Xue
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2023/10/17
Panax
multicomponent characterization
quantitative assay
gut microbiota
in vitro biotransformation
liquid chromatography-massspectrometry
Discovery of novel non-peptidic and non-covalent small-molecule 3CL(pro) inhibitors as potential candidate for COVID-19 treatment
期刊论文
OAI收割
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2023, 卷号: 8, 期号: 1, 页码: 4
作者:
Jiang, Zhidong
;
Feng, Bo
;
Zhang, Yumin
;
Nie, Tianqing
;
Liu, Hong
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2023/10/17
Distribution patterns of landslides triggered by the 2022 Ms 6.8 Luding earthquake, Sichuan, China
期刊论文
OAI收割
JOURNAL OF MOUNTAIN SCIENCE, 2023, 卷号: N/A
作者:
Zhang, Jian-qiang
;
Yang, Zong-ji
;
Meng, Qing-kai
;
Wang, Jiao
;
Hu, Kai-heng
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2024/01/04
2022 Luding earthquake
Earthquake-triggered landslide
Landslide inventory
Distribution patterns