中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
广州生物医药与健康... [11]
上海药物研究所 [1]
采集方式
OAI收割 [12]
内容类型
期刊论文 [12]
发表日期
2019 [1]
2016 [7]
2014 [2]
2013 [2]
学科主题
Pharmacolo... [8]
Chemistry [2]
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Effective Virtual Screening Strategy toward heme-containing proteins: Identification of novel IDO1 inhibitors
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 184, 页码: 23
作者:
Zou, Yi
;
Hu, Yue
;
Ge, Shushan
;
Zheng, Yingbo
;
Li, Yuezhen
  |  
收藏
  |  
浏览/下载:36/0
  |  
提交时间:2020/07/01
IDO1
Heme
T cell
Cancer immunotherapy
Virtual screening
Drug design
Molecular dynamics simulation
Discovery of New Monocarbonyl Ligustrazine-Curcumin Hybrids for Intervention of Drug-Sensitive and Drug-Resistant Lung Cancer
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 5, 页码: 1747-1760
Ai, Yong
;
Zhu, Bin
;
Ren, Caiping
;
Kang, Fenghua
;
Lo, Jinlong
;
Huang, Zhangjian
;
Lai, Yisheng
;
Peng, Sixun
;
Ding, Ke
;
Tian, Jide
;
Zhang, Yihua
收藏
  |  
浏览/下载:46/0
  |  
提交时间:2016/12/16
Discovery of New Monocarbonyl Ligustrazine-Curcumin Hybrids for Intervention of Drug-Sensitive and Drug-Resistant Lung Cancer
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 5, 页码: 1747-1760
作者:
Lai, Yisheng
;
Peng, Sixun
;
Ding, Ke
;
Tian, Jide
;
Zhang, Yihua
  |  
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2018/12/13
Structure-based discovery of novel 4,5,6-trisubstituted pyrimidines as potent covalent Bruton's tyrosine kinase inhibitors
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2016, 卷号: 26, 期号: 13, 页码: 3052-3059
作者:
Zhang, Yihua
;
Lai, Yisheng
;
Zou, Yi
;
Xiao, Jianhu
;
Tu, Zhengchao
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2018/12/13
Structure-based discovery of novel 4,5,6-trisubstituted pyrimidines as potent covalent Bruton's tyrosine kinase inhibitors
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2016, 卷号: 26, 期号: 13, 页码: 3052-3059
作者:
Luo, Minghao
;
Lai, Yisheng
;
Zhang, Yihua
;
Ding, Ke
;
Zou, Yi
  |  
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2018/12/21
Structure-based discovery of novel 4,5,6-trisubstituted pyrimidines as potent covalent Bruton's tyrosine kinase inhibitors
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2016, 卷号: 26, 期号: 13, 页码: 3052-3059
作者:
Zou, Yi
;
Xiao, Jianhu
;
Tu, Zhengchao
;
Yao, Kun
;
Lai, Yisheng
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2018/12/13
Structure-based discovery of novel 4,5,6-trisubstituted pyrimidines as potent covalent Bruton's tyrosine kinase inhibitors
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2016, 卷号: 26, 期号: 13, 页码: 3052-3059
Zou, Yi
;
Xiao, Jianhu
;
Tu, Zhengchao
;
Zhang, Yingyi
;
Yao, Kun
;
Luo, Minghao
;
Ding, Ke
;
Zhang, Yihua
;
Lai, Yisheng
收藏
  |  
浏览/下载:38/0
  |  
提交时间:2016/12/16
Structure-based discovery of novel 4,5,6-trisubstituted pyrimidines as potent covalent Bruton's tyrosine kinase inhibitors
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2016, 卷号: 26, 期号: 13, 页码: 3052-3059
作者:
Xiao, Jianhu
;
Zou, Yi
;
Tu, Zhengchao
;
Zhang, Yingyi
;
Yao, Kun
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2018/12/13
Synthesis and evaluation of 2-anilinopyrimidines bearing 3-aminopropamides as potential epidermal growth factor receptor inhibitors
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2014, 卷号: 77, 页码: 75-83
作者:
Peng, Sixun
;
Zhang, Yihua
;
Lai, Yisheng
;
Huang, Zhangjian
;
Ding, Ke
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2018/12/13
Synthesis and evaluation of 2-anilinopyrimidines bearing 3-aminopropamides as potential epidermal growth factor receptor inhibitors
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2014, 卷号: 77, 页码: 75-83
Han, Chun
;
Wan, Ledong
;
Ji, Hongbin
;
Ding, Ke
;
Huang, Zhangjian
;
Lai, Yisheng
;
Peng, Sixun
;
Zhang, Yihua
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2016/12/16