中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共10条,第1-10条 帮助

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PROTAC derivatization of natural products for target identification and drug discovery: Design of evodiamine-based PROTACs as novel REXO4 degraders 期刊论文  OAI收割
JOURNAL OF ADVANCED RESEARCH, 2024, 卷号: 63, 页码: 219-230
作者:  
Chen, Shuqiang;  Bi, Kaijian;  Liang, Huixin;  Wu, Zhe;  Huang, Min
  |  收藏  |  浏览/下载:15/0  |  提交时间:2024/10/21
Discovery of Dual Function Agents That Exhibit Anticancer Activity via Catastrophic Nicotinamide Adenine Dinucleotide Depletion 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 24, 页码: 16694-16703
作者:  
Fu, Yixian;  Huang, Yahui;  Zhou, Chenchen;  Li, Xinge;  Dong, Guoqiang
  |  收藏  |  浏览/下载:18/0  |  提交时间:2024/01/26
Stimuli-activatable PROTACs for precise protein degradation and cancer therapy 期刊论文  OAI收割
SCIENCE BULLETIN, 2023, 卷号: 68, 期号: 10, 页码: 1069-1085
作者:  
Gao, Jing;  Yang, Lei;  Lei, Shumin;  Zhou, Feng;  Nie, Huijun
  |  收藏  |  浏览/下载:21/0  |  提交时间:2023/10/17
Discovery of Highly Potent Nicotinamide Phosphoribosyltransferase Degraders for Efficient Treatment of Ovarian Cancer 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 页码: 15
作者:  
Bi, Kaijian;  Cheng, Junfei;  He, Shipeng;  Fang, Yuxin;  Huang, Min
  |  收藏  |  浏览/下载:26/0  |  提交时间:2023/04/10
Making Protein Degradation Visible: Discovery of Theranostic PROTACs for Detecting and Degrading NAMPT 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 页码: 13
作者:  
Cheng, Junfei;  He, Shipeng;  Xu, Jun;  Huang, Min;  Dong, Guoqiang
  |  收藏  |  浏览/下载:16/0  |  提交时间:2023/04/10
NAMPT-targeting PROTAC promotes antitumor immunity via suppressing myeloid-derived suppressor cell expansion 期刊论文  OAI收割
ACTA PHARMACEUTICA SINICA B, 2022, 卷号: 12, 期号: 6, 页码: 2859-2868
作者:  
Wu, Ying;  Pu, Congying;  Fu, Yixian;  Dong, Guoqiang;  Huang, Min
  |  收藏  |  浏览/下载:10/0  |  提交时间:2024/03/21
Evodiamine-Inspired Topoisomerase-Histone Deacetylase Dual Inhibitors: Novel Orally Active Antitumor Agents for Leukemia Therapy br 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 6, 页码: 4818-4831
作者:  
Wu, Shanchao;  Huang, Yahui;  Wang, Ting;  Li, Keliang;  Lu, Junjie
  |  收藏  |  浏览/下载:57/0  |  提交时间:2022/08/16
Discovery of Potent Benzofuran-Derived Diapophytoene Desaturase (CrtN) Inhibitors with Enhanced Oral Bioavailability for the Treatment of Methicillin-Resistant Staphylococcus aureus (MRSA) Infections 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 7, 页码: 3215-3230
作者:  
Wang, Youxin;  Chen, Feifei;  Di, Hongxia;  Xu, Yong;  Xiao, Qiang
  |  收藏  |  浏览/下载:15/0  |  提交时间:2019/01/08
ψ-Bufarenogin, a novel anti-tumor compound, suppresses liver cancer growth by inhibiting receptor tyrosine kinase-mediated signaling 期刊论文  OAI收割
Oncotarget, 2015, 卷号: 6, 期号: 13, 页码: 11627
作者:  
Jin Ding;  Wen Wen;  Daimin Xiang;  Peipei Yin;  Liu YF(刘艳芳)
收藏  |  浏览/下载:21/0  |  提交时间:2016/11/24
psi-Bufarenogin, a novel anti-tumor compound, suppresses liver cancer growth by inhibiting receptor tyrosine kinase-mediated signaling 期刊论文  OAI收割
oncotarget, 2015, 卷号: 6, 期号: 13, 页码: 11627-11639
作者:  
Ding, Jin;  Wen, Wen;  Xiang, Daimin;  Yin, Peipei;  Liu, Yanfang
收藏  |  浏览/下载:59/0  |  提交时间:2015/11/17