中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [8]
大连化学物理研究所 [2]
采集方式
OAI收割 [10]
内容类型
期刊论文 [10]
发表日期
2024 [1]
2023 [2]
2022 [4]
2016 [1]
2015 [2]
学科主题
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PROTAC derivatization of natural products for target identification and drug discovery: Design of evodiamine-based PROTACs as novel REXO4 degraders
期刊论文
OAI收割
JOURNAL OF ADVANCED RESEARCH, 2024, 卷号: 63, 页码: 219-230
作者:
Chen, Shuqiang
;
Bi, Kaijian
;
Liang, Huixin
;
Wu, Zhe
;
Huang, Min
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2024/10/21
PROTAC
Natural products
Target identification
Quantitative proteomics
Antitumor activities
Discovery of Dual Function Agents That Exhibit Anticancer Activity via Catastrophic Nicotinamide Adenine Dinucleotide Depletion
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 24, 页码: 16694-16703
作者:
Fu, Yixian
;
Huang, Yahui
;
Zhou, Chenchen
;
Li, Xinge
;
Dong, Guoqiang
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2024/01/26
Stimuli-activatable PROTACs for precise protein degradation and cancer therapy
期刊论文
OAI收割
SCIENCE BULLETIN, 2023, 卷号: 68, 期号: 10, 页码: 1069-1085
作者:
Gao, Jing
;
Yang, Lei
;
Lei, Shumin
;
Zhou, Feng
;
Nie, Huijun
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2023/10/17
PROTAC
Stimuli-activatable prodrug
Precise protein degradation
Nanomedicine
Combinatory therapy
Discovery of Highly Potent Nicotinamide Phosphoribosyltransferase Degraders for Efficient Treatment of Ovarian Cancer
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 页码: 15
作者:
Bi, Kaijian
;
Cheng, Junfei
;
He, Shipeng
;
Fang, Yuxin
;
Huang, Min
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2023/04/10
Making Protein Degradation Visible: Discovery of Theranostic PROTACs for Detecting and Degrading NAMPT
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 页码: 13
作者:
Cheng, Junfei
;
He, Shipeng
;
Xu, Jun
;
Huang, Min
;
Dong, Guoqiang
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2023/04/10
NAMPT-targeting PROTAC promotes antitumor immunity via suppressing myeloid-derived suppressor cell expansion
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2022, 卷号: 12, 期号: 6, 页码: 2859-2868
作者:
Wu, Ying
;
Pu, Congying
;
Fu, Yixian
;
Dong, Guoqiang
;
Huang, Min
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2024/03/21
NAMPT
Non-enzymatic function
eNAMPT
Cancer
MDSC
PROTAC
Tumor immunity
Immunotherapy
Evodiamine-Inspired Topoisomerase-Histone Deacetylase Dual Inhibitors: Novel Orally Active Antitumor Agents for Leukemia Therapy br
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 6, 页码: 4818-4831
作者:
Wu, Shanchao
;
Huang, Yahui
;
Wang, Ting
;
Li, Keliang
;
Lu, Junjie
  |  
收藏
  |  
浏览/下载:57/0
  |  
提交时间:2022/08/16
Discovery of Potent Benzofuran-Derived Diapophytoene Desaturase (CrtN) Inhibitors with Enhanced Oral Bioavailability for the Treatment of Methicillin-Resistant Staphylococcus aureus (MRSA) Infections
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 7, 页码: 3215-3230
作者:
Wang, Youxin
;
Chen, Feifei
;
Di, Hongxia
;
Xu, Yong
;
Xiao, Qiang
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2019/01/08
ψ-Bufarenogin, a novel anti-tumor compound, suppresses liver cancer growth by inhibiting receptor tyrosine kinase-mediated signaling
期刊论文
OAI收割
Oncotarget, 2015, 卷号: 6, 期号: 13, 页码: 11627
作者:
Jin Ding
;
Wen Wen
;
Daimin Xiang
;
Peipei Yin
;
Liu YF(刘艳芳)
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2016/11/24
psi-Bufarenogin, a novel anti-tumor compound, suppresses liver cancer growth by inhibiting receptor tyrosine kinase-mediated signaling
期刊论文
OAI收割
oncotarget, 2015, 卷号: 6, 期号: 13, 页码: 11627-11639
作者:
Ding, Jin
;
Wen, Wen
;
Xiang, Daimin
;
Yin, Peipei
;
Liu, Yanfang
收藏
  |  
浏览/下载:59/0
  |  
提交时间:2015/11/17
psi-Bufarenogin
hepatocellular carcinoma
epithelial growth factor receptor
hepatocyte growth factor receptor