中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [51]
上海硅酸盐研究所 [24]
地理科学与资源研究... [17]
合肥物质科学研究院 [5]
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期刊论文 [122]
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2025 [2]
2024 [6]
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2022 [9]
2021 [18]
2020 [2]
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Optics [4]
光学材料;晶体 [3]
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A natural small molecule isoginkgetin alleviates hypercholesterolemia and atherosclerosis by targeting ACLY
期刊论文
OAI收割
THERANOSTICS, 2025, 卷号: 15, 期号: 10, 页码: 4325-4344
作者:
Zhang, Zhidan
;
Chen, Meijie
;
Xu, Yitong
;
Wang, Zhihua
;
Liu, Zhenghong
  |  
收藏
  |  
浏览/下载:0/0
  |  
提交时间:2025/06/23
Atherosclerosis
Hyperlipidemia
ATP-Citrate lyase (ACLY)
lipid metabolism
Isoginkgetin
A Phase I Study to Evaluate the Safety, Tolerability, Pharmacokinetics of BGT-002, a Novel ATP-Citrate Lyase Inhibitor, in Healthy Chinese Subjects
期刊论文
OAI收割
DRUG DESIGN DEVELOPMENT AND THERAPY, 2025, 卷号: 19, 页码: 1783-1794
作者:
Liu, Yun
;
Yu, Chengyin
;
Zhang, Yifan
;
Xie, Zhifu
;
Wang, Yating
  |  
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2025/04/24
safety
tolerability
pharmacokinetics
pharmacodynamics
BGT-002
novel ACLY inhibitor
Discovery of a Potent, selective and orally bioavailable CDK9 degrader for targeting transcription regulation in Triple-Negative breast cancer
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2024, 卷号: 153, 页码: 16
作者:
Nie, Hui-Jun
;
Li, Ben-Fu
;
Sun, Jingya
;
Yuan, Yali
;
Zhang, Zhi-Gao
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2024/11/26
Triple-negative breast cancer
Targeting transcription regulation
Orally bioavailable degrader
PROTAC
Cyclin-dependent Kinase 9
Discovery of Alkyl Conjugated Diene Diacids as Novel ACLY Inhibitors
期刊论文
OAI收割
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2024, 卷号: 44, 期号: 11, 页码: 3476-3489
作者:
Cheng, Tingting
;
Song, Gaolei
;
Cheng, Long
;
Wang, Fan
;
Sun, Xinyu
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2025/02/28
metabolic diseases
ATP-citrate lyase (ACLY)
lipogenesis
ACLY inhibitors
dienyldicarboxylic acid
Discovery of Orally Bioavailable and Potent CDK9 Inhibitors for Targeting Transcription Regulation in Triple-Negative Breast Cancer
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 12, 页码: 10035-10056
作者:
Wang, Wen-Jing
;
Gao, Lixin
;
Wang, Simei
;
Huang, Wensi
;
Meng, Xin-Yu
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2024/08/20
Comparison of three source apportionment methods based on observed and initial HCHO in Taiyuan, China
期刊论文
OAI收割
SCIENCE OF THE TOTAL ENVIRONMENT, 2024, 卷号: 926, 页码: 12
作者:
Cui, Yang
;
Hua, Jingya
;
He, Qiusheng
;
Guo, Lili
;
Wang, Yonghong
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2024/09/13
Formaldehyde
Photochemical losses
Multiple linear regression
Photochemical age -based parameterization method
PMF model
DRAK2 suppresses autophagy by phosphorylating ULK1 at Ser
56
to diminish pancreatic β cell function upon overnutrition
期刊论文
OAI收割
SCIENCE TRANSLATIONAL MEDICINE, 2024, 卷号: 16, 期号: 733, 页码: 16
作者:
Lu, Yuting
;
Xu, Junyu
;
Li, Yufeng
;
Wang, Ruoran
;
Dai, Chengqiu
  |  
收藏
  |  
浏览/下载:43/0
  |  
提交时间:2024/03/13
Increased frequency of extreme climatic events weakens the community stability of natural grassland under directional climate changes by reducing resilience
期刊论文
OAI收割
GLOBAL ECOLOGY AND BIOGEOGRAPHY, 2024, 卷号: 33, 期号: 6
作者:
Liu, Peipei
;
Lv, Wangwang
;
Sun, Jianping
;
Piao, Shilong
;
Wang, Yanfen
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2024/11/27
Glutamine Production by Glul Promotes Thermogenic Adipocyte Differentiation Through Prdm9-Mediated H3K4me3 and Transcriptional Reprogramming
期刊论文
OAI收割
DIABETES, 2023, 卷号: 72, 期号: 11, 页码: 24
作者:
  |  
收藏
  |  
浏览/下载:34/0
  |  
提交时间:2024/03/25
Changes in Dissolved Inorganic Carbon Across Yangtze River Regulated by Dam and River-Lake Exchange
期刊论文
OAI收割
GLOBAL BIOGEOCHEMICAL CYCLES, 2023, 卷号: 37, 期号: 9, 页码: 19
作者:
Zhao, Chu
;
Wang, Chuan
;
Li, Jianhong
;
Meng, Lize
;
Xue, Jingya
  |  
收藏
  |  
浏览/下载:36/0
  |  
提交时间:2023/10/30
dissolved inorganic carbon
stable isotope
hydrological recharge
Three Gorges Dam
Yangtze River