中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共49条,第1-10条 帮助

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Design, Synthesis, and Biological Evaluation of Novel Diaminopyrimidine Macrocycles as Fourth Generation Reversible EGFR Inhibitors That Overcome Clinical Resistance to Osimertinib Mediated by C797S Mutation 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 22, 页码: 20531-20558
作者:  
Hu, Shiliang;  Tong, Linjiang;  Qin, Qiao;  Wen, Jiaxin;  Li, Yan
  |  收藏  |  浏览/下载:8/0  |  提交时间:2024/12/11
Branched-chain amino acid transaminase 1 confers EGFR-TKI resistance through epigenetic glycolytic activation 期刊论文  OAI收割
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2024, 卷号: 9, 期号: 1, 页码: 17
作者:  
Zhang, Tao;  Pan, Zilu;  Gao, Jing;  Wu, Qingqing;  Bai, Gang
  |  收藏  |  浏览/下载:16/0  |  提交时间:2024/10/21
Comprehensive Attribute Prediction Learning for Person Search by Language 期刊论文  OAI收割
IEEE TRANSACTIONS ON IMAGE PROCESSING, 2024, 卷号: 33, 页码: 1990-2003
作者:  
Niu, Kai;  Huang, Linjiang;  Long, Yuzhou;  Huang, Yan;  Wang, Liang
  |  收藏  |  浏览/下载:19/0  |  提交时间:2024/07/03
Preclinical and early clinical studies of a novel compound SYHA1813 that efficiently crosses the blood-brain barrier and exhibits potent activity against glioblastoma 期刊论文  OAI收割
ACTA PHARMACEUTICA SINICA B, 2023, 卷号: 13, 期号: 12, 页码: 4748-4764
作者:  
  |  收藏  |  浏览/下载:24/0  |  提交时间:2024/01/26
Improving Inconspicuous Attributes Modeling for Person Search by Language 期刊论文  OAI收割
IEEE TRANSACTIONS ON IMAGE PROCESSING, 2023, 卷号: 32, 页码: 3429-3441
作者:  
Niu, Kai;  Huang, Tao;  Huang, Linjiang;  Wang, Liang
  |  收藏  |  浏览/下载:6/0  |  提交时间:2023/11/17
Novel Sphingosine Kinase 1 Inhibitor Suppresses Growth of Solid Tumor and Inhibits the Lung Metastasis of Triple-Negative Breast Cancer 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 11, 页码: 7697-7716
作者:  
Zhang, Shurui;  Chen, Xiaoxu;  Wu, Chenglin;  Xu, Hui;  Xie, Xiong
  |  收藏  |  浏览/下载:36/0  |  提交时间:2022/08/16
SLC1A1-mediated cellular and mitochondrial influx of R-2-hydroxyglutarate in vascular endothelial cells promotes tumor angiogenesis in IDH1-mutant solid tumors 期刊论文  OAI收割
CELL RESEARCH, 2022, 页码: 21
作者:  
Wang, Xiaomin;  Chen, Ziqi;  Xu, Jun;  Tang, Shuai;  An, Nan
  |  收藏  |  浏览/下载:61/0  |  提交时间:2022/06/15
Discovery of N-(3-bromo-1H-indol-5-yl)-quinazolin-4-amine as an effective molecular skeleton to develop reversible/irreversible pan-HER inhibitors 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 233, 页码: 13
作者:  
Tang, Qidong;  Peng, Ting;  Hu, Jie;  Zhang, Tao;  Chen, Pengqin
  |  收藏  |  浏览/下载:45/0  |  提交时间:2022/08/16
Multi-Modality Self-Distillation for Weakly Supervised Temporal Action Localization 期刊论文  OAI收割
IEEE TRANSACTIONS ON IMAGE PROCESSING, 2022, 卷号: 31, 页码: 1504-1519
作者:  
Huang, Linjiang;  Wang, Liang;  Li, Hongsheng
  |  收藏  |  浏览/下载:32/0  |  提交时间:2022/03/17
LS-106, a novel EGFR inhibitor targeting C797S, exhibits antitumor activities both in vitro and in vivo 期刊论文  OAI收割
CANCER SCIENCE, 2021, 页码: 12
作者:  
Liu, Yingqiang;  Lai, Mengzhen;  Li, Shan;  Wang, Yanan;  Feng, Fang
  |  收藏  |  浏览/下载:110/0  |  提交时间:2022/01/18