中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共57条,第1-10条 帮助

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Discovery of pyrrolo[2,3-d]pyrimidine derivatives as novel FLT3/ IRAK4 inhibitors 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 296, 页码: 23
作者:  
Yuan, Haibin;  Gao, Yue;  Wang, Peipei;  Dong, Xiaowu;  Li, Jia
  |  收藏  |  浏览/下载:1/0  |  提交时间:2025/08/20
Design, synthesis, and evaluation of Menin-targeting compounds for the treatment of acute Myelocytic leukemia (AML) 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 296, 页码: 17
作者:  
Mo, Jun;  Wang, Yuxian;  Pan, Youlu;  Xiao, Qitao;  Zhao, Jinyi
  |  收藏  |  浏览/下载:4/0  |  提交时间:2025/08/20
Proteogenomic characterization of non-functional clinically relevant subgroups 期刊论文  OAI收割
CANCER CELL, 2025, 卷号: 43, 期号: 4, 页码: 36
作者:  
Ji, Shunrong;  Cao, Lihua;  Gao, Jing;  Du, Yang;  Ye, Zeng
  |  收藏  |  浏览/下载:29/0  |  提交时间:2025/06/23
Auto-RapTAC: A Versatile and Sustainable Platform for the Automated Rapid Synthesis and Evaluation of PROTAC 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 页码: 15
作者:  
Chen, Jiexuan;  Wu, Mingfei;  Mo, Jun;  Hong, Ju;  Wang, Wei
  |  收藏  |  浏览/下载:31/0  |  提交时间:2025/04/01
Discovery of N-Benzylpiperidinol derivatives as USP7 inhibitors against Hematology 期刊论文  OAI收割
BIOORGANIC CHEMISTRY, 2024, 卷号: 153, 页码: 13
作者:  
Pan, Youlu;  Chen, Haifeng;  Fu, Jingfeng;  Zhang, Jingyu;  Wang, Peipei
  |  收藏  |  浏览/下载:40/0  |  提交时间:2024/10/21
Single-cell sequencing reveals the heterogeneity of pancreatic neuroendocrine tumors under genomic instability and histological grading 期刊论文  OAI收割
ISCIENCE, 2024, 卷号: 27, 期号: 9, 页码: 18
作者:  
Ye, Zeng;  Zhou, Yan;  Hu, Yuheng;  Li, Qiang;  Xu, Zijin
  |  收藏  |  浏览/下载:31/0  |  提交时间:2024/11/05
Discovery of a Highly Potent and Selective BRD9 PROTAC Degrader Based on E3 Binder Investigation for the Treatment of Hematological Tumors 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 28
作者:  
Duan, Haiting;  Zhang, Jingyu;  Gui, Renzhao;  Lu, Yang;  Pang, Ao
  |  收藏  |  浏览/下载:32/0  |  提交时间:2024/08/20
Discovery of potent small molecule ubiquitin-specific protease 10 inhibitors with anti-hepatocellular carcinoma activity through regulating YAP expression 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 272, 页码: 21
作者:  
Lu, Yang;  Gao, Jian;  Wang, Peipei;  Chen, Haifeng;  He, Xinjun
  |  收藏  |  浏览/下载:25/0  |  提交时间:2024/07/12
Structure-based identification of new orally bioavailable BRD9-PROTACs for treating acute myelocytic leukemia 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 262, 页码: 18
作者:  
Zhang, Jingyu;  Duan, Haiting;  Gui, Renzhao;  Wu, Mingfei;  Shen, Liteng
  |  收藏  |  浏览/下载:168/0  |  提交时间:2023/12/19
Effects of quenching temperature on the microstructure and impact toughness of 50CrMnSiVNb spring steel 期刊论文  OAI收割
MATERIALS SCIENCE AND ENGINEERING A-STRUCTURAL MATERIALS PROPERTIES MICROSTRUCTURE AND PROCESSING, 2023, 卷号: 870, 页码: 14
作者:  
Xia, Bo;  Zhang, Peng;  Wang, Bin;  Li, Xiaowu;  Zhang, Zhefeng
  |  收藏  |  浏览/下载:15/0  |  提交时间:2024/01/07