中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [17]
金属研究所 [12]
西安光学精密机械研究... [8]
广州地球化学研究所 [7]
地理科学与资源研究所 [5]
烟台海岸带研究所 [4]
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OAI收割 [62]
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期刊论文 [60]
会议论文 [2]
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2024 [2]
2023 [4]
2022 [3]
2021 [5]
2020 [13]
2019 [3]
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Chemistry [2]
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Discovery of Alkyl Conjugated Diene Diacids as Novel ACLY Inhibitors
期刊论文
OAI收割
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2024, 卷号: 44, 期号: 11, 页码: 3476-3489
作者:
Cheng, Tingting
;
Song, Gaolei
;
Cheng, Long
;
Wang, Fan
;
Sun, Xinyu
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2025/02/28
metabolic diseases
ATP-citrate lyase (ACLY)
lipogenesis
ACLY inhibitors
dienyldicarboxylic acid
Simultaneous determination of BGT-002 and its acyl glucuronide metabolite ZM326E-M2 in human plasma by liquid chromatography-tandem mass spectrometry and its application to a pharmacokinetic study
期刊论文
OAI收割
JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS, 2024, 卷号: 243, 页码: 8
作者:
Zhu, Xueran
;
Cui, Shumin
;
Liu, Xinjing
;
Zhang, Mei
;
Xie, Zhifu
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2024/05/31
ATP-Citrate Lyase
BGT-002
Acyl glucuronide metabolite
Pseudo-MRM
LC-MS/MS
Pharmacokinetics
Fast Adiabatic Mode Evolution Assisted 2 x 2 Broadband 3 dB Coupler Using Silicon-on-Insulator Fishbone-like Grating Waveguides
期刊论文
OAI收割
NANOMATERIALS, 2023, 卷号: 13, 期号: 20
作者:
Xue, Yulong
;
Zhang, Lingxuan
;
Ren, Yangming
;
Lei, Yufang
;
Sun, Xiaochen
  |  
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2023/11/20
fast adiabatic
broadband coupler
grating waveguides
power splitter
local eigenmodes
Suppressing grating lobes of large-aperture optical phased array with circular array design
期刊论文
OAI收割
APPLIED OPTICS, 2023, 卷号: 62, 期号: 15, 页码: 4110-4114
作者:
Lei, Yufang
;
Zhang, Lingxuan
;
Xue, Yulong
;
Ren, Yangming
;
Zhang, Qihao
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2023/08/28
Si Photonics FMCW LiDAR Chip with Solid-State Beam Steering by Interleaved Coaxial Optical Phased Array
期刊论文
OAI收割
MICROMACHINES, 2023, 卷号: 14, 期号: 5
作者:
Lei, Yufang
;
Zhang, Lingxuan
;
Yu, Zhiyuan
;
Xue, Yulong
;
Ren, Yangming
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2023/07/03
LiDAR
optical phased array
integrated optics
Development of the novel ACLY inhibitor 326E as a promising treatment for hypercholesterolemia
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2023, 卷号: 13, 期号: 2, 页码: 739-753
作者:
Xie, Zhifu
;
Zhang, Mei
;
Song, Qian
;
Cheng, Long
;
Zhang, Xinwen
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2024/03/27
Hypercholesterolemia
Atherosclerosis
Liver
ATP-Citrate lyase (ACLY)
Lipogenesis
Cholesterol efflux
ACLY inhibitor
Two-dimensional single-lobe Si photonic optical phased array with minimal antennas using a non-uniform large spacing array design
期刊论文
OAI收割
APPLIED OPTICS, 2022, 卷号: 61, 期号: 24, 页码: 7158-7162
作者:
Xue, Yulong
;
Zhang, Qihao
;
Ren, Yangming
;
Lei, Yufang
;
Sun, Xiaochen
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2022/09/29
The HDAC inhibitor GCJ-490A suppresses c-Met expression through IKK? and overcomes gefitinib resistance in non-small cell lung cancer
期刊论文
OAI收割
CANCER BIOLOGY & MEDICINE, 2022, 卷号: 19, 期号: 8, 页码: 1172-1192
作者:
He, Ting
;
Gao, Yinglei
;
Fang, Yanfen
;
Zhang, Yangming
;
Zhang, Shuwei
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2024/03/21
HDAC inhibitor
c-Met
IKK?
NSCLC
gefitinib
Dephosphorylation of AMP-activated protein kinase exacerbates ischemia/reperfusion-induced acute kidney injury via mitochondrial dysfunction
期刊论文
OAI收割
KIDNEY INTERNATIONAL, 2022, 卷号: 101, 期号: 2, 页码: 315-330
作者:
Ma, Haijian
;
Guo, Xiaozhen
;
Cui, Shichao
;
Wu, Yongmei
;
Zhang, Yangming
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2024/03/21
acute kidney injury
AMPK
autophagy
lipid metabolism
Optimization and Development of a Scalable Palladium-Catalyzed C-H Activation Process for the Geometry-Selective Preparation of Kilograms of YLF466D, a Potent AMP-Activated Protein Kinase Activator
期刊论文
OAI收割
ORGANIC PROCESS RESEARCH & DEVELOPMENT, 2021, 卷号: 25, 期号: 10, 页码: 2260-2269
作者:
Yin, Jianpeng
;
Zhan, Desheng
;
Ma, Hui
;
Liu, Huanan
;
Yu, Lifang
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2021/12/16
YLF466D
AMPK activator
glucose metabolism
lipid metabolism
MIRI
domino reaction
C-H activation