中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共40条,第1-10条 帮助

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Multiplexed Isotope-Coded Mass Spectrometry Footprinting Enables Broad Heteroatom-Residue Mapping and Uncovers Noncanonical Ligand-Binding Sites in Amyloidosis Proteins 期刊论文  OAI收割
ANALYTICAL CHEMISTRY, 2026, 页码: 13
作者:  
Yang, Kuoqi;  Zheng, Wei;  Bai, Lin;  Wang, Kai;  Zhang, Jian
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Design, synthesis, and biological evaluation of KDM5B degraders against hematologic malignancy cells 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 296, 页码: 17
作者:  
Liu, Xiaowen;  Li, Jiarong;  Guo, Yihao;  Xie, Zhicheng;  Geng, Meiyu
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Fine structural design of 3βHSD1 inhibitors for prostate cancer 期刊论文  OAI收割
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2025, 卷号: 122, 期号: 26, 页码: 12
作者:  
He, Dongyin;  Zhang, Luyao;  Yu, Leiye;  Zhang, Yuhang;  Chen, Jingjing
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Novel Aryl Sulfonium Modification on Vancomycin to Tackle MRSA and VRE In Vitro and In Vivo through Dual Enhanced Cell-Wall and Membrane Inhibition 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 8, 页码: 8310-8329
作者:  
Xie, Yuanyuan;  Wang, Xiaowen;  Chang, Taopeng;  Chen, Zhifu;  Luo, Youhong
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Discovery of 2,4-quinazolinedione derivatives as LC3B recruiters in the facilitation of protein complex degradations 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 287, 页码: 10
作者:  
Zeng, Yanping;  Xiao, Jian;  Shi, Li;  Li, Yangsha;  Xu, Yuanxin
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Single Amine or Guanidine Modification on Norvancomycin and Vancomycin to Overcome Multidrug-Resistance through Augmented Lipid II Binding and Increased Membrane Activity 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 22, 页码: 20639-20663
作者:  
Bian, Xiaolei;  Chen, Zhifu;  Li, Fang;  Xie, Yuanyuan;  Li, Yi
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Structural Optimization of Isoquinoline Derivatives from Lycobetaine and Their Inhibitory Activity against Neuroendocrine Prostate Cancer Cells 期刊论文  OAI收割
MOLECULES, 2024, 卷号: 29, 期号: 18, 页码: 28
作者:  
Zhang, Zhuo;  Shen, Qianqian;  Ji, Yiyi;  Ma, Yanjie;  Hou, Haiyang
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A novel BODIPY-based theranostic agent for in vivo fluorescence imaging of cerebral Aβ and ameliorating Aβ-associated disorders in Alzheimer's disease transgenic mice 期刊论文  OAI收割
RSC MEDICINAL CHEMISTRY, 2024, 页码: 9
作者:  
Zhang, Jingjing;  Ren, Wenming;  Liu, Xiaohui;  Chen, Jingjing;  Zeng, Yuteng
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Crop/Plant Modeling Supports Plant Breeding II. Guidance of Functional Plant Phenotyping for Trait Discovery 期刊论文  OAI收割
PLANT PHENOMICS, 2023, 卷号: 5, 页码: 19
作者:  
Zhang, Pengpeng;  Huang, Jingyao;  Ma, Yuntao;  Wang, Xiujuan;  Kang, Mengzhen
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Discovery of (S)-N-(2-Amino-4-fluorophenyl)-4-(1-(3-(4-((dimethylamino)methyl)phenyl)-6-oxopyridazin-1(6H)-yl)ethyl)benzamide as Potent Class I Selective HDAC Inhibitor for Oral Anticancer Drug Candidate 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 10, 页码: 7016-7037
作者:  
Li, Daqiang
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