中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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上海药物研究所 [91]
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Novel imidazo[1,2,4] triazole derivatives: Synthesis, fluorescence, bioactivity for SHP1
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 265, 页码: 15
作者:
Yan, Xue
;
Zhang, Chun
;
Gao, Li-Xin
;
Liu, Min -Min
;
Yang, Yu-Ting
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2024/02/27
Imidazo[124] triazole derivatives
Fluorescence property
SHP1
Bioactivity
Cellular imaging
A novel pterostilbene compound DCZ0825 induces macrophage M1 differentiation and Th1 polarization to exert anti-myeloma and immunomodulatory
期刊论文
OAI收割
INTERNATIONAL IMMUNOPHARMACOLOGY, 2024, 卷号: 127, 页码: 14
作者:
Zhang, Hui
;
Hu, Ke
;
Lu, Yumeng
;
Xu, Zhijian
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2024/03/25
Multiple myeloma
M1 macrophages
Th1 cells
Immunomodulatory
Scintillation Arc from FRB 20220912A
期刊论文
OAI收割
SCIENCE CHINA-PHYSICS MECHANICS & ASTRONOMY, 2024, 卷号: 67, 期号: 1
作者:
Wu, Zi-Wei
;
Main, Robert A.
;
Zhu, Wei-Wei
;
Zhang, Bing
;
Jiang, Peng
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2024/03/29
fast radio burst
scintillation
FRB 20220912A
Structure-based identification of new orally bioavailable BRD9-PROTACs for treating acute myelocytic leukemia
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 262, 页码: 18
作者:
Zhang, Jingyu
;
Duan, Haiting
;
Gui, Renzhao
;
Wu, Mingfei
;
Shen, Liteng
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2023/12/19
Acute myeloid leukemia
Bromodomain-containing protein 9
Proteolysis-targeting chimera
Orally bioavailable
Docking
Exploring the mechanism of the PTP1B inhibitors by molecular dynamics and experimental study
期刊论文
OAI收割
JOURNAL OF MOLECULAR GRAPHICS & MODELLING, 2023, 卷号: 125, 页码: 12
作者:
Zhao, Tian-Tian
;
Hu, Hao-Jie
;
Gao, Li-Xin
;
Zhou, Yu-Bo
;
Zhu, Yun-Long
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2023/10/17
Protein tyrosine phosphatases inhibitors
PTP1B inhibitors
Mechanism study
Molecular dynamics
Pyroxenite-harzburgite sequences in the Dazhuqu ophiolite (Southern Tibet) formed through hydrous melt infiltration and melt-peridotite reaction
期刊论文
OAI收割
CONTRIBUTIONS TO MINERALOGY AND PETROLOGY, 2023, 卷号: 178, 期号: 12, 页码: 30
作者:
Zhang, Zhen-Yu
;
Liu, Chuan-Zhou
;
Liang, Yan
;
Liu, Tong
;
Zhang, Chang
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2024/01/02
Pyroxenite
Melt-rock reaction
Hydrous melt infiltration
The Yarlung-Tsangbo ophiolites
Concentration gradient
A first-in-human phase 1 study of simnotrelvir, a 3CL-like protease inhibitor for treatment of COVID-19, in healthy adult subjects
期刊论文
OAI收割
EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES, 2023, 卷号: 191, 页码: 9
作者:
Yang, Xin-Mei
;
Yang, Yang
;
Yao, Bu-Fan
;
Ye, Pan-Pan
;
Xu, Yan
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2023/12/11
COVID-19
Simnotrelvir
Safety
Pharmacokinetics
Healthy subjects
Thermochemical non-equilibrium flow characteristics of high Mach number inlet in a wide operation range
期刊论文
OAI收割
CHINESE JOURNAL OF AERONAUTICS, 2023, 卷号: 36, 期号: 12, 页码: 164-184
作者:
Dai, Chunliang
  |  
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2024/02/19
Scramjet inlet
Starting ability
Thermochemical
Work performance
n-Alkane
13
C/
12
C indicates differential metabolic controls of fatty lipid chain extension in C
3
and C
4
grasses
期刊论文
OAI收割
PLANT PHYSIOLOGY, 2023, 页码: 5
作者:
Zhao, Yu
;
Yang, Hubiao
;
Yan, Qiulin
;
Zhu, Zhenyu
;
Wang, Bo
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2024/01/26
A neuroimaging biomarker for Individual Brain-Related Abnormalities In Neurodegeneration (IBRAIN): a cross-sectional study
期刊论文
OAI收割
ECLINICALMEDICINE, 2023, 卷号: 65, 页码: 14
作者:
Zhao, Kun
;
Chen, Pindong
;
Alexander-Bloch, Aaron
;
Wei, Yongbin
;
Dyrba, Martin
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2024/02/22
Alzheimer's disease
Neuroimaging biomarker
Multisite
Specific
Longitudinal progression