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浏览/检索结果: 共31条，第1-10条 帮助

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Thiazole-fused thiazoliniums with ketone warheads as covalent inhibitors targeting Cys44 of SARS-CoV-2 3CLpro 期刊论文  OAI收割
CHEMICO-BIOLOGICAL INTERACTIONS, 2025, 卷号: 418, 页码: 12
作者:  Cao, Qizhen;  Zhang, Zhaoqin;  Zhu, Guanghao;  Dong, Sanfeng;  Sun, Xue
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Covalent sortase A inhibitor, α, β-unsaturated aldehydes, prevents Staphylococcus aureus infection 期刊论文  OAI收割
MICROBIAL PATHOGENESIS, 2025, 卷号: 204, 页码: 12
作者:  Wang, Jianchao;  He, Yuan
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Discovery of Covalent and Cell-Active ALKBH5 Inhibitors with Potent Antileukemia Effects In Vivo 期刊论文  OAI收割
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2025, 页码: 9
作者:  Wu, Hengbo;  Lai, Gan-Qiang;  Cheng, Ruixiang;  Huang, Hui;  Wang, Ju
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In vitro and In vivo Drug Metabolism Analysis of BPI-460372-A Covalent TEAD1/3/4 Inhibitor 期刊论文  OAI收割
CURRENT DRUG METABOLISM, 2025, 页码: 15
作者:  Liu, Xiaoyun;  Zhong, Dafang;  Tang, Chongzhuang;  Xu, Xiaofeng;  Lan, Hong
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Identifying a non-conserved site for achieving allosteric covalent inhibition of CECR2 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2025, 页码: 16
作者:  Tang, Cai-ling;  Li, Yuan-qing;  Du, Xi-kun;  Fang, Xiao-xia;  Guang, Yi-man
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Design and development of a series of 4-(piperazin-1-yl)pyrimidines as irreversible menin inhibitors 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 280, 页码: 20
作者:  Luo, Menglan;  Ye, Yunfei;  Tang, Lu;  Kan, Weijuan;  Chen, Lin
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DNA-Encoded Noncanonical Substrate Library for Protease Profiling 期刊论文  OAI收割
CHEMBIOCHEM, 2024, 页码: 12
作者:  Zhang, Huiya;  Xing, Yuyu;  Yang, Yixuan;  Tang, Bixi;  Zong, Zhaoyun
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Identification of benzo[ b ]thiophene-1,1-dioxide derivatives as novel PHGDH covalent inhibitors 期刊论文  OAI收割
BIOORGANIC CHEMISTRY, 2024, 卷号: 146, 页码: 15
作者:  Cao, Xin-Yu;  Li, Xinge;  Wang, Feng;  Duan, Yichen;  Wu, Xingmei
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Discovery of a potent and selective covalent threonine tyrosine kinase (TTK) inhibitor 期刊论文  OAI收割
BIOORGANIC CHEMISTRY, 2024, 卷号: 143, 页码: 16
作者:  Sun, Yaoliang;  Chen, Zhiwen;  Liu, Guobin;  Chen, Xiaoai;  Shi, Zihan
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Discovery of a highly potent NPAS3 heterodimer inhibitor by covalently modifying ARNT 期刊论文  OAI收割
BIOORGANIC CHEMISTRY, 2023, 卷号: 139, 页码: 10
作者:  Li, Peizhuo;  Tian, Yucheng;  Shang, Qinghong;  Tang, Cailing;  Hou, Zeng
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