中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共89条,第1-10条 帮助

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LC-MS/MS assay of fluoropezil and its two major metabolites in human plasma: an application to pharmacokinetic studies 期刊论文  OAI收割
BIOANALYSIS, 2022, 页码: 13
作者:  
Guo, Runcong;  Hu, Jiafeng;  Jing, Jiao;  Liu, Ying;  Li, Jian
  |  收藏  |  浏览/下载:24/0  |  提交时间:2022/08/16
Novel inhibitors of AChE and A0 aggregation with neuroprotective properties as lead compounds for the treatment of Alzheimer's disease 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 235, 页码: 22
作者:  
Liu, Yulin;  Uras, Giuseppe;  Onuwaje, Itse;  Li, Wenlong;  Yao, Hong
  |  收藏  |  浏览/下载:27/0  |  提交时间:2022/08/16
Design, synthesis, in vitro evaluation of a new pyrrolo[1,2-a]thiazolo[5,4-d]pyrimidinone derivatives as cholinesterase inhibitors against Alzheimer's disease 期刊论文  OAI收割
JOURNAL OF HETEROCYCLIC CHEMISTRY, 2022, 页码: 16
作者:  
Zeng, Yan;  Nie, Lifei;  Liu, Liu;  Niu, Chao;  Li, Yi
  |  收藏  |  浏览/下载:26/0  |  提交时间:2022/06/15
Fawcettimine型石松生物碱中间体合成研究 学位论文  OAI收割
2021
作者:  
欧玉飞
  |  收藏  |  浏览/下载:13/0  |  提交时间:2024/03/20
Kinetics-Driven Drug Design Strategy for Next-Generation Acetylcholinesterase Inhibitors to Clinical Candidate 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 4, 页码: 1844-1855
作者:  
Zhou, Yu;  Fu, Yan;  Yin, Wanchao;  Li, Jian;  Wang, Wei
  |  收藏  |  浏览/下载:22/0  |  提交时间:2021/05/24
Discovery and Biological Evaluation of New Selective Acetylcholinesterase Inhibitors with Anti-A beta Aggregation Activity through Molecular Docking-Based Virtual Screening 期刊论文  OAI收割
CHEMICAL & PHARMACEUTICAL BULLETIN, 2020, 卷号: 68, 期号: 2, 页码: 161-166
作者:  
Liu, Guangpu;  Jiao, Yang;  Lin, Yongqiang;  Hao, Haifang;  Dou, Yanli
  |  收藏  |  浏览/下载:22/0  |  提交时间:2020/07/01
Design, synthesis and biological evaluation of novel copper-chelating acetylcholinesterase inhibitors with pyridine and N-benzylpiperidine fragments 期刊论文  OAI收割
BIOORGANIC CHEMISTRY, 2019, 卷号: 93, 页码: 13
作者:  
Zhou, Yeheng;  Sun, Wei;  Peng, Jiale;  Yan, Hui;  Zhang, Li
  |  收藏  |  浏览/下载:35/0  |  提交时间:2020/03/18
Donepezil, a drug for Alzheimer's disease, promotes oligodendrocyte generation and remyelination 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2019, 卷号: 40, 期号: 11, 页码: 1386-1393
作者:  
Cui, Xue;  Guo, Yu-e;  Fang, Jia-hui;  Shi, Chang-jie;  Suo, Na
  |  收藏  |  浏览/下载:32/0  |  提交时间:2020/07/01
Quantitative visualization and detection of acetylcholinesterase activity and its inhibitor based on the oxidation character of ultrathin MnO2 nanosheets. Analytical Methods, Analytical Methods, 2019, 期刊论文  OAI收割
Analytical Methods, 2019, 卷号: 11, 期号: -, 页码: 4931–4938
作者:  
Cai-Hong Li;  Jun-Li Yang;  Wei-Feng Wang;  Won Keun Oh;  Dang Lan Huong
  |  收藏  |  浏览/下载:55/0  |  提交时间:2019/11/11
Discovery of New Selective Butyrylcholinesterase (BChE) Inhibitors with Anti-A beta Aggregation Activity: Structure-Based Virtual Screening, Hit Optimization and Biological Evaluation 期刊论文  OAI收割
MOLECULES, 2019, 卷号: 24, 期号: 14, 页码: 21
作者:  
Jiang, Cheng-Shi;  Ge, Yong-Xi;  Cheng, Zhi-Qiang;  Wang, Yin-Yin;  Tao, Hong-Rui
  |  收藏  |  浏览/下载:20/0  |  提交时间:2020/07/01