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Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
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上海药物研究所 [44]
昆明植物研究所 [11]
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LC-MS/MS assay of fluoropezil and its two major metabolites in human plasma: an application to pharmacokinetic studies
期刊论文
OAI收割
BIOANALYSIS, 2022, 页码: 13
作者:
Guo, Runcong
;
Hu, Jiafeng
;
Jing, Jiao
;
Liu, Ying
;
Li, Jian
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2022/08/16
assay
bioanalysis
DC20
fluoropezil
LC-MS
MS
metabolites
pharmacokinetics
Novel inhibitors of AChE and A0 aggregation with neuroprotective properties as lead compounds for the treatment of Alzheimer's disease
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 235, 页码: 22
作者:
Liu, Yulin
;
Uras, Giuseppe
;
Onuwaje, Itse
;
Li, Wenlong
;
Yao, Hong
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2022/08/16
Alzheimer's disease
Donepezil
Sulfone group
AChE inhibitor
Inhibiting A 0 aggregation
Neuroprotection
Design, synthesis, in vitro evaluation of a new pyrrolo[1,2-a]thiazolo[5,4-d]pyrimidinone derivatives as cholinesterase inhibitors against Alzheimer's disease
期刊论文
OAI收割
JOURNAL OF HETEROCYCLIC CHEMISTRY, 2022, 页码: 16
作者:
Zeng, Yan
;
Nie, Lifei
;
Liu, Liu
;
Niu, Chao
;
Li, Yi
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2022/06/15
Fawcettimine型石松生物碱中间体合成研究
学位论文
OAI收割
2021
作者:
欧玉飞
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2024/03/20
Kinetics-Driven Drug Design Strategy for Next-Generation Acetylcholinesterase Inhibitors to Clinical Candidate
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 4, 页码: 1844-1855
作者:
Zhou, Yu
;
Fu, Yan
;
Yin, Wanchao
;
Li, Jian
;
Wang, Wei
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2021/05/24
Discovery and Biological Evaluation of New Selective Acetylcholinesterase Inhibitors with Anti-A beta Aggregation Activity through Molecular Docking-Based Virtual Screening
期刊论文
OAI收割
CHEMICAL & PHARMACEUTICAL BULLETIN, 2020, 卷号: 68, 期号: 2, 页码: 161-166
作者:
Liu, Guangpu
;
Jiao, Yang
;
Lin, Yongqiang
;
Hao, Haifang
;
Dou, Yanli
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2020/07/01
selective acetylcholinesterase inhibitor
amyloid beta aggregation
neuroprotectant
molecular docking
molecular dynamics simulation
Design, synthesis and biological evaluation of novel copper-chelating acetylcholinesterase inhibitors with pyridine and N-benzylpiperidine fragments
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2019, 卷号: 93, 页码: 13
作者:
Zhou, Yeheng
;
Sun, Wei
;
Peng, Jiale
;
Yan, Hui
;
Zhang, Li
  |  
收藏
  |  
浏览/下载:35/0
  |  
提交时间:2020/03/18
Acetylcholinesterase
Drug design
N-acylhydrazone
Dementia
Copper-chelating
N-Benzylpiperidine
Donepezil, a drug for Alzheimer's disease, promotes oligodendrocyte generation and remyelination
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2019, 卷号: 40, 期号: 11, 页码: 1386-1393
作者:
Cui, Xue
;
Guo, Yu-e
;
Fang, Jia-hui
;
Shi, Chang-jie
;
Suo, Na
  |  
收藏
  |  
浏览/下载:32/0
  |  
提交时间:2020/07/01
donepezil
aricept
oligodendrocyte
oligodendrocyte progenitor cell
differentiation
myelin sheaths
remyelination
CNS demyelinating disorders
multiple sclerosis
Quantitative visualization and detection of acetylcholinesterase activity and its inhibitor based on the oxidation character of ultrathin MnO2 nanosheets. Analytical Methods, Analytical Methods, 2019,
期刊论文
OAI收割
Analytical Methods, 2019, 卷号: 11, 期号: -, 页码: 4931–4938
作者:
Cai-Hong Li
;
Jun-Li Yang
;
Wei-Feng Wang
;
Won Keun Oh
;
Dang Lan Huong
  |  
收藏
  |  
浏览/下载:55/0
  |  
提交时间:2019/11/11
Acetylcholinesterase
AChE–MnO2–OPD
Discovery of New Selective Butyrylcholinesterase (BChE) Inhibitors with Anti-A beta Aggregation Activity: Structure-Based Virtual Screening, Hit Optimization and Biological Evaluation
期刊论文
OAI收割
MOLECULES, 2019, 卷号: 24, 期号: 14, 页码: 21
作者:
Jiang, Cheng-Shi
;
Ge, Yong-Xi
;
Cheng, Zhi-Qiang
;
Wang, Yin-Yin
;
Tao, Hong-Rui
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2020/07/01
selective BChE inhibitor
virtual screening
structural optimization
molecular dynamics
anti-A beta aggregation