中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共155条,第1-10条 帮助

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Structure-Activity Relationships of 2-(Arylthio)benzoic Acid FTO Inhibitors 期刊论文  OAI收割
ISRAEL JOURNAL OF CHEMISTRY, 2024, 页码: 13
作者:  
Yan, Chao;  Zhang, Qian;  Xiao, Pan;  Xie, Xinyun;  Li, Ming
  |  收藏  |  浏览/下载:19/0  |  提交时间:2024/03/25
Structure-based identification of new orally bioavailable BRD9-PROTACs for treating acute myelocytic leukemia 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 262, 页码: 18
作者:  
Zhang, Jingyu;  Duan, Haiting;  Gui, Renzhao;  Wu, Mingfei;  Shen, Liteng
  |  收藏  |  浏览/下载:8/0  |  提交时间:2023/12/19
Discovery of 5-trifluoromethyl-2-aminopyrimidine derivatives as potent dual inhibitors of FLT3 and CHK1 期刊论文  OAI收割
RSC MEDICINAL CHEMISTRY, 2023, 页码: 14
作者:  
Deng, Minjie;  Gao, Yue;  Wang, Peipei;  Du, Wenjing;  Xu, Gaoya
  |  收藏  |  浏览/下载:5/0  |  提交时间:2024/02/19
Design, synthesis and biological evaluation of 2-aminopyrimidine derivatives as potent FLT3 inhibitors 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2023, 卷号: 96, 页码: 5
作者:  
Lian, Xuanmin;  Gao, Yue;  Li, Xuemei;  Wang, Peipei;  Tong, Lexian
  |  收藏  |  浏览/下载:4/0  |  提交时间:2023/12/11
Discovery, Structure-Activity Relationship and In Vitro Anticancer Activity of Small-Molecule Inhibitors of the Protein-Protein Interactions between AF9/ENL and AF4 or DOT1L 期刊论文  OAI收割
CANCERS, 2023, 卷号: 15, 期号: 21, 页码: 28
作者:  
Li, Xin;  Wu, Xiaowei;  Nie, Shenyou;  Zhao, Jidong;  Yao, Yuan
  |  收藏  |  浏览/下载:5/0  |  提交时间:2023/12/19
Chemical Inhibitors Targeting the Oncogenic m6A Modifying Proteins 期刊论文  OAI收割
ACCOUNTS OF CHEMICAL RESEARCH, 2023, 卷号: 56, 期号: 21, 页码: 3010-3022
作者:  
Huang, Yue;  Xia, Wenyang;  Dong, Ze;  Yang, Cai-Guang
  |  收藏  |  浏览/下载:4/0  |  提交时间:2023/12/11
Assessment of the structure-activity relationship and antileukemic activity of diacylpyramide compounds as human ClpP agonists 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 258, 页码: 17
作者:  
Zhang, Ranran;  Wang, Pengyu;  Wei, Bingyan;  Chen, Liang;  Song, Xiaomin
  |  收藏  |  浏览/下载:19/0  |  提交时间:2023/10/17
Rational Design of RNA Demethylase FTO Inhibitors with Enhanced Antileukemia Drug-Like Properties 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 页码: 22
作者:  
Xiao, Pan;  Duan, Zongliang;  Liu, Zeyu;  Chen, Liang;  Zhang, Deyan
  |  收藏  |  浏览/下载:11/0  |  提交时间:2023/10/17
Chloroquine enhances the efficacy of chemotherapy drugs against acute myeloid leukemia by inactivating the autophagy pathway 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2023, 页码: 11
作者:  
Wang, Han-lin;  Li, Jia-nan;  Kan, Wei-juan;  Xu, Gao-ya;  Luo, Guang-hao
  |  收藏  |  浏览/下载:17/0  |  提交时间:2023/10/17
Design, synthesis of novel benzimidazole derivatives as ENL inhibitors suppressing leukemia cells viability via downregulating the expression of MYC 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 248, 页码: 14
作者:  
Guo, Siqi;  Jia, Tongguan;  Xu, Xiaoming;  Yang, Feng;  Xiao, Senhao
  |  收藏  |  浏览/下载:18/0  |  提交时间:2023/04/10