中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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Structure-Activity Relationships of 2-(Arylthio)benzoic Acid FTO Inhibitors
期刊论文
OAI收割
ISRAEL JOURNAL OF CHEMISTRY, 2024, 页码: 13
作者:
Yan, Chao
;
Zhang, Qian
;
Xiao, Pan
;
Xie, Xinyun
;
Li, Ming
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2024/03/25
RNA modification
m(6)A
FTO
anticancer
Discovery of a 1,6-naphthyridin-4-one-based AXL inhibitor with improved pharmacokinetics and enhanced in vivo antitumor efficacy
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 265, 页码: 17
作者:
Lan, Yaohan
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2024/02/27
AXL inhibitor
In vivo antitumor efficacy
6-Naphthyridin-4-one derivatives
Scaffold hopping
Structure-based drug design
pH-responsive nanogels with enhanced antioxidant and antitumor activities on drug delivery and smart drug release
期刊论文
OAI收割
INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES, 2024, 卷号: 257, 页码: 16
作者:
Ma, Bing
;
Li, Qing
;
Mi, Yingqi
;
Zhang, Jingjing
;
Tan, Wenqiang
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2024/01/26
Benzimidazole-chitosan quaternary ammonium
salt
Nanogels
pH-responsive
Antioxidant activity
Antitumor activity
JC-010a, a novel selective SHP2 allosteric inhibitor, overcomes RTK/non-RTK-mediated drug resistance in multiple oncogene-addicted cancers
期刊论文
OAI收割
CANCER LETTERS, 2024, 卷号: 582, 页码: 15
作者:
Lu, Xuxiu
;
Yu, Rilei
;
Li, Zhen
;
Yang, Mengke
;
Dai, Jiajia
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2024/04/07
Acquired resistance
Cancer
NSCLC
JC-010a
SHP2
Extracellular Matrix-Trapped Bioinspired Lipoprotein Prolongs Tumor Retention to Potentiate Antitumor Immunity
期刊论文
OAI收割
ADVANCED MATERIALS, 2024, 页码: 14
作者:
Wu, Yao
;
Li, Yongping
;
Hu, Zixin
;
Li, Yuan
;
Zhang, Shixuan
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2024/02/27
antitumor responses
bioinspired lipoprotein
extracellular matrix
pomalidomide
tumor retention
The promise and challenges of combination therapies with antibody-drug conjugates in solid tumors
期刊论文
OAI收割
JOURNAL OF HEMATOLOGY & ONCOLOGY, 2024, 卷号: 17, 期号: 1, 页码: 32
作者:
Wei, Qing
;
Li, Peijing
;
Yang, Teng
;
Zhu, Jiayu
;
Sun, Lu
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2024/02/27
Antibody-drug conjugate
Solid tumor
Combination therapy
Immunotherapy
Targeted therapy
Enhanced biological activities of coumarin-functionalized polysaccharide derivatives: Chemical modification and activity assessment
期刊论文
OAI收割
INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES, 2023, 卷号: 253, 页码: 13
作者:
Li, Qing
;
Yang, Yunhui
;
Li, Yijian
;
Mi, Yingqi
;
Ma, Xuanxuan
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2023/11/15
Polysaccharide
Chemical modification
Coumarins
Discovery of Dual Function Agents That Exhibit Anticancer Activity via Catastrophic Nicotinamide Adenine Dinucleotide Depletion
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 24, 页码: 16694-16703
作者:
Fu, Yixian
;
Huang, Yahui
;
Zhou, Chenchen
;
Li, Xinge
;
Dong, Guoqiang
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2024/01/26
Dual stimuli-activatable versatile nanoplatform for photodynamic therapy and chemotherapy of triple-negative breast cancer
期刊论文
OAI收割
CHINESE CHEMICAL LETTERS, 2023, 卷号: 34, 期号: 12, 页码: 9
作者:
Xu, Jie
;
Lai, Yi
;
Wang, Fengyang
;
Zou, Zhifeng
;
Pei, Renjun
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2023/12/08
Cancer theranostics
Precise therapy
Combinatorial therapy
Photodynamic therapy
Triple-negative breast cancer
Jin-Fu-An decoction manipulation of macrophage polarization via β-catenin (CTNNB1) synergizes with cisplatin in lung cancer
期刊论文
OAI收割
BIOMEDICINE & PHARMACOTHERAPY, 2023, 卷号: 168, 页码: 17
作者:
Tang, Yang
;
Sun, Zhe
;
Wu, Siqi
;
Zhang, Chengyu
;
Zhang, Yanling
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2024/01/16
Lung cancer
Jin-Fu-An decoction
Tumor-associated macrophages
Macrophage polarization
beta-catenin
Infiltration of cytotoxic T cells