中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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上海药物研究所 [154]
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期刊论文 [334]
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Functional structural domain synthesis of anti-pancreatic carcinoma pectin-like polysaccharide RN1
期刊论文
OAI收割
CARBOHYDRATE POLYMERS, 2024, 卷号: 327, 页码: 11
作者:
Cai, Deqin
;
He, Fei
;
Wu, Shengjie
;
Wang, Zixuan
;
Bian, Ya
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2024/02/19
Polysaccharide
Pectin
Functional structural domain
Pancreatic cancer
Glycan synthesis
RN1
Structure-Activity Relationships of 2-(Arylthio)benzoic Acid FTO Inhibitors
期刊论文
OAI收割
ISRAEL JOURNAL OF CHEMISTRY, 2024, 页码: 13
作者:
Yan, Chao
;
Zhang, Qian
;
Xiao, Pan
;
Xie, Xinyun
;
Li, Ming
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2024/03/25
RNA modification
m(6)A
FTO
anticancer
Discovery and Optimization of WDR5 Inhibitors via Cascade Deoxyribonucleic Acid-Encoded Library Selection Approach
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 2, 页码: 1079-1092
作者:
Qin, Shaozhao
;
Feng, Lijian
;
Zhao, Qingyi
;
Yan, Ziqin
;
Lyu, Xilin
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2024/02/27
Discovery of 5-trifluoromethyl-2-aminopyrimidine derivatives as potent dual inhibitors of FLT3 and CHK1
期刊论文
OAI收割
RSC MEDICINAL CHEMISTRY, 2023, 页码: 14
作者:
Deng, Minjie
;
Gao, Yue
;
Wang, Peipei
  |  
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2024/02/19
Design, synthesis and biological evaluation of 2-aminopyrimidine derivatives as potent FLT3 inhibitors
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2023, 卷号: 96, 页码: 5
作者:
Lian, Xuanmin
;
Gao, Yue
;
Li, Xuemei
;
Wang, Peipei
;
Tong, Lexian
  |  
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2023/12/11
2-aminopyrimidine
FLT3 inhibitors
MV4-11
FLT3 mutations
Identification of [1,2,4]Triazolo[4,3-a]pyrazine PARP1 inhibitors with overcome acquired resistance activities
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 259, 页码: 19
作者:
Wang, Pingyuan
;
Zhu, Wen-Ting
;
Wang, Yajing
;
Song, Shan-Shan
;
Xi, Yong
  |  
收藏
  |  
浏览/下载:57/0
  |  
提交时间:2023/10/17
PARP1 inhibitor
Synthetic lethality
Drug resistance
Anticancer
Structure -activity relationship
The anticancer potential of chemical constituents of Moringa oleifera targeting CDK-2 inhibition in estrogen receptor positive breast cancer using in-silico and in vitro approches
期刊论文
OAI收割
BMC COMPLEMENTARY MEDICINE AND THERAPIES, 2023, 卷号: 23, 期号: 1, 页码: 17
作者:
Sultan, Rida
;
Ahmed, Abrar
;
Wei, Li
;
Saeed, Hamid
;
Islam, Muhammad
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2023/12/19
CDK2
ER+ Breast cancer
Molecular Docking
MM-GBSA
Molecular Dynamic Simulations
MTT assay
Moringa oleifera
Phytoconstituents
Chlorogenic acid
Design, synthesis of auristatins-glucuronide conjugates targeting the β-glucuronidase in tumor microenvironment
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2023, 卷号: 95, 页码: 5
作者:
Wang, Yujie
;
Xu, Keshi
;
Liu, Hongchun
;
Zhang, Wei
;
Hu, Chun
  |  
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2023/12/19
Auristatin E
beta-Glucuronidase
Antiproliferation
Tumor microenvironment
Design, synthesis, and biological evaluation of novel spirocyclic compounds as potential anti-glioblastoma agents
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 258, 页码: 22
作者:
Zhu, Heping
;
Song, Xiaomin
;
Pan, Yihui
;
Li, Ming
;
Chen, Liang
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2023/10/17
Glioblastoma
Spirocyclic compounds
Drug design
Antiproliferation
A zinc-modified
Anemarrhena asphodeloides
polysaccharide complex enhances immune activity
via
the NF-?B and MAPK signaling pathways
期刊论文
OAI收割
INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES, 2023, 卷号: 249, 页码: 12
作者:
Zhang, Shaojie
;
Zhang, Qian
;
Li, Chong
;
Xing, Na
;
Zhou, Pengfei
  |  
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2023/12/08
Anemarrhena asphodeloides Bunge
Zinc modification
Immunoregulatory activity
Zebrafish
NF-kappa B signaling pathway
MAPKs signaling pathway