中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共22条,第1-10条 帮助

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Design, synthesis of auristatins-glucuronide conjugates targeting the β-glucuronidase in tumor microenvironment 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2023, 卷号: 95, 页码: 5
作者:  
Wang, Yujie;  Xu, Keshi;  Liu, Hongchun;  Zhang, Wei;  Hu, Chun
  |  收藏  |  浏览/下载:3/0  |  提交时间:2023/12/19
Discovery of a Novel Bifunctional Steroid Analog, YXG-158, as an Androgen Receptor Degrader and CYP17A1 Inhibitor for the Treatment of Enzalutamide-Resistant Prostate Cancer 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 14, 页码: 9972-9991
作者:  
Wang, Ao;  Luo, Xianggang;  Meng, Xin;  Lu, Zhengyu;  Chen, Kaixian
  |  收藏  |  浏览/下载:9/0  |  提交时间:2023/10/17
Simulating androgen receptor selection in designer yeast 期刊论文  OAI收割
SYNTHETIC AND SYSTEMS BIOTECHNOLOGY, 2022, 卷号: 7
作者:  
Zhang, Haoran;  Zhang, Lu;  Xu, Yipeng;  Chen, Shaoyong;  Ma, Zhenyi
  |  收藏  |  浏览/下载:18/0  |  提交时间:2022/12/23
Gain-Assisted Giant Third-Order Nonlinearity of Epsilon-Near-Zero Multilayered Metamaterials 期刊论文  OAI收割
NANOMATERIALS, 2022, 卷号: 12, 期号: 19
作者:  
Shi, Wenjuan;  Liu, Hongjun;  Wang, Zhaolu
  |  收藏  |  浏览/下载:12/0  |  提交时间:2022/10/25
Design, Synthesis, and Biological Evaluation of Androgen Receptor Degrading and Antagonizing Bifunctional Steroidal Analogs for the Treatment of Advanced Prostate Cancer 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 页码: 22
作者:  
Wang, Ao;  Luo, Xianggang;  Wang, Yawan;  Meng, Xin;  Lu, Zhengyu
  |  收藏  |  浏览/下载:30/0  |  提交时间:2022/11/11
Discovery of a Novel Androgen Receptor Antagonist Manifesting Evidence to Disrupt the Dimerization of the Ligand-Binding Domain via Attenuating the Hydrogen-Bonding Network Between the Two Monomers 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64
作者:  
Fu, Weitao;  Zhang, Minkui;  Liao, Jianing;  Tang, Qing;  Lei, Yixuan
  |  收藏  |  浏览/下载:30/0  |  提交时间:2022/03/21
Polarization-Independent Large Third-Order-Nonlinearity of Orthogonal Nanoantennas Coupled to an Epsilon-Near-Zero Material 期刊论文  OAI收割
NANOMATERIALS, 2021, 卷号: 11, 期号: 12
作者:  
Shi, Wenjuan;  Liu, Hongjun;  Wang, Zhaolu
  |  收藏  |  浏览/下载:71/0  |  提交时间:2022/01/27
Palladium-Catalyzed Tandem Carbonylative Aza-Wacker-Type Cyclization of Nucleophile Tethered Alkene to Access Fused N-Heterocycles 期刊论文  OAI收割
Chinese Journal of Chemistry, 2021, 卷号: 39, 期号: 2, 页码: 317-322
作者:  
Shi Lijun;  Wen Mingshan;  Li Fuwei
  |  收藏  |  浏览/下载:42/0  |  提交时间:2021/11/20
Modulation of photoelectric properties of indium tin oxide thin films via oxygen control, and its application to epsilon-near-zero properties for an infrared absorber 期刊论文  OAI收割
JOURNAL OF APPLIED PHYSICS, 2020, 期号: 18
作者:  
Chai, X;  Zhang, YZ;  Cao, YZ;  Wu, LN;  Ma, JY
  |  收藏  |  浏览/下载:21/0  |  提交时间:2020/12/23
Discovery of Novel Androgen Receptor Ligands by Structure-based Virtual Screening and Bioassays 期刊论文  OAI收割
GENOMICS PROTEOMICS & BIOINFORMATICS, 2019, 卷号: 16, 期号: 6, 页码: 416-427
作者:  
Hou, Tingjun;  Li, Dan;  Chang, Shan;  Xu, Lei;  Sun, Huiyong
  |  收藏  |  浏览/下载:260/0  |  提交时间:2019/06/24