中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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上海药物研究所 [16]
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Design, synthesis, and biological evaluation of novel carbazole derivatives as potent DNMT1 inhibitors with reasonable PK properties
期刊论文
OAI收割
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 2022, 卷号: 37, 期号: 1, 页码: 1537-1555
作者:
Li, Ennian
;
Wang, Kai
;
Zhang, Bei
;
Guo, Siqi
;
Xiao, Senhao
  |  
收藏
  |  
浏览/下载:37/0
  |  
提交时间:2022/08/16
DNMT1 inhibitor
A549 cell lines
HCT116 cell lines
antitumor activity
pharmacokinetic
Pharmacokinetics and Pharmacodynamics of a Depolymerized Glycosaminoglycan from Holothuria fuscopunctata, a Novel Anticoagulant Candidate, in Rats by Bioanalytical Methods
期刊论文
OAI收割
MARINE DRUGS, 2021, 卷号: 19, 期号: 4, 页码: 212
作者:
Liu,Shuang
;
Zhang,Taocui
;
Sun,Huifang
;
Lin,Lisha
;
Gao,Na
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2022/04/02
pharmacokinetics
pharmacodynamics
anticoagulant
fucosylated glycosaminoglycan
dHG-5
method validation
The Nonclinical Pharmacokinetics and Prediction of Human Pharmacokinetics of SPH3127, a Novel Direct Renin Inhibitor
期刊论文
OAI收割
EUROPEAN JOURNAL OF DRUG METABOLISM AND PHARMACOKINETICS, 2020, 卷号: 45, 期号: 1, 页码: 15-26
作者:
Zhang, Leduo
;
Mao, Yu
;
Gao, Zhiwei
;
Chen, Xiaoyan
;
Li, Xin
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2020/07/01
Trained Macrophage Bioreactor for Penetrating Delivery of Fused Antitumor Protein
期刊论文
OAI收割
ACS APPLIED MATERIALS & INTERFACES, 2019, 卷号: 11, 期号: 26, 页码: 23018-23025
作者:
Zhang, Yu
;
Zhang, Yujie
;
Guo, Qin
;
Guo, Zhongyuan
;
Chen, Xinli
  |  
收藏
  |  
浏览/下载:33/0
  |  
提交时间:2020/07/01
macromolecular protein delivery
cell vector
tumor targeting
intratumoral drug distribution
breast cancer therapy
Pyrrole-Hemoglobin Adducts, a More Feasible Potential Biomarker of Pyrrolizidine Alkaloid Exposure
期刊论文
OAI收割
CHEMICAL RESEARCH IN TOXICOLOGY, 2019, 卷号: 32, 期号: 6, 页码: 1027-1039
作者:
Ma, Jiang
;
Ruan, Jianqing
;
Chen, Xinmeng
;
Li, Dongping
;
Yao, Sheng
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2020/07/01
Human pharmacokinetics of ginkgo terpene lactones and impact of carboxylation in blood on their platelet-activating factor antagonistic activity
期刊论文
OAI收割
Acta pharmacologica Sinica, 2018, 卷号: 39, 期号: 12, 页码: 1935-1946
作者:
Liu, Xin-Wei
;
Yang, Jun-Ling
;
Niu, Wei
;
Jia, Wei-Wei
;
Olaleye, Olajide E
  |  
收藏
  |  
浏览/下载:104/0
  |  
提交时间:2019/01/08
Pharmacokinetics and disposition of anlotinib, an oral tyrosine kinase inhibitor, in experimental animal species
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2018, 卷号: 39, 期号: 6, 页码: 1048-1063
作者:
Zhong, Chen-chun
;
Chen, Feng
;
Yang, Jun-ling
;
Jia, Wei-wei
;
Li, Li
  |  
收藏
  |  
浏览/下载:41/0
  |  
提交时间:2019/01/08
anlotinib
tyrosine kinase inhibitor
absorption
distribution
metabolism
excretion
pharmacokinetics
QUANTITATIVE MONITORING OF CEFRADINE IN HUMAN URINE USING A LUMINOL/SULFOBUTYLETHER-beta-CYCLODEXTRIN CHEMILUMINESCENCE SYSTEM
期刊论文
OAI收割
JOURNAL OF APPLIED SPECTROSCOPY, 2018, 卷号: 85, 期号: 2, 页码: 327-334
作者:
Shen, M. X.
;
Tan, X. J.
;
Song, Zh. H.
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2018/09/21
Cefradine
Sulfobutylether-beta-cyclodextrin
Luminol
Chemiluminescence
Flow Injection Technique
Extra Sugar on Vancomycin: New Analogues for Combating Multidrug-Resistant Staphylococcus aureus and Vancomycin-Resistant Enterococci
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 61, 期号: 1, 页码: 286-304
作者:
Guan, Dongliang
;
Chen, Feifei
;
Xiong, Lun
;
Tang, Feng
;
Faridoon
  |  
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2019/01/08
Pharmacokinetics of Florfenicol in the Orange-spotted Grouper, Epinephelus coioides, Following Oral Administration in Warm Seawater
期刊论文
OAI收割
JOURNAL OF THE WORLD AQUACULTURE SOCIETY, 2018, 卷号: 49, 期号: 6, 页码: 1058, 1067
作者:
Ruan, Hui-Ting
;
Dong, Jun-De
;
Luo, Jun-Zhi
;
Feng, Jing-Bin
;
Chen, Hai-Gang
  |  
收藏
  |  
浏览/下载:74/0
  |  
提交时间:2019/08/28
absorption
distribution
elimination
florfenicol
grouper
pharmacokinetics