机构

• 上海药物研究所 [29]
• 中国科学院大学 [3]
• 海洋研究所 [3]
• 武汉病毒研究所 [2]
• 昆明植物研究所 [2]
• 过程工程研究所 [2]
• 更多

采集方式

• OAI收割 [42]
• iSwitch采集 [5]

内容类型

• 期刊论文 [44]
• 学位论文 [3]

发表日期

• 2023 [2]
• 2022 [1]
• 2021 [5]
• 2019 [1]
• 2018 [2]
• 2017 [4]
• 更多

学科主题

• Biochemist... [1]
• Marine & F... [1]

筛选

浏览/检索结果: 共47条，第1-10条 帮助 条数/页： 5101520253035404550556065707580859095100 排序方式： 请选择提交时间升序提交时间降序发表日期升序发表日期降序题名升序题名降序作者升序作者降序 Otilonium Bromide acts as a selective USP28 inhibitor and exhibits cytotoxic activity against multiple human cancer cell lines 期刊论文  OAI收割 BIOCHEMICAL PHARMACOLOGY, 2023, 卷号: 215, 页码: 14 作者:  Xu, Zhuo;  Wang, Hui;  Meng, Qian;  Ding, Yiluan;  Zhu, Mengying   |  收藏  |  浏览/下载：10/0  |  提交时间：2023/10/17 Otilonium Bromide  Deubiquitinase  USP28  Selective inhibitor   Design, synthesis and biological evaluation of salicylanilides as novel allosteric inhibitors of human pancreatic lipase 期刊论文  OAI收割 BIOORGANIC & MEDICINAL CHEMISTRY, 2023, 卷号: 91, 页码: 11 作者:  Zhao, Yitian;  Zhang, Min;  Hou, Xudong;  Han, Jiaxin;  Qin, Xiaoya   |  收藏  |  浏览/下载：11/0  |  提交时间：2023/10/17 Salicylanilide  hPL inhibitor  Structure -activity relationship  Anti -obesity   The discovery of a non-competitive GOT1 inhibitor, hydralazine hydrochloride, via a coupling reaction-based high-throughput screening assay 期刊论文  OAI收割 BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2022, 卷号: 73, 页码: 6 作者:  Wu, Qiqi;  Sun, Zhongya;  Chen, Zhifeng;  Liu, Jingqiu;  Ding, Hong   |  收藏  |  浏览/下载：53/0  |  提交时间：2022/08/30 Glutamate oxaloacetate transaminase 1  Inhibitor  Hydralazine hydrochloride  High -throughput screening   Novel tetrahydrobenzo[b]thiophen-2-yl)urea derivatives as novel alpha-glucosidase inhibitors: Synthesis, kinetics study, molecular docking, and in vivo anti-hyperglycemic evaluation 期刊论文  OAI收割 BIOORGANIC CHEMISTRY, 2021, 卷号: 115, 页码: 17 作者:  Xie, Hong-Xu;  Zhang, Juan;  Li, Yue;  Zhang, Jin-He;  Liu, Shan-Kui   |  收藏  |  浏览/下载：67/0  |  提交时间：2021/11/04 Tetrahydrobenzo[b]thiophen-2-yl)urea  alpha-Glucosidase inhibitors  Non-competitive inhibitor  Molecular docking  Anti-hyperglycaemic activity  Type 2 diabetes   Polyoxypregnanes as safe, potent, and specific ABCB1-inhibitory pro-drugs to overcome multidrug resistance in cancer chemotherapy in vitro and in vivo 期刊论文  OAI收割 ACTA PHARMACEUTICA SINICA B, 2021, 卷号: 11, 期号: 7, 页码: 1885-1902 作者:  Wu, Xu;  Yin, Chun;  Ma, Jiang;  Chai, Stella;  Zhang, Chunyuan   |  收藏  |  浏览/下载：42/0  |  提交时间：2021/11/04 Multidrug resistance  ABCB1  Polyoxypregnane  Combination chemotherapy  Marsdenia tenacissima   Nitrate on localized corrosion of carbon steel and stainless steel in aqueous solutions 期刊论文  OAI收割 ELECTROCHIMICA ACTA, 2021, 卷号: 369, 页码: 13 作者:  Xu, Weichen;  Zhang, Binbin;  Deng, Yu;  Yang, Lihui;  Zhang, Jie   |  收藏  |  浏览/下载：18/0  |  提交时间：2021/04/14 An efficient and concise synthesis of a selective small molecule non-peptide inhibitor of cathepsin L: KGP94 期刊论文  OAI收割 BIOORGANIC CHEMISTRY, 2021, 卷号: 116, 页码: 105317 作者:  Munikishore,Rachakunta;  Wang,Liang-Liang;  Zhang,Shuqun;  Zhao,Qin-Shi;  Zuo,Zhili   |  收藏  |  浏览/下载：46/0  |  提交时间：2022/04/02 Cathepsin L  small-molecule inhibitor  gram-scale synthesis  KGP94  cancer  FUNCTIONALIZED BENZOPHENONE  BIOLOGICAL EVALUATION  TUMOR PROGRESSION  CELL INVASION  EXPRESSION  ANALOGS  SUPPRESSION  DERIVATIVES  ACID   Discovery and characterization of a novel glucose-6-phosphate dehydrogenase (G6PD) inhibitor via high-throughput screening 期刊论文  OAI收割 BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2021, 卷号: 40, 页码: 127905 作者:  Luo, Zhongyuan;  Du, Daohai;  Liu, Yanjun;  Lu, Tian;  Liu, Liping   |  收藏  |  浏览/下载：14/0  |  提交时间：2024/03/21 Glucose-6-phosphate dehydrogenase inhibitor  High-throughput screening  Enzyme kinetics assay  Absorption photometry assay   An Aggregation-induced Emission Probe Based on Host-Guest Inclusion Composed of the Tetraphenylethylene Motif and gamma-Cyclodextrin for the Detection of alpha-Amylase 期刊论文  OAI收割 CHEMISTRY-AN ASIAN JOURNAL, 2019, 卷号: 14, 期号: 6, 页码: 847-852 作者:  Tang, Bo;  Li, Lu;  Shangguan, Huijuan;  Wan, Chuyun;  Chai, Zhaofei   |  收藏  |  浏览/下载：86/0  |  提交时间：2019/06/24 aggregation-induced emission  fluorescence  fluorescent probes  host-guest systems  alpha-amylase   Suppressor of cytokine signalling-2 limits igf1r-mediated regulation of epithelial-mesenchymal transition in lung adenocarcinoma 期刊论文  iSwitch采集 Cell death & disease, 2018, 卷号: 9, 页码: 14 作者:  Zhou, Yue;  Zhang, Zhilei;  Wang, Ning;  Chen, Jizheng;  Zhang, Xu 收藏  |  浏览/下载：77/0  |  提交时间：2019/05/08