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上海药物研究所 [222]
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Discovery, Optimization, and Evaluation of Novel Pyridin-2(1
H
)-one Analogues as Potent TRK Inhibitors for Cancer Treatment
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 2, 页码: 1168-1183
作者:
Xu, Zichao
;
Peng, Xia
;
Zhang, Renjie
;
Ji, Yinchun
;
You, Mengke
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2024/02/27
Rational design of oral delivery nanosystems for hypoglycemic peptides
期刊论文
OAI收割
NANO TODAY, 2023, 卷号: 53, 页码: 19
作者:
Peng, Taoxing
;
Shao, Xinyue
;
Long, Li
;
Liu, Han
;
Song, Wenqin
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2024/01/16
Hypoglycemic peptides
Oral delivery
Mucus penetration
Endocytosis
Intracellular trafficking
Exocytosis
Cyclodextrin MOFs modified dry powder inhalers quadruple bioavailability of luteolin to ameliorate fibrosing interstitial lung disease
期刊论文
OAI收割
INTERNATIONAL JOURNAL OF PHARMACEUTICS, 2023, 卷号: 645, 页码: 9
作者:
Ren, Xiaohong
;
Yang, Ting
;
Zhang, Kaikai
;
Liu, Yujie
;
Wang, Caifen
  |  
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2023/12/08
Fibrosing interstitial lung disease
Luteolin
Cyclodextrin metal -organic frameworks
Dry powder inhalers
Loratadine oral bioavailability enhancement via solid dispersion loaded oro-dispersible films: Formulation, characterization and pharmacokinetics
期刊论文
OAI收割
COLLOIDS AND SURFACES B-BIOINTERFACES, 2023, 卷号: 230
作者:
Islam, Nayyer
;
Khan, Naveed Ullah
;
Razzaq, Anam
;
Menaa, Farid
;
Khan, Zaheer Ullah
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2023/11/17
Loratadine
Solid dispersion
Oro-dispersible film
Bioavailability
Urticaria
Oral Delivery of Gemcitabine-Loaded Glycocholic Acid-Modified Micelles for Cancer Therapy
期刊论文
OAI收割
ACS NANO, 2023, 卷号: 17, 期号: 18, 页码: 18074-18088
作者:
Zang, Wenqing
;
Gao, Duo
;
Yu, Miaorong
;
Long, Manmei
;
Zhang, Zhuan
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2023/12/08
oral delivery
gemcitabine
micelles
glycocholic acid
chemotherapy
Discovery of ARD-1676 as a Highly Potent and Orally Efficacious AR PROTAC Degrader with a Broad Activity against AR Mutants for the Treatment of AR plus Human Prostate Cancer
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 18, 页码: 13280-13303
作者:
Xiang, Weiguo
;
Zhao, Lijie
;
Han, Xin
;
Xu, Tianfeng
;
Kregel, Steven
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2023/12/08
Enhancing the oral bioavailability of poorly water-soluble amisupiride with solid nanodispersion
期刊论文
OAI收割
JOURNAL OF DRUG DELIVERY SCIENCE AND TECHNOLOGY, 2023, 卷号: 86, 页码: 6
作者:
Zhang, Xinyue
;
Li, Jie
;
Rong, Rong
;
Wang, Dangge
;
Wang, Donghai
  |  
收藏
  |  
浏览/下载:65/0
  |  
提交时间:2023/10/17
Solid dispersion
Oral bioavailability
Amisupiride
Nanoparticle
Poorly water-soluble drugs
Magnesium lithospermate B ameliorates diabetic nephropathy by suppressing the uremic toxin formation mediated by gut microbiota
期刊论文
OAI收割
EUROPEAN JOURNAL OF PHARMACOLOGY, 2023, 卷号: 953, 页码: 12
作者:
Zhu, Nanlin
;
Duan, Haonan
;
Feng, Yingying
;
Xu, Wenwei
;
Shen, Jianhua
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2023/10/17
Diabetic nephropathy
Magnesium lithospermate B
Gut microbiota
Uremic toxins
p -Cresyl sulfate metabolism
Pharmacokinetics of fucoidan and low molecular weight fucoidan from Saccharina japonica after oral administration to mice
期刊论文
OAI收割
JOURNAL OF OCEANOLOGY AND LIMNOLOGY, 2023, 页码: 10
作者:
Tan, Jiaojiao
;
Song, Yimin
;
Wang, Jing
;
Wu, Ning
;
Yue, Yang
  |  
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2023/12/13
fucoidan
low molecular weight fucoidan
pharmacokinetics
bioavailability
tissue distribution
Optimization of potent, selective and orally bioavailable biphenyl scaffold as FABP4 inhibitors for anti-inflammation
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 253, 页码: 16
作者:
He, Yulong
;
Li, Shunyi
;
Zhu, Yueyue
;
Wang, Yujie
;
Chen, Yuqi
  |  
收藏
  |  
浏览/下载:62/0
  |  
提交时间:2023/10/17
Structure-activity relationship
FABP4 inhibitor
Biphenyl scaffold
Selectivity
Oral bioavailability
Anti-inflammation