中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共12条,第1-10条 帮助

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Structure-based identification of new orally bioavailable BRD9-PROTACs for treating acute myelocytic leukemia 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 262, 页码: 18
作者:  
Zhang, Jingyu;  Duan, Haiting;  Gui, Renzhao;  Wu, Mingfei;  Shen, Liteng
  |  收藏  |  浏览/下载:8/0  |  提交时间:2023/12/19
Discovery of Highly Potent Nicotinamide Phosphoribosyltransferase Degraders for Efficient Treatment of Ovarian Cancer 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 页码: 15
作者:  
Bi, Kaijian;  Cheng, Junfei;  He, Shipeng;  Fang, Yuxin;  Huang, Min
  |  收藏  |  浏览/下载:14/0  |  提交时间:2023/04/10
Design, synthesis, and biological evaluation of Wee1 kinase degraders 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 243, 页码: 21
作者:  
Zhu, Shulei;  Liu, Jieyu;  Xiao, Donghuai;  Wang, Peipei;  Ma, Jingkun
  |  收藏  |  浏览/下载:34/0  |  提交时间:2022/11/11
Making Protein Degradation Visible: Discovery of Theranostic PROTACs for Detecting and Degrading NAMPT 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 页码: 13
作者:  
Cheng, Junfei;  He, Shipeng;  Xu, Jun;  Huang, Min;  Dong, Guoqiang
  |  收藏  |  浏览/下载:10/0  |  提交时间:2023/04/10
A heterobifunctional molecule recruits cereblon to an RNA scaffold and activates its PROTAC function 期刊论文  OAI收割
CELL REPORTS PHYSICAL SCIENCE, 2022, 卷号: 3, 期号: 10, 页码: 12
作者:  
Xu, Yan;  Fu, Dingqiang;  Yuan, Yi;  Peng, Yan;  Dong, Juan
  |  收藏  |  浏览/下载:15/0  |  提交时间:2023/04/10
Discovery of a potent and selective proteolysis targeting chimera (PROTAC) degrader of NSD3 histone methyltransferase 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 239, 页码: 18
作者:  
Sun, Yaoliang;  Zhang, Ying;  Chen, Xiaoai;  Yu, Aisong;  Du, Wenhao
  |  收藏  |  浏览/下载:41/0  |  提交时间:2022/08/30
Discovery of a Potent and Selective Degrader for USP7 期刊论文  OAI收割
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2022, 卷号: 61, 期号: 33, 页码: e202204395
作者:  
Pei, Yuan;  Fu, Jingfeng;  Shi, Yunkai;  Zhang, Mengmeng;  Luo, Guanghao
  |  收藏  |  浏览/下载:9/0  |  提交时间:2024/03/21
NAMPT-targeting PROTAC promotes antitumor immunity via suppressing myeloid-derived suppressor cell expansion 期刊论文  OAI收割
ACTA PHARMACEUTICA SINICA B, 2022, 卷号: 12, 期号: 6, 页码: 2859-2868
作者:  
Wu, Ying;  Pu, Congying;  Fu, Yixian;  Dong, Guoqiang;  Huang, Min
  |  收藏  |  浏览/下载:6/0  |  提交时间:2024/03/21
The PROTAC selectively degrading Bcl-x(L) represents a novel Hedgehog pathway inhibitor with capacity of combating resistance to Smoothened inhibitors while bone 期刊论文  OAI收割
THERANOSTICS, 2022, 卷号: 12, 期号: 17, 页码: 7476-7490
作者:  
Zhang, Shaoqing;  Chen, Yue;  Xu, Zhongli;  Yang, Jun;  Sun, Renhong
  |  收藏  |  浏览/下载:6/0  |  提交时间:2023/04/10
Discovery of thalidomide-based PROTAC small molecules as the highly efficient SHP2 degraders 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 218, 页码: 14
作者:  
Yang, Xiangbo;  Wang, Zhijia;  Pei, Yuan;  Song, Ning;  Xu, Lei
  |  收藏  |  浏览/下载:28/0  |  提交时间:2021/08/17